IL133800A0 - Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders - Google Patents
Imidazopyrimidines and imidazopyridines for the treatment of neurological disordersInfo
- Publication number
- IL133800A0 IL133800A0 IL13380098A IL13380098A IL133800A0 IL 133800 A0 IL133800 A0 IL 133800A0 IL 13380098 A IL13380098 A IL 13380098A IL 13380098 A IL13380098 A IL 13380098A IL 133800 A0 IL133800 A0 IL 133800A0
- Authority
- IL
- Israel
- Prior art keywords
- imidazopyrimidines
- imidazopyridines
- treatment
- neurological disorders
- neurological
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5162897P | 1997-07-03 | 1997-07-03 | |
US8066598P | 1998-04-03 | 1998-04-03 | |
PCT/US1998/013913 WO1999001454A1 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Publications (1)
Publication Number | Publication Date |
---|---|
IL133800A0 true IL133800A0 (en) | 2001-04-30 |
Family
ID=26729655
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL13380098A IL133800A0 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Country Status (20)
Country | Link |
---|---|
US (3) | US6143743A (pt) |
EP (1) | EP0994877A1 (pt) |
JP (1) | JP2002507996A (pt) |
KR (1) | KR20010014431A (pt) |
CN (1) | CN1268137A (pt) |
AR (1) | AR016307A1 (pt) |
AU (1) | AU746706B2 (pt) |
BR (1) | BR9810508A (pt) |
CA (1) | CA2294117A1 (pt) |
EE (1) | EE04280B1 (pt) |
HR (1) | HRP980375A2 (pt) |
HU (1) | HUP0100179A3 (pt) |
IL (1) | IL133800A0 (pt) |
MY (1) | MY132871A (pt) |
NO (1) | NO316119B1 (pt) |
NZ (1) | NZ502642A (pt) |
PL (1) | PL337888A1 (pt) |
SK (1) | SK179899A3 (pt) |
TW (1) | TW589309B (pt) |
WO (1) | WO1999001454A1 (pt) |
Families Citing this family (74)
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US6365589B1 (en) * | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
SI1140941T1 (en) * | 1998-12-23 | 2005-04-30 | Bristol-Myers Squibb Pharma Company | Nitrogen containing heterobicycles as factor xa inhibitors |
US6271380B1 (en) * | 1998-12-30 | 2001-08-07 | Dupont Pharmaceuticals Company | 1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands |
WO2000059908A2 (en) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6432989B1 (en) | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
AU3264201A (en) * | 1999-12-17 | 2001-06-25 | Du Pont Pharmaceuticals Company | Imidazopyrimidinyl and imidazopyridinyl derivatives |
WO2001058489A1 (fr) * | 2000-02-14 | 2001-08-16 | Japan Tobacco Inc. | Agents prophylactiques/therapeutiques contre le stress postoperatoire |
US20040077605A1 (en) * | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
AR028782A1 (es) * | 2000-07-05 | 2003-05-21 | Taisho Pharmaceutical Co Ltd | Derivados heterociclicos tetrahidropiridino o piperidino |
HUP0301801A2 (hu) | 2000-07-14 | 2003-09-29 | Bristol-Myers Squibb Pharma Company | Imidazo[1,2-a]pirazin-származékok és az ezeket tartalmazó gyógyszerkészítmények |
EP1854798A3 (en) | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
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EE200300342A (et) | 2001-01-26 | 2003-12-15 | Bristol-Myers Squibb Company | Imidasolüüli derivaadid kui kortikotropiini vabastava faktori inhibiitorid, nende saamismeetodid ning kasutamine |
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US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
