BR9304466A - Derivados do androstano, composiçao farmacêutica contendo esses derivados, processo para preparaçao dos mesmos, compostos intermediários, processo para preparaçao da dita composiçao e processo para bloquear a transmissao de impulsos nervosos (estímulos) a músculos estriados - Google Patents

Derivados do androstano, composiçao farmacêutica contendo esses derivados, processo para preparaçao dos mesmos, compostos intermediários, processo para preparaçao da dita composiçao e processo para bloquear a transmissao de impulsos nervosos (estímulos) a músculos estriados

Info

Publication number
BR9304466A
BR9304466A BR9304466A BR9304466A BR9304466A BR 9304466 A BR9304466 A BR 9304466A BR 9304466 A BR9304466 A BR 9304466A BR 9304466 A BR9304466 A BR 9304466A BR 9304466 A BR9304466 A BR 9304466A
Authority
BR
Brazil
Prior art keywords
preparing
derivatives
stimuli
blocking
transmission
Prior art date
Application number
BR9304466A
Other languages
English (en)
Inventor
Zoltan Tuba
E Szilveszter Vizi
Francis F Foldes
Sandor Maho
Original Assignee
Zoltan Tuba
E Szilveszter Vizi
Francis F Foldes
Sandor Maho
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zoltan Tuba, E Szilveszter Vizi, Francis F Foldes, Sandor Maho filed Critical Zoltan Tuba
Publication of BR9304466A publication Critical patent/BR9304466A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J13/00Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/001Oxiranes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BR9304466A 1992-11-02 1993-11-03 Derivados do androstano, composiçao farmacêutica contendo esses derivados, processo para preparaçao dos mesmos, compostos intermediários, processo para preparaçao da dita composiçao e processo para bloquear a transmissao de impulsos nervosos (estímulos) a músculos estriados BR9304466A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU9203436A HU210076B (en) 1992-11-02 1992-11-02 Process for producing androstane derivatives substituted with quaternisaeted amino group in 16-position and for producing pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
BR9304466A true BR9304466A (pt) 1994-06-14

Family

ID=10982503

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9304466A BR9304466A (pt) 1992-11-02 1993-11-03 Derivados do androstano, composiçao farmacêutica contendo esses derivados, processo para preparaçao dos mesmos, compostos intermediários, processo para preparaçao da dita composiçao e processo para bloquear a transmissao de impulsos nervosos (estímulos) a músculos estriados

Country Status (19)

Country Link
US (1) US5591735A (pt)
EP (1) EP0608495B1 (pt)
JP (1) JP2834651B2 (pt)
KR (1) KR0179399B1 (pt)
CN (1) CN1041937C (pt)
AT (1) ATE154030T1 (pt)
AU (1) AU665866B2 (pt)
BR (1) BR9304466A (pt)
CA (1) CA2108741A1 (pt)
DE (1) DE69311295T2 (pt)
DK (1) DK0608495T3 (pt)
EE (1) EE03073B1 (pt)
ES (1) ES2103413T3 (pt)
GR (1) GR3024011T3 (pt)
HU (1) HU210076B (pt)
IL (1) IL107331A (pt)
NZ (1) NZ248956A (pt)
RU (1) RU2124021C1 (pt)
UA (1) UA27230C2 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020123928A1 (en) * 2001-01-11 2002-09-05 Eldering Charles A. Targeting ads to subscribers based on privacy-protected subscriber profiles
US7200804B1 (en) * 1998-12-08 2007-04-03 Yodlee.Com, Inc. Method and apparatus for providing automation to an internet navigation application
WO2001065453A1 (en) * 2000-02-29 2001-09-07 Expanse Networks, Inc. Privacy-protected targeting system
KR20070085703A (ko) * 2005-09-13 2007-08-27 시코르, 인크. 로큐로늄 브로마이드의 합성 방법
CN102675402A (zh) * 2012-05-16 2012-09-19 武汉大学 4,16β-二胺基甾体季铵盐衍生物及其制备方法和应用
CN109053855B (zh) * 2018-10-08 2020-02-14 台州仙琚药业有限公司 一种16β-四氢吡咯基雄甾-2α-环氧-17-酮的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU165600B (pt) * 1972-07-27 1974-09-28
US4177190A (en) * 1975-08-01 1979-12-04 Richter Gedeon Vegyeszeti Gyar Rt. Diamino-androstanes and a process for the preparation of the said compounds
EP0008824B1 (en) * 1978-09-05 1982-04-28 Akzo N.V. Acid addition salts of 16-beta-monoquaternary ammonium derivatives of 2-beta, 16-beta-bis-piperidino-androstanes and pharmaceutical preparations containing same
GB8708886D0 (en) * 1987-04-14 1987-05-20 Akzo Nv 2beta-morpholino-androstane derivatives
GB8804579D0 (en) * 1988-02-26 1988-03-30 Akzo Nv Novel 16-homo-piperidino-androstane derivatives & processes for their preparation

Also Published As

Publication number Publication date
KR0179399B1 (ko) 1999-04-01
US5591735A (en) 1997-01-07
JPH06192288A (ja) 1994-07-12
AU665866B2 (en) 1996-01-18
ATE154030T1 (de) 1997-06-15
KR940011476A (ko) 1994-06-21
DE69311295D1 (de) 1997-07-10
DK0608495T3 (da) 1997-08-04
RU2124021C1 (ru) 1998-12-27
CN1090852A (zh) 1994-08-17
HUT66162A (en) 1994-09-28
EP0608495A2 (en) 1994-08-03
GR3024011T3 (en) 1997-10-31
HU210076B (en) 1995-01-30
CA2108741A1 (en) 1994-05-03
NZ248956A (en) 1995-08-28
EP0608495A3 (en) 1995-12-20
UA27230C2 (uk) 2000-08-15
HU9203436D0 (en) 1993-01-28
IL107331A (en) 1998-12-06
EP0608495B1 (en) 1997-06-04
IL107331A0 (en) 1994-01-25
CN1041937C (zh) 1999-02-03
DE69311295T2 (de) 1997-10-30
ES2103413T3 (es) 1997-09-16
JP2834651B2 (ja) 1998-12-09
AU4900593A (en) 1995-06-08
EE03073B1 (et) 1998-02-16

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Legal Events

Date Code Title Description
GB Transfer
EE Request for examination
EG Technical examination (opinion): publication of technical examination (opinion)
FC Decision: refusal