IL107331A - History of androstane converted to 61st place in a quarterly ammonium group, pharmaceutical mixtures containing them and process for their preparation - Google Patents

History of androstane converted to 61st place in a quarterly ammonium group, pharmaceutical mixtures containing them and process for their preparation

Info

Publication number
IL107331A
IL107331A IL10733193A IL10733193A IL107331A IL 107331 A IL107331 A IL 107331A IL 10733193 A IL10733193 A IL 10733193A IL 10733193 A IL10733193 A IL 10733193A IL 107331 A IL107331 A IL 107331A
Authority
IL
Israel
Prior art keywords
group
acetyloxy
bromide
androstan
formula
Prior art date
Application number
IL10733193A
Other languages
English (en)
Hebrew (he)
Other versions
IL107331A0 (en
Original Assignee
Maruishi Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Maruishi Pharma filed Critical Maruishi Pharma
Publication of IL107331A0 publication Critical patent/IL107331A0/xx
Publication of IL107331A publication Critical patent/IL107331A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL10733193A 1992-11-02 1993-10-20 History of androstane converted to 61st place in a quarterly ammonium group, pharmaceutical mixtures containing them and process for their preparation IL107331A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU9203436A HU210076B (en) 1992-11-02 1992-11-02 Process for producing androstane derivatives substituted with quaternisaeted amino group in 16-position and for producing pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
IL107331A0 IL107331A0 (en) 1994-01-25
IL107331A true IL107331A (en) 1998-12-06

Family

ID=10982503

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10733193A IL107331A (en) 1992-11-02 1993-10-20 History of androstane converted to 61st place in a quarterly ammonium group, pharmaceutical mixtures containing them and process for their preparation

Country Status (19)

Country Link
US (1) US5591735A (fr)
EP (1) EP0608495B1 (fr)
JP (1) JP2834651B2 (fr)
KR (1) KR0179399B1 (fr)
CN (1) CN1041937C (fr)
AT (1) ATE154030T1 (fr)
AU (1) AU665866B2 (fr)
BR (1) BR9304466A (fr)
CA (1) CA2108741A1 (fr)
DE (1) DE69311295T2 (fr)
DK (1) DK0608495T3 (fr)
EE (1) EE03073B1 (fr)
ES (1) ES2103413T3 (fr)
GR (1) GR3024011T3 (fr)
HU (1) HU210076B (fr)
IL (1) IL107331A (fr)
NZ (1) NZ248956A (fr)
RU (1) RU2124021C1 (fr)
UA (1) UA27230C2 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020123928A1 (en) * 2001-01-11 2002-09-05 Eldering Charles A. Targeting ads to subscribers based on privacy-protected subscriber profiles
US7200804B1 (en) * 1998-12-08 2007-04-03 Yodlee.Com, Inc. Method and apparatus for providing automation to an internet navigation application
WO2001065453A1 (fr) * 2000-02-29 2001-09-07 Expanse Networks, Inc. Systeme de ciblage a confidentialite protegee
KR20070085703A (ko) * 2005-09-13 2007-08-27 시코르, 인크. 로큐로늄 브로마이드의 합성 방법
CN102675402A (zh) * 2012-05-16 2012-09-19 武汉大学 4，16β-二胺基甾体季铵盐衍生物及其制备方法和应用
CN109053855B (zh) * 2018-10-08 2020-02-14 台州仙琚药业有限公司 一种16β-四氢吡咯基雄甾-2α-环氧-17-酮的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU165600B (fr) * 1972-07-27 1974-09-28
US4177190A (en) * 1975-08-01 1979-12-04 Richter Gedeon Vegyeszeti Gyar Rt. Diamino-androstanes and a process for the preparation of the said compounds
EP0008824B1 (fr) * 1978-09-05 1982-04-28 Akzo N.V. Sels d'addition acides de 2-bêta, 16-bêta-bis pipéridino-androstane-16 bêta-monoammonium quaternaire et préparations pharmaceutiques les contenant
GB8708886D0 (en) * 1987-04-14 1987-05-20 Akzo Nv 2beta-morpholino-androstane derivatives
GB8804579D0 (en) * 1988-02-26 1988-03-30 Akzo Nv Novel 16-homo-piperidino-androstane derivatives & processes for their preparation

Also Published As

Publication number Publication date
KR0179399B1 (ko) 1999-04-01
US5591735A (en) 1997-01-07
JPH06192288A (ja) 1994-07-12
AU665866B2 (en) 1996-01-18
ATE154030T1 (de) 1997-06-15
KR940011476A (ko) 1994-06-21
DE69311295D1 (de) 1997-07-10
DK0608495T3 (da) 1997-08-04
BR9304466A (pt) 1994-06-14
RU2124021C1 (ru) 1998-12-27
CN1090852A (zh) 1994-08-17
HUT66162A (en) 1994-09-28
EP0608495A2 (fr) 1994-08-03
GR3024011T3 (en) 1997-10-31
HU210076B (en) 1995-01-30
CA2108741A1 (fr) 1994-05-03
NZ248956A (en) 1995-08-28
EP0608495A3 (en) 1995-12-20
UA27230C2 (uk) 2000-08-15
HU9203436D0 (en) 1993-01-28
EP0608495B1 (fr) 1997-06-04
IL107331A0 (en) 1994-01-25
CN1041937C (zh) 1999-02-03
DE69311295T2 (de) 1997-10-30
ES2103413T3 (es) 1997-09-16
JP2834651B2 (ja) 1998-12-09
AU4900593A (en) 1995-06-08
EE03073B1 (et) 1998-02-16

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
FF Patent granted
KB Patent renewed
RH1 Patent not in force