IL108979A - A83543 Compounds process for production thereof pesticidal compositions containing them and intermediates therefor - Google Patents
A83543 Compounds process for production thereof pesticidal compositions containing them and intermediates thereforInfo
- Publication number
- IL108979A IL108979A IL10897994A IL10897994A IL108979A IL 108979 A IL108979 A IL 108979A IL 10897994 A IL10897994 A IL 10897994A IL 10897994 A IL10897994 A IL 10897994A IL 108979 A IL108979 A IL 108979A
- Authority
- IL
- Israel
- Prior art keywords
- compound
- formula
- nrrl
- hydrogen
- compounds
- Prior art date
Links
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- 238000000034 method Methods 0.000 title claims abstract description 54
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- 239000001257 hydrogen Substances 0.000 claims description 31
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- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
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-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P19/00—Preparation of compounds containing saccharide radicals
- C12P19/44—Preparation of O-glycosides, e.g. glucosides
- C12P19/60—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
- C12P19/62—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12R—INDEXING SCHEME ASSOCIATED WITH SUBCLASSES C12C - C12Q, RELATING TO MICROORGANISMS
- C12R2001/00—Microorganisms ; Processes using microorganisms
- C12R2001/01—Bacteria or Actinomycetales ; using bacteria or Actinomycetales
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S424/00—Drug, bio-affecting and body treating compositions
- Y10S424/08—Systemic pesticides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S424/00—Drug, bio-affecting and body treating compositions
- Y10S424/10—Insect repellent
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S435/00—Chemistry: molecular biology and microbiology
- Y10S435/8215—Microorganisms
- Y10S435/822—Microorganisms using bacteria or actinomycetales
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- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- General Health & Medical Sciences (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Engineering & Computer Science (AREA)
- Microbiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Dentistry (AREA)
- Virology (AREA)
- Biomedical Technology (AREA)
- Environmental Sciences (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Manufacturing Of Printed Wiring (AREA)
- Devices That Are Associated With Refrigeration Equipment (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Saccharide Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3052293A | 1993-03-12 | 1993-03-12 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL108979A0 IL108979A0 (en) | 1994-06-24 |
| IL108979A true IL108979A (en) | 1999-09-22 |
Family
ID=21854619
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL10897994A IL108979A (en) | 1993-03-12 | 1994-03-15 | A83543 Compounds process for production thereof pesticidal compositions containing them and intermediates therefor |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US5840861A (mo) |
| EP (1) | EP0688332B1 (mo) |
| JP (1) | JP4258575B2 (mo) |
| AT (1) | ATE150758T1 (mo) |
| AU (1) | AU685107B2 (mo) |
| BR (1) | BR9406587A (mo) |
| CA (1) | CA2156194C (mo) |
| DE (1) | DE69402308T2 (mo) |
| DK (1) | DK0688332T3 (mo) |
| ES (1) | ES2099604T3 (mo) |
