IL144761A0 - Solid-state form of celecoxib having enhanced bioavailability - Google Patents

Solid-state form of celecoxib having enhanced bioavailability

Info

Publication number
IL144761A0
IL144761A0 IL14476100A IL14476100A IL144761A0 IL 144761 A0 IL144761 A0 IL 144761A0 IL 14476100 A IL14476100 A IL 14476100A IL 14476100 A IL14476100 A IL 14476100A IL 144761 A0 IL144761 A0 IL 144761A0
Authority
IL
Israel
Prior art keywords
celecoxib
amorphous
drug substance
solid
crystallization
Prior art date
Application number
IL14476100A
Other languages
English (en)
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26865450&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL144761(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of IL144761A0 publication Critical patent/IL144761A0/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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IL14476100A 1999-12-08 2000-12-06 Solid-state form of celecoxib having enhanced bioavailability IL144761A0 (en)

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US16985699P 1999-12-08 1999-12-08
PCT/US2000/032435 WO2001042221A1 (en) 1999-12-08 2000-12-06 Solid-state form of celecoxib having enhanced bioavailability
US09/730,663 US6964978B2 (en) 1999-12-08 2000-12-06 Solid-state form of celecoxib having enhanced bioavailability

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NZ513964A (en) 2004-01-30
HUP0201450A2 (hu) 2002-12-28
AU784572B2 (en) 2006-05-04
CA2362673A1 (en) 2001-06-14
CY1107389T1 (el) 2012-12-19
DK1150959T3 (da) 2008-06-02
DE60038162T2 (de) 2009-02-26
US6964978B2 (en) 2005-11-15
SK12682001A3 (sk) 2002-07-02
US20020006951A1 (en) 2002-01-17
JP2004500358A (ja) 2004-01-08
US20050267190A1 (en) 2005-12-01
PL349223A1 (en) 2002-07-01
EA200100873A1 (ru) 2002-02-28
US7220867B2 (en) 2007-05-22
NO20013855L (no) 2001-10-05
ATE387431T1 (de) 2008-03-15
PL203262B1 (pl) 2009-09-30
US20070202160A1 (en) 2007-08-30
WO2001042221A1 (en) 2001-06-14
EP1150959B1 (en) 2008-02-27
BR0008058A (pt) 2002-03-26
EP1150959A1 (en) 2001-11-07
EA003612B1 (ru) 2003-06-26
ES2299441T3 (es) 2008-06-01
AU1931101A (en) 2001-06-18
DE60038162D1 (de) 2008-04-10
CN1376146B (zh) 2011-04-06
IL144761A (en) 2007-07-24
NO320844B1 (no) 2006-02-06

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