DK1030838T3 - Fremgangsmåde til syntese af pyrrolamider - Google Patents
Fremgangsmåde til syntese af pyrrolamiderInfo
- Publication number
- DK1030838T3 DK1030838T3 DK98946678T DK98946678T DK1030838T3 DK 1030838 T3 DK1030838 T3 DK 1030838T3 DK 98946678 T DK98946678 T DK 98946678T DK 98946678 T DK98946678 T DK 98946678T DK 1030838 T3 DK1030838 T3 DK 1030838T3
- Authority
- DK
- Denmark
- Prior art keywords
- reaction
- pyrrolamides
- synthesis
- followed
- cycloakane
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/83—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6542297P | 1997-11-13 | 1997-11-13 | |
| US7426698P | 1998-02-10 | 1998-02-10 | |
| PCT/IB1998/001672 WO1999025684A1 (en) | 1997-11-13 | 1998-10-21 | Method of synthesis of pyrrole amides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1030838T3 true DK1030838T3 (da) | 2003-02-24 |
Family
ID=26745584
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK98946678T DK1030838T3 (da) | 1997-11-13 | 1998-10-21 | Fremgangsmåde til syntese af pyrrolamider |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US6262272B1 (da) |
| EP (1) | EP1030838B1 (da) |
| JP (1) | JP3497469B2 (da) |
| KR (1) | KR100386722B1 (da) |
| CN (2) | CN1280566A (da) |
| AT (1) | ATE231492T1 (da) |
| AU (1) | AU745788B2 (da) |
| BG (1) | BG64530B1 (da) |
| BR (1) | BR9814161A (da) |
| CA (1) | CA2310095A1 (da) |
| CZ (1) | CZ20001769A3 (da) |
| DE (1) | DE69810959T2 (da) |
| DK (1) | DK1030838T3 (da) |
| DZ (1) | DZ2651A1 (da) |
| EA (1) | EA002243B1 (da) |
| ES (1) | ES2186232T3 (da) |
| HR (1) | HRP20000298A2 (da) |
| HU (1) | HUP0100235A3 (da) |
| ID (1) | ID24135A (da) |
| IL (1) | IL135710A0 (da) |
| IS (1) | IS5469A (da) |
| MA (1) | MA24697A1 (da) |
| NO (1) | NO20002214L (da) |
| NZ (1) | NZ503916A (da) |
| OA (1) | OA11378A (da) |
| PA (1) | PA8462901A1 (da) |
| PL (1) | PL340554A1 (da) |
| PT (1) | PT1030838E (da) |
| SK (1) | SK6872000A3 (da) |
| TN (1) | TNSN98204A1 (da) |
| TR (1) | TR200001343T2 (da) |
| TW (1) | TW509675B (da) |
| UY (1) | UY25249A1 (da) |
| WO (1) | WO1999025684A1 (da) |
| YU (1) | YU27300A (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1210328A1 (en) * | 1999-08-31 | 2002-06-05 | Neurogen Corporation | Fused pyrrolecarboxamides: a new class of gaba brain receptor ligands |
| US6656941B2 (en) | 2000-09-06 | 2003-12-02 | Neurogen Corporation | Aryl substituted tetrahydroindazoles |
| CA2430841A1 (en) * | 2000-12-04 | 2002-06-13 | Pfizer Products Inc. | Synthesis of fused pyrrolecarboxamides |
| JP2005525333A (ja) | 2002-02-07 | 2005-08-25 | ニューロジェン コーポレイション | 置換縮合ピラゾールカルボン酸アリールアミド及び関連化合物 |
| US20080153629A1 (en) * | 2004-05-07 | 2008-06-26 | Sullivan Michael J | Thick Outer Cover Layer Golf Ball |
| CN102786458B (zh) * | 2012-06-04 | 2014-02-12 | 天津渤海职业技术学院 | 吡咯甲酰胺衍生物、其制备方法和用途 |
| CA2937074A1 (en) * | 2014-01-24 | 2015-07-30 | Abbvie Inc. | Furo-3-carboxamide derivatives and methods of use |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5750702A (en) | 1993-10-27 | 1998-05-12 | Neurogen Corporation | Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands |
| US5484944A (en) | 1993-10-27 | 1996-01-16 | Neurogen Corporation | Certain fused pyrrolecarboxanilides and their use as GABA brain receptor ligands |
| US5804686A (en) | 1996-01-19 | 1998-09-08 | Neurogen Corporation | fused pyrrolecarboxamides; a new class of GABA brain receptor ligands |
| WO1997034870A1 (en) | 1996-03-22 | 1997-09-25 | Neurogen Corporation | Certain fused pyrrolecarboxamides as gaba brain receptor ligands |
-
1998
- 1998-10-21 AU AU93639/98A patent/AU745788B2/en not_active Ceased
- 1998-10-21 TR TR2000/01343T patent/TR200001343T2/xx unknown
- 1998-10-21 EA EA200000413A patent/EA002243B1/ru not_active IP Right Cessation
- 1998-10-21 NZ NZ503916A patent/NZ503916A/xx unknown
- 1998-10-21 SK SK687-2000A patent/SK6872000A3/sk unknown
- 1998-10-21 IL IL13571098A patent/IL135710A0/xx unknown
- 1998-10-21 PL PL98340554A patent/PL340554A1/xx not_active Application Discontinuation
- 1998-10-21 ES ES98946678T patent/ES2186232T3/es not_active Expired - Lifetime
- 1998-10-21 DK DK98946678T patent/DK1030838T3/da active