| FI (1) | FI107266B (mo) |
| IL (1) | IL108979A (mo) |
| TW (1) | TW294672B (mo) |
| WO (1) | WO1994020518A1 (mo) |
Families Citing this family (59)
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|---|---|---|---|---|
| AU711185B2 (en) * | 1995-06-14 | 1999-10-07 | Dow Agrosciences Llc | Synthetic modification to spinosyn compounds |
| DE19823397B4 (de) | 1998-05-26 | 2011-07-28 | Bayer CropScience AG, 40789 | Verwendung von Spinosynen zum Einsatz als Bodeninsektizide |
| DE19823396A1 (de) * | 1998-05-26 | 1999-12-02 | Bayer Ag | Synergistische insektizide Mischungen |
| CA2337789C (en) * | 1998-07-02 | 2010-10-26 | Eli Lilly And Company | Formulations for controlling human lice |
| US6927210B1 (en) | 1999-08-12 | 2005-08-09 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
| US6933318B1 (en) | 1999-08-12 | 2005-08-23 | Eli Lilly And Company | Topical organic ectoparasiticidal formulations |
| EP1207756B1 (en) | 1999-08-12 | 2006-04-26 | Eli Lilly And Company | Use of spinosad or a formulation comprising spinosad |
| WO2001011962A1 (en) * | 1999-08-12 | 2001-02-22 | Eli Lilly And Company | Topical treatment for insect pests in companion animals |
| JP2003508050A (ja) | 1999-08-27 | 2003-03-04 | バイエル アクチェンゲゼルシャフト | スピノシン生合成の酵素活性をコードする核酸 |
| UA71997C2 (en) * | 1999-09-13 | 2005-01-17 | Dow Agrosciences Llc | Pesticide macrolide, a method for the preparation thereof, strain saccharopolyspora producing macrolide and a mixture based thereon and a method for controlling insecticides and acaricides |
| AUPQ441699A0 (en) | 1999-12-02 | 2000-01-06 | Eli Lilly And Company | Pour-on formulations |
| AUPQ634300A0 (en) * | 2000-03-20 | 2000-04-15 | Eli Lilly And Company | Synergistic formulations |
| US6585990B1 (en) | 2001-03-05 | 2003-07-01 | Dow Agrosciences, Llc | Compositions and devices using a spinosyn compound for control of insects |
| ES2496940T3 (es) * | 2001-03-21 | 2014-09-22 | Dow Agrosciences, Llc | Derivados plaguicidas de las espinosinas |
| WO2002079184A1 (de) * | 2001-03-29 | 2002-10-10 | Bayer Cropscience Ag | Zwischenverbindungen zur herstellung von spinosynen |
| AR033022A1 (es) | 2001-03-30 | 2003-12-03 | Dow Agrosciences Llc | Genes biosinteticos para la produccion de insecticida de butenilespinosina |
| US6727228B2 (en) * | 2001-04-25 | 2004-04-27 | Johnson & Johnson Consumer Companies, Inc. | Pediculicidal and ovacidal treatment compositions and methods for killing head lice and their eggs |
| DE10135550A1 (de) * | 2001-07-20 | 2003-01-30 | Bayer Cropscience Ag | Verfahren zum Herstellen von neuen Spinosyn-Derivaten |
| IL160619A0 (en) | 2001-09-17 | 2004-07-25 | Lilly Co Eli | Pesticidal formulations pesticidal formulations |
| TWI330183B (mo) * | 2001-10-22 | 2010-09-11 | Eisai R&D Man Co Ltd | |
| EP1492404B1 (en) | 2002-02-19 | 2011-12-28 | Dow AgroSciences LLC | Novel spinosyn-producing polyketide synthases |
| US20070049631A1 (en) * | 2003-11-04 | 2007-03-01 | Akzo Nobel N.V. | Ectoparasiticidal formulations of spinosyms and azole pesticides |
| EP1849363A1 (en) * | 2006-03-09 | 2007-10-31 | Cheminova A/S | Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin |
| AU2009214930B2 (en) * | 2008-02-12 | 2014-04-10 | Corteva Agriscience Llc | Pesticidal compositions |
| CN101560477B (zh) * | 2008-04-16 | 2012-04-25 | 上海医药工业研究院 | 发酵多杀菌素产生菌的培养基 |
| US9514283B2 (en) | 2008-07-09 | 2016-12-06 | Baxter International Inc. | Dialysis system having inventory management including online dextrose mixing |