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HUP0401292A3 (en) | 2001-04-27 | 2011-01-28 | Eisai R & D Man Co | Pyrazolo[1,5-a]pyridines, pharmaceutical compositions containing the same and process for preparation thereof |
PL366577A1 (en) | 2001-05-14 | 2005-02-07 | Bristol-Myers Squibb Pharma Company | Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands |
AU2002354575A1 (en) | 2001-07-12 | 2003-01-29 | Bristol-Myers Squibb Pharma Company | Tetrahydropurinones as corticotropin releasing factor |
WO2003006015A1 (en) | 2001-07-13 | 2003-01-23 | Bristol-Myers Squibb Pharma Company | Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands |
US20070129334A1 (en) * | 2001-10-30 | 2007-06-07 | Conforma Therapeutics Corporation | Orally Active Purine-Based Inhibitors of Heat Shock Protein 90 |
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-
1998
- 1998-07-02 WO PCT/US1998/013913 patent/WO1999001454A1/en not_active Application Discontinuation
- 1998-07-02 JP JP50744099A patent/JP2002507996A/ja active Pending
- 1998-07-02 AU AU81819/98A patent/AU746706B2/en not_active Ceased
- 1998-07-02 HR HR60/080,665A patent/HRP980375A2/hr not_active Application Discontinuation
- 1998-07-02 CN CN98808584A patent/CN1268137A/zh active Pending
- 1998-07-02 HU HU0100179A patent/HUP0100179A3/hu unknown
- 1998-07-02 EE EEP199900607A patent/EE04280B1/xx not_active IP Right Cessation
- 1998-07-02 EP EP98931795A patent/EP0994877A1/en not_active Withdrawn
- 1998-07-02 NZ NZ502642A patent/NZ502642A/en unknown
- 1998-07-02 US US09/109,877 patent/US6143743A/en not_active Expired - Lifetime
- 1998-07-02 BR BR9810508-6A patent/BR9810508A/pt not_active IP Right Cessation
- 1998-07-02 KR KR1019997012619A patent/KR20010014431A/ko not_active Application Discontinuation
- 1998-07-02 SK SK1798-99A patent/SK179899A3/sk unknown
- 1998-07-02 MY MYPI98003027A patent/MY132871A/en unknown
- 1998-07-02 PL PL98337888A patent/PL337888A1/xx unknown
- 1998-07-02 IL IL13380098A patent/IL133800A0/xx unknown
- 1998-07-02 CA CA002294117A patent/CA2294117A1/en not_active Abandoned
- 1998-07-02 TW TW087110857A patent/TW589309B/zh active
- 1998-07-03 AR ARP980103234A patent/AR016307A1/es not_active Application Discontinuation
- 1998-12-10 US US09/208,778 patent/US6362180B1/en not_active Expired - Lifetime
-
1999
- 1999-12-27 NO NO19996483A patent/NO316119B1/no not_active IP Right Cessation
-
2001
- 2001-11-07 US US10/053,475 patent/US6642230B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
US20030114468A1 (en) | 2003-06-19 |
AU8181998A (en) | 1999-01-25 |
US6362180B1 (en) | 2002-03-26 |
JP2002507996A (ja) | 2002-03-12 |
HRP980375A2 (en) | 1999-04-30 |
KR20010014431A (ko) | 2001-02-26 |
TW589309B (en) | 2004-06-01 |
CA2294117A1 (en) | 1999-01-14 |
NO996483D0 (no) | 1999-12-27 |
US6642230B2 (en) | 2003-11-04 |
WO1999001454A1 (en) | 1999-01-14 |
HUP0100179A2 (hu) | 2001-11-28 |
EE04280B1 (et) | 2004-04-15 |
HUP0100179A3 (en) | 2002-12-28 |
CN1268137A (zh) | 2000-09-27 |
AR016307A1 (es) | 2001-07-04 |
AU746706B2 (en) | 2002-05-02 |
NO996483L (no) | 2000-03-02 |
US6143743A (en) | 2000-11-07 |
EP0994877A1 (en) | 2000-04-26 |
MY132871A (en) | 2007-10-31 |
EE9900607A (et) | 2000-08-15 |
SK179899A3 (en) | 2001-12-03 |
PL337888A1 (en) | 2000-09-11 |
NZ502642A (en) | 2002-06-28 |
NO316119B1 (no) | 2003-12-15 |
BR9810508A (pt) | 2000-09-05 |
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