- 1998-10-21 WO PCT/IB1998/001672 patent/WO1999025684A1/en not_active Application Discontinuation
- 1998-10-21 CN CN98811119A patent/CN1280566A/zh active Pending
- 1998-10-21 CZ CZ20001769A patent/CZ20001769A3/cs unknown
- 1998-10-21 EP EP98946678A patent/EP1030838B1/en not_active Expired - Lifetime
- 1998-10-21 CN CNA031594727A patent/CN1508129A/zh active Pending
- 1998-10-21 DE DE69810959T patent/DE69810959T2/de not_active Expired - Fee Related
- 1998-10-21 CA CA002310095A patent/CA2310095A1/en not_active Abandoned
- 1998-10-21 ID IDW20000893A patent/ID24135A/id unknown
- 1998-10-21 PT PT98946678T patent/PT1030838E/pt unknown
- 1998-10-21 HU HU0100235A patent/HUP0100235A3/hu unknown
- 1998-10-21 YU YU27300A patent/YU27300A/sh unknown
- 1998-10-21 BR BR9814161-9A patent/BR9814161A/pt not_active Application Discontinuation
- 1998-10-21 JP JP2000521068A patent/JP3497469B2/ja not_active Expired - Fee Related
- 1998-10-21 AT AT98946678T patent/ATE231492T1/de not_active IP Right Cessation
- 1998-10-21 US US09/403,985 patent/US6262272B1/en not_active Expired - Fee Related
- 1998-10-21 KR KR10-2000-7005185A patent/KR100386722B1/ko not_active IP Right Cessation
- 1998-11-10 PA PA19988462901A patent/PA8462901A1/es unknown
- 1998-11-10 TW TW087118708A patent/TW509675B/zh not_active IP Right Cessation
- 1998-11-11 DZ DZ980261A patent/DZ2651A1/xx active
- 1998-11-11 MA MA25342A patent/MA24697A1/fr unknown
- 1998-11-11 TN TNTNSN98204A patent/TNSN98204A1/fr unknown
- 1998-11-13 UY UY25249A patent/UY25249A1/es not_active IP Right Cessation
-
2000
- 2000-04-26 IS IS5469A patent/IS5469A/is unknown
- 2000-04-28 NO NO20002214A patent/NO20002214L/no unknown
- 2000-05-09 BG BG104413A patent/BG64530B1/bg unknown
- 2000-05-12 HR HR20000298A patent/HRP20000298A2/hr not_active Application Discontinuation
- 2000-05-12 OA OA1200000136A patent/OA11378A/en unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK0861223T3 (da) | Fremgangsmåde til syntese af curcumin-relaterede forbindelser | |
| DK1012144T3 (da) | Fremgangsmåde til fremstilling af (hetero)aromatiske hydroxylaminer | |
| DE69813792T2 (de) | Zwischenprodukte und verfahren zu ihrer herstellung | |
| ATE148100T1 (de) | Verfahren zur herstellung substituierter aromatischer amine | |
| DK1030838T3 (da) | Fremgangsmåde til syntese af pyrrolamider | |
| DK0787124T3 (da) | Fremgangsmåde til fremstilling af substituerede 3-aminobenzonitriler | |
| EA199900821A1 (ru) | Способ получения производных пиразола | |
| DK1097130T3 (da) | Fremgangsmåde til fremstilling af hydroxymethylthiosmörsyre | |
| DE60102008D1 (de) | Herstellungsverfahren für ein bekanntes terazolderivat | |
| WO2002048098A1 (fr) | Arylbis (perfluoroalkylsulfonyl) methane, son sel metallique et leurs procedes de production | |
| DK1099676T3 (da) | Fremgangsmåde til fremstilling af 1,1,4,4-tetramethoxybuten-2 | |
| DK0924195T3 (da) | Fremgangsmåde til fremstilling af aminocyanacetamid | |
| DK167481A (da) | Fremgangsmaade til syntese af substituerede biphenyl-2-carboxaldehyder | |
| DK0971907T3 (da) | Fremgangsmåde til fremstilling af 1,3-disubstituerede 2-nitroguanidiner | |
| DK0934256T3 (da) | Fremgangsmåde til fremstilling af cyanocinnamamider | |
| DK1001929T3 (da) | Fremgangsmåde til fremstilling af 3-cyano-2,4-dihalogen-5-flour-benzoesyrer | |
| BR0115874A (pt) | Sìntese de pirrole-amidas | |
| DK0922686T3 (da) | Fremgangsmåde til fremstilling af ethynylcyclopropan | |
| FR2743066B1 (fr) | Procede de synthese d'un derive aromatique orthodisubstitue par un atome d'halogene autre que le fluor et par un groupe cyano | |
| DK0704438T3 (da) | Fremgangsmåde til fremstilling af 2-cyaniminothiazolidin | |
| DE59908757D1 (de) | Verfahren zur herstellung von atropasäureethylester | |
| BR9909570A (pt) | Processo altamente seletivo, produto preparado pelo mesmo, e, processo para preparar uma quinonaimina a partir de uma hidroxifenilamina correspondente | |
| HUP9900171A2 (hu) | Eljárás azo-metinek és alfa-halogén-acetanilidek előállítására | |
| DK1070082T3 (da) | Fremgangsmåde til fremstilling af 4,4-dimethyl-5alfa-cholesta-8,14,24-trien-3beta-ol og mellemprodukter i fremgangsmåden (I) |