| CN102202506B (zh) | 2008-09-22 | 2015-07-29 | 克里斯廷·克里蒂考 | 刺糖多孢菌素防污组合物、其使用方法、以及受到保护而免于附着污损生物的制品 |
| US8268975B2 (en) | 2009-04-03 | 2012-09-18 | Dow Agrosciences Llc | Demulsification compositions, systems and methods for demulsifying and separating aqueous emulsions |
| TW201041510A (en) | 2009-04-30 | 2010-12-01 | Dow Agrosciences Llc | Pesticide compositions exhibiting enhanced activity |
| TW201041508A (en) | 2009-04-30 | 2010-12-01 | Dow Agrosciences Llc | Pesticide compositions exhibiting enhanced activity |
| TW201041509A (en) | 2009-04-30 | 2010-12-01 | Dow Agrosciences Llc | Pesticide compositions exhibiting enhanced activity |
| TW201041507A (en) | 2009-04-30 | 2010-12-01 | Dow Agrosciences Llc | Pesticide compositions exhibiting enhanced activity and methods for preparing same |
| WO2010150100A1 (en) | 2009-06-24 | 2010-12-29 | Entarco Sa | The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer |
| WO2011143291A1 (en) | 2010-05-11 | 2011-11-17 | Dow Agrosciences Llc | Spnk strains |
| US20160184340A1 (en) | 2010-12-22 | 2016-06-30 | Christine Kritikou | The use of spinosyns and spinosyn compositions as local anesthetics and as antiarrhythmic agents |
| CN103402357B (zh) * | 2010-12-29 | 2016-12-07 | 陶氏益农公司 | 防治昆虫的方法 |
| EP2520653B1 (en) | 2011-05-03 | 2017-03-29 | Dow AgroSciences LLC | Integration of genes into the chromosome of saccharopolyspora spinosa |
| US8741603B2 (en) | 2011-05-03 | 2014-06-03 | Agrigenetics Inc. | Enhancing spinosyn production with oxygen binding proteins |
| US9404107B2 (en) | 2011-05-03 | 2016-08-02 | Dow Agrosciences Llc | Integration of genes into the chromosome of Saccharopolyspora spinosa |
| US9631195B2 (en) | 2011-12-28 | 2017-04-25 | Dow Agrosciences Llc | Identification and characterization of the spinactin biosysnthesis gene cluster from spinosyn producing saccharopolyspora spinosa |
| CN110251509A (zh) | 2012-02-06 | 2019-09-20 | 勃林格殷格翰动物保健美国公司 | 包含全身性地起作用的活性剂的杀寄生虫口服兽用组合物、方法及其用途 |
| JO3626B1 (ar) | 2012-02-23 | 2020-08-27 | Merial Inc | تركيبات موضعية تحتوي على فيبرونيل و بيرميثرين و طرق استخدامها |
| AU2012233000B2 (en) * | 2012-09-28 | 2016-01-21 | Elanco New Zealand | Ectoparasitic Treatment Method and Composition |
| AU2015247463B2 (en) | 2014-04-17 | 2018-03-29 | Basf, Se | Use of malononitrile compounds for protecting animals from parasites |
| JP6616786B2 (ja) | 2014-05-19 | 2019-12-04 | メリアル インコーポレイテッド | 駆虫性化合物 |
| CA2952857A1 (en) | 2014-06-19 | 2015-12-23 | Merial, Inc. | Parasiticidal compositions comprising indole derivatives, methods and uses thereof |
| US10306887B2 (en) | 2014-08-05 | 2019-06-04 | The Board Of Regents Of The University Of Texas Systems | Composition and methods for modulation of the octopamine receptor and its homologs |
| UY36570A (es) | 2015-02-26 | 2016-10-31 | Merial Inc | Formulaciones inyectables de acción prolongada que comprenden un agente activo isoxazolina, métodos y usos de las mismas |
| BR112017024773A2 (pt) | 2015-05-20 | 2018-11-06 | Merial, Inc. | compostos depsipeptídeos anti-helmínticos |
| WO2018039508A1 (en) | 2016-08-25 | 2018-03-01 | Merial, Inc. | Method for reducing unwanted effects in parasiticidal treatments |
| BR112019009977A2 (pt) | 2016-11-16 | 2019-08-27 | Boehringer Ingelheim Animal Health Usa Inc | compostos depsipeptídicos anti-helmínticos |
| CN110914425B (zh) | 2017-06-06 | 2024-06-25 | 齐默尔根公司 | 用于改良刺糖多孢菌的高通量(htp)基因组工程改造平台 |
