IL128504A - 2-HETEROARYL-N-PHENYL (ALKYL) THIENO [2,3-d] PYRIMIDIN-4-AMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

2-HETEROARYL-N-PHENYL (ALKYL) THIENO [2,3-d] PYRIMIDIN-4-AMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
IL128504A
IL128504A IL12850497A IL12850497A IL128504A IL 128504 A IL128504 A IL 128504A IL 12850497 A IL12850497 A IL 12850497A IL 12850497 A IL12850497 A IL 12850497A IL 128504 A IL128504 A IL 128504A
Authority
IL
Israel
Prior art keywords
thieno
pyrimidin
heteroaryl
phenyl
alkyl
Prior art date
Application number
IL12850497A
Other languages
English (en)
Other versions
IL128504A0 (en
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of IL128504A0 publication Critical patent/IL128504A0/xx
Publication of IL128504A publication Critical patent/IL128504A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL12850497A 1996-08-12 1997-07-30 2-HETEROARYL-N-PHENYL (ALKYL) THIENO [2,3-d] PYRIMIDIN-4-AMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IL128504A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19632423A DE19632423A1 (de) 1996-08-12 1996-08-12 Thienopyrimidine
PCT/EP1997/004139 WO1998006722A1 (de) 1996-08-12 1997-07-30 Thienopyrimidine

Publications (2)

Publication Number Publication Date
IL128504A0 IL128504A0 (en) 2000-01-31
IL128504A true IL128504A (en) 2003-01-12

Family

ID=7802392

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12850497A IL128504A (en) 1996-08-12 1997-07-30 2-HETEROARYL-N-PHENYL (ALKYL) THIENO [2,3-d] PYRIMIDIN-4-AMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (28)

Country Link
US (1) US6110920A (cg-RX-API-DMAC10.html)
EP (1) EP0920431B1 (cg-RX-API-DMAC10.html)
JP (1) JP4405593B2 (cg-RX-API-DMAC10.html)
KR (1) KR100502271B1 (cg-RX-API-DMAC10.html)
CN (1) CN1081638C (cg-RX-API-DMAC10.html)
AR (1) AR009052A1 (cg-RX-API-DMAC10.html)
AT (1) ATE233265T1 (cg-RX-API-DMAC10.html)
AU (1) AU725227B2 (cg-RX-API-DMAC10.html)
BR (1) BR9711062A (cg-RX-API-DMAC10.html)
CA (1) CA2263561C (cg-RX-API-DMAC10.html)
CZ (1) CZ287772B6 (cg-RX-API-DMAC10.html)
DE (2) DE19632423A1 (cg-RX-API-DMAC10.html)
DK (1) DK0920431T3 (cg-RX-API-DMAC10.html)
ES (1) ES2191192T3 (cg-RX-API-DMAC10.html)
HU (1) HUP0001607A3 (cg-RX-API-DMAC10.html)
IL (1) IL128504A (cg-RX-API-DMAC10.html)
NO (1) NO990643D0 (cg-RX-API-DMAC10.html)
NZ (1) NZ334600A (cg-RX-API-DMAC10.html)
PL (1) PL190174B1 (cg-RX-API-DMAC10.html)
PT (1) PT920431E (cg-RX-API-DMAC10.html)
RU (1) RU2199541C2 (cg-RX-API-DMAC10.html)
SI (1) SI0920431T1 (cg-RX-API-DMAC10.html)
SK (1) SK282823B6 (cg-RX-API-DMAC10.html)
TR (1) TR199900308T2 (cg-RX-API-DMAC10.html)
TW (1) TW359672B (cg-RX-API-DMAC10.html)
UA (1) UA55421C2 (cg-RX-API-DMAC10.html)
WO (1) WO1998006722A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA977156B (cg-RX-API-DMAC10.html)

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Also Published As

Publication number Publication date
SK16499A3 (en) 1999-06-11
IL128504A0 (en) 2000-01-31
PT920431E (pt) 2003-07-31
PL190174B1 (pl) 2005-11-30
CN1081638C (zh) 2002-03-27
TR199900308T2 (xx) 1999-04-21
KR100502271B1 (ko) 2005-07-22
NO990643L (no) 1999-02-11
HUP0001607A3 (en) 2002-09-30
CN1227560A (zh) 1999-09-01
SI0920431T1 (en) 2003-08-31
DE19632423A1 (de) 1998-02-19
AU4203597A (en) 1998-03-06
HUP0001607A2 (hu) 2000-10-28
EP0920431B1 (de) 2003-02-26
ES2191192T3 (es) 2003-09-01
AR009052A1 (es) 2000-03-08
CZ287772B6 (en) 2001-01-17
US6110920A (en) 2000-08-29
DE59709404D1 (en) 2003-04-03
AU725227B2 (en) 2000-10-12
DK0920431T3 (da) 2003-06-02
EP0920431A1 (de) 1999-06-09
HK1021731A1 (en) 2000-06-30
WO1998006722A1 (de) 1998-02-19
KR20000029932A (ko) 2000-05-25
BR9711062A (pt) 1999-08-17
CA2263561A1 (en) 1998-02-19
SK282823B6 (sk) 2002-12-03
CA2263561C (en) 2007-02-20
JP4405593B2 (ja) 2010-01-27
ZA977156B (en) 1998-02-19
JP2000516223A (ja) 2000-12-05
NZ334600A (en) 2000-07-28
PL331538A1 (en) 1999-07-19
NO990643D0 (no) 1999-02-11
CZ44899A3 (cs) 1999-05-12
TW359672B (en) 1999-06-01
ATE233265T1 (de) 2003-03-15
RU2199541C2 (ru) 2003-02-27
UA55421C2 (uk) 2003-04-15

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