IL134871A - Polymeric derivatives of camptothecins, process for producing such derivatives and pharmaceutical compositions containing them - Google Patents

Polymeric derivatives of camptothecins, process for producing such derivatives and pharmaceutical compositions containing them

Info

Publication number
IL134871A
IL134871A IL13487198A IL13487198A IL134871A IL 134871 A IL134871 A IL 134871A IL 13487198 A IL13487198 A IL 13487198A IL 13487198 A IL13487198 A IL 13487198A IL 134871 A IL134871 A IL 134871A
Authority
IL
Israel
Prior art keywords
derivatives
camptothecins
producing
pharmaceutical compositions
compositions containing
Prior art date
Application number
IL13487198A
Other languages
English (en)
Other versions
IL134871A0 (en
Original Assignee
Pharmacia Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Italia Spa filed Critical Pharmacia Italia Spa
Publication of IL134871A0 publication Critical patent/IL134871A0/xx
Publication of IL134871A publication Critical patent/IL134871A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
IL13487198A 1997-10-03 1998-09-22 Polymeric derivatives of camptothecins, process for producing such derivatives and pharmaceutical compositions containing them IL134871A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9721069.4A GB9721069D0 (en) 1997-10-03 1997-10-03 Polymeric derivatives of camptothecin
PCT/EP1998/006048 WO1999017804A1 (en) 1997-10-03 1998-09-22 Polymeric derivatives of camptothecins

Publications (2)

Publication Number Publication Date
IL134871A0 IL134871A0 (en) 2001-05-20
IL134871A true IL134871A (en) 2005-11-20

Family

ID=10820048

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13487198A IL134871A (en) 1997-10-03 1998-09-22 Polymeric derivatives of camptothecins, process for producing such derivatives and pharmaceutical compositions containing them

Country Status (28)

Country Link
US (1) US6328953B1 (ru)
EP (1) EP1019090B1 (ru)
JP (1) JP2001518521A (ru)
KR (1) KR100559068B1 (ru)
CN (1) CN1154512C (ru)
AR (1) AR013535A1 (ru)
AT (1) ATE259662T1 (ru)
AU (1) AU749321B2 (ru)
BG (1) BG64894B1 (ru)
BR (1) BR9815236A (ru)
CA (1) CA2303097A1 (ru)
DE (1) DE69821783T2 (ru)
DK (1) DK1019090T3 (ru)
EA (1) EA002030B1 (ru)
ES (1) ES2216317T3 (ru)
GB (1) GB9721069D0 (ru)
HK (1) HK1032005A1 (ru)
HU (1) HUP0003690A3 (ru)
IL (1) IL134871A (ru)
MY (1) MY116287A (ru)
NO (1) NO20001628D0 (ru)
NZ (1) NZ503879A (ru)
PL (1) PL191609B1 (ru)
PT (1) PT1019090E (ru)
TW (1) TW564178B (ru)
UA (1) UA70930C2 (ru)
WO (1) WO1999017804A1 (ru)
ZA (1) ZA988923B (ru)

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Also Published As

Publication number Publication date
TW564178B (en) 2003-12-01
BG64894B1 (bg) 2006-08-31
AU749321B2 (en) 2002-06-20
US6328953B1 (en) 2001-12-11
CN1272796A (zh) 2000-11-08
PT1019090E (pt) 2004-05-31
PL191609B1 (pl) 2006-06-30
HUP0003690A3 (en) 2003-08-28
EA002030B1 (ru) 2001-12-24
AR013535A1 (es) 2000-12-27
PL339574A1 (en) 2000-12-18
DK1019090T3 (da) 2004-04-26
DE69821783T2 (de) 2004-12-30
CA2303097A1 (en) 1999-04-15
KR100559068B1 (ko) 2006-03-10
BR9815236A (pt) 2002-07-23
ES2216317T3 (es) 2004-10-16
ZA988923B (en) 1999-04-12
GB9721069D0 (en) 1997-12-03
BG104355A (en) 2001-01-31
HK1032005A1 (en) 2001-07-06
ATE259662T1 (de) 2004-03-15
KR20010015687A (ko) 2001-02-26
AU9627398A (en) 1999-04-27
NO20001628L (no) 2000-03-29
EP1019090B1 (en) 2004-02-18
WO1999017804A1 (en) 1999-04-15
DE69821783D1 (de) 2004-03-25
MY116287A (en) 2003-12-31
CN1154512C (zh) 2004-06-23
IL134871A0 (en) 2001-05-20
EA200000376A1 (ru) 2000-10-30
HUP0003690A2 (hu) 2001-09-28
EP1019090A1 (en) 2000-07-19
NO20001628D0 (no) 2000-03-29
UA70930C2 (ru) 2004-11-15
NZ503879A (en) 2002-03-28
JP2001518521A (ja) 2001-10-16

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Free format text: IN JOURNAL 7/2005 P. 1943 PATENT APPLICATION NO. 134871 CORRECT NAME OF APPLICANT TO - PHARMACIA & UPJOHN S.P.A.

MM9K Patent not in force due to non-payment of renewal fees