| KR20250044476A (ko) | 2018-07-09 | 2025-03-31 | 베링거잉겔하임베트메디카게엠베하 | 구충성 헤테로시클릭 화합물 |
| WO2020023943A1 (en) | 2018-07-27 | 2020-01-30 | Aperta Biosciences, Llc | Spinosyn formulations for treatment of demodex-induced ocular and facial conditions |
| CN113260419A (zh) | 2018-11-20 | 2021-08-13 | 勃林格殷格翰动物保健美国公司 | 吲唑基氰基乙基氨基化合物、其组合物、其制备方法和其使用方法 |
| WO2020150032A1 (en) | 2019-01-16 | 2020-07-23 | Boehringer Ingelheim Animal Health USA Inc. | Topical compositions comprising a neonicotinoid and a macrocyclic lactone, methods and uses thereof |
| KR20220002890A (ko) | 2019-03-19 | 2022-01-07 | 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 | 구충성 아자-벤조티오펜 및 아자-벤조푸란 화합물 |
| CN110734467B (zh) * | 2019-09-10 | 2021-08-27 | 北大方正集团有限公司 | 一种从发酵液中提取纯化多杀霉素的方法 |
| KR20230028268A (ko) | 2020-05-29 | 2023-02-28 | 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 | 구충성 헤테로시클릭 화합물 |
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| US3725385A (en) * | 1970-11-02 | 1973-04-03 | Abbott Lab | Process for the demethylation of 3-amino macrolides |
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| JPS62226925A (ja) * | 1986-03-28 | 1987-10-05 | Ss Pharmaceut Co Ltd | 抗マイコプラズマ剤 |
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-
1994
- 1994-03-11 ES ES94912774T patent/ES2099604T3/es not_active Expired - Lifetime
- 1994-03-11 WO PCT/US1994/002674 patent/WO1994020518A1/en not_active Ceased
- 1994-03-11 CA CA002156194A patent/CA2156194C/en not_active Expired - Lifetime
- 1994-03-11 JP JP52034194A patent/JP4258575B2/ja not_active Expired - Lifetime
- 1994-03-11 EP EP94912774A patent/EP0688332B1/en not_active Expired - Lifetime
- 1994-03-11 AU AU65187/94A patent/AU685107B2/en not_active Expired
- 1994-03-11 AT AT94912774T patent/ATE150758T1/de active
- 1994-03-11 BR BR9406587A patent/BR9406587A/pt not_active IP Right Cessation
- 1994-03-11 DE DE69402308T patent/DE69402308T2/de not_active Expired - Lifetime
- 1994-03-11 DK DK94912774.0T patent/DK0688332T3/da active
- 1994-03-15 IL IL10897994A patent/IL108979A/en not_active IP Right Cessation
- 1994-03-21 TW TW083102553A patent/TW294672B/zh not_active IP Right Cessation
-
1995
- 1995-02-08 US US08/385,497 patent/US5840861A/en not_active Expired - Lifetime
- 1995-06-07 US US08/483,440 patent/US5670486A/en not_active Expired - Lifetime
- 1995-06-07 US US08/474,026 patent/US5670364A/en not_active Expired - Lifetime
- 1995-09-11 FI FI954246A patent/FI107266B/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| WO1994020518A1 (en) | 1994-09-15 |
| IL108979A0 (en) | 1994-06-24 |
| CA2156194A1 (en) | 1994-09-15 |
| JPH08507533A (ja) | 1996-08-13 |
| DE69402308T2 (de) | 1997-10-23 |
| FI954246A0 (fi) | 1995-09-11 |
| DE69402308D1 (de) | 1997-04-30 |
| US5840861A (en) | 1998-11-24 |
| ATE150758T1 (de) | 1997-04-15 |
| JP4258575B2 (ja) | 2009-04-30 |
| BR9406587A (pt) | 1996-01-02 |
| FI107266B (fi) | 2001-06-29 |
| TW294672B (mo) | 1997-01-01 |
| CA2156194C (en) | 2008-01-08 |
| AU6518794A (en) | 1994-09-26 |
| ES2099604T3 (es) | 1997-05-16 |
| EP0688332B1 (en) | 1997-03-26 |
| US5670364A (en) | 1997-09-23 |
| US5670486A (en) | 1997-09-23 |
| AU685107B2 (en) | 1998-01-15 |
| EP0688332A1 (en) | 1995-12-27 |
| FI954246L (fi) | 1995-09-11 |
| DK0688332T3 (da) | 1997-10-13 |
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| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| EXP | Patent expired |