IL135710A0 - Method of synthesis of pyrrole amides - Google Patents

Method of synthesis of pyrrole amides

Info

Publication number
IL135710A0
IL135710A0 IL13571098A IL13571098A IL135710A0 IL 135710 A0 IL135710 A0 IL 135710A0 IL 13571098 A IL13571098 A IL 13571098A IL 13571098 A IL13571098 A IL 13571098A IL 135710 A0 IL135710 A0 IL 135710A0
Authority
IL
Israel
Prior art keywords
synthesis
reaction
followed
pyrrole amides
pyrrole
Prior art date
Application number
IL13571098A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL135710A0 publication Critical patent/IL135710A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/83Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Furan Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Tea And Coffee (AREA)
  • Fats And Perfumes (AREA)
  • Treatment Of Liquids With Adsorbents In General (AREA)
IL13571098A 1997-11-13 1998-10-21 Method of synthesis of pyrrole amides IL135710A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US6542297P 1997-11-13 1997-11-13
US7426698P 1998-02-10 1998-02-10
PCT/IB1998/001672 WO1999025684A1 (fr) 1997-11-13 1998-10-21 Procede de synthese d'amides de pyrrol

Publications (1)

Publication Number Publication Date
IL135710A0 true IL135710A0 (en) 2001-05-20

Family

ID=26745584

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13571098A IL135710A0 (en) 1997-11-13 1998-10-21 Method of synthesis of pyrrole amides

Country Status (35)

Country Link
US (1) US6262272B1 (fr)
EP (1) EP1030838B1 (fr)
JP (1) JP3497469B2 (fr)
KR (1) KR100386722B1 (fr)
CN (2) CN1280566A (fr)
AT (1) ATE231492T1 (fr)
AU (1) AU745788B2 (fr)
BG (1) BG64530B1 (fr)
BR (1) BR9814161A (fr)
CA (1) CA2310095A1 (fr)
CZ (1) CZ20001769A3 (fr)
DE (1) DE69810959T2 (fr)
DK (1) DK1030838T3 (fr)
DZ (1) DZ2651A1 (fr)
EA (1) EA002243B1 (fr)
ES (1) ES2186232T3 (fr)
HR (1) HRP20000298A2 (fr)
HU (1) HUP0100235A3 (fr)
ID (1) ID24135A (fr)
IL (1) IL135710A0 (fr)
IS (1) IS5469A (fr)
MA (1) MA24697A1 (fr)
NO (1) NO20002214L (fr)
NZ (1) NZ503916A (fr)
OA (1) OA11378A (fr)
PA (1) PA8462901A1 (fr)
PL (1) PL340554A1 (fr)
PT (1) PT1030838E (fr)
SK (1) SK6872000A3 (fr)
TN (1) TNSN98204A1 (fr)
TR (1) TR200001343T2 (fr)
TW (1) TW509675B (fr)
UY (1) UY25249A1 (fr)
WO (1) WO1999025684A1 (fr)
YU (1) YU27300A (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EE200200111A (et) * 1999-08-31 2003-06-16 Neurogen Corporation Kondenseerunud pürroolkarboksamiidid: aju GABA-retseptori ligandid
MXPA03001945A (es) * 2000-09-06 2003-09-10 Neurogen Corp Tetrahidroindazoles sustituidos con arilo y su uso como ligandos para el receptor gaba-a.
JP2004515491A (ja) * 2000-12-04 2004-05-27 ファイザー・プロダクツ・インク 縮合ピロールカルボキサミド類の合成
US6852730B2 (en) 2002-02-07 2005-02-08 Neurogen Corporation Substituted fused pyrazolecarboxylic acid arylamides and related compounds
US20080153629A1 (en) * 2004-05-07 2008-06-26 Sullivan Michael J Thick Outer Cover Layer Golf Ball
CN102786458B (zh) * 2012-06-04 2014-02-12 天津渤海职业技术学院 吡咯甲酰胺衍生物、其制备方法和用途
SG11201605915WA (en) * 2014-01-24 2016-08-30 Abbvie Inc Furo-3-carboxamide derivatives and methods of use

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5750702A (en) 1993-10-27 1998-05-12 Neurogen Corporation Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands
US5484944A (en) * 1993-10-27 1996-01-16 Neurogen Corporation Certain fused pyrrolecarboxanilides and their use as GABA brain receptor ligands
US5804686A (en) * 1996-01-19 1998-09-08 Neurogen Corporation fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
WO1997034870A1 (fr) 1996-03-22 1997-09-25 Neurogen Corporation Certains pyrrolecarboxamides fusionnes utilises comme ligands de recepteurs cerebraux gaba

Also Published As

Publication number Publication date
KR20010032063A (ko) 2001-04-16
DE69810959T2 (de) 2003-06-05
ATE231492T1 (de) 2003-02-15
BG104413A (en) 2001-02-28
HUP0100235A2 (hu) 2001-12-28
BG64530B1 (bg) 2005-06-30
US6262272B1 (en) 2001-07-17
AU9363998A (en) 1999-06-07
YU27300A (sh) 2002-10-18
EP1030838A1 (fr) 2000-08-30
UY25249A1 (es) 1999-07-19
EA200000413A1 (ru) 2000-12-25
DK1030838T3 (da) 2003-02-24
TW509675B (en) 2002-11-11
CA2310095A1 (fr) 1999-05-27
SK6872000A3 (en) 2002-02-05
HRP20000298A2 (en) 2001-02-28
EA002243B1 (ru) 2002-02-28
AU745788B2 (en) 2002-03-28
HUP0100235A3 (en) 2002-04-29
JP2001523660A (ja) 2001-11-27
ES2186232T3 (es) 2003-05-01
DZ2651A1 (fr) 2003-03-15
DE69810959D1 (de) 2003-02-27
CN1508129A (zh) 2004-06-30
OA11378A (en) 2004-01-27
PT1030838E (pt) 2003-03-31
JP3497469B2 (ja) 2004-02-16
EP1030838B1 (fr) 2003-01-22
IS5469A (is) 2000-04-26
NO20002214D0 (no) 2000-04-28
NO20002214L (no) 2000-05-12
MA24697A1 (fr) 1999-07-01
WO1999025684A1 (fr) 1999-05-27
NZ503916A (en) 2002-08-28
CZ20001769A3 (cs) 2001-09-12
PL340554A1 (en) 2001-02-12
KR100386722B1 (ko) 2003-06-09
TNSN98204A1 (fr) 2005-03-15
BR9814161A (pt) 2000-09-26
ID24135A (id) 2000-07-06
PA8462901A1 (es) 2000-05-24
CN1280566A (zh) 2001-01-17
TR200001343T2 (tr) 2001-02-21

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