IE47271B1 - Process for the preparation of 1-n-acyl-aminoglycosides - Google Patents

Process for the preparation of 1-n-acyl-aminoglycosides

Info

Publication number
IE47271B1
IE47271B1 IE842/78A IE84278A IE47271B1 IE 47271 B1 IE47271 B1 IE 47271B1 IE 842/78 A IE842/78 A IE 842/78A IE 84278 A IE84278 A IE 84278A IE 47271 B1 IE47271 B1 IE 47271B1
Authority
IE
Ireland
Prior art keywords
amino
groups
aminoglycoside
polysilylated
formula
Prior art date
Application number
IE842/78A
Other languages
English (en)
Other versions
IE780842L (en
Inventor
Martin John Cron
John Gerard Keil
Jeng Shyong Lin
Mariano Vecchio Ruggeri
Derek Walker
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of IE780842L publication Critical patent/IE780842L/xx
Publication of IE47271B1 publication Critical patent/IE47271B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IE842/78A 1977-04-28 1978-04-27 Process for the preparation of 1-n-acyl-aminoglycosides IE47271B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79180677A 1977-04-28 1977-04-28
US88858578A 1978-03-20 1978-03-20

Publications (2)

Publication Number Publication Date
IE780842L IE780842L (en) 1978-10-28
IE47271B1 true IE47271B1 (en) 1984-02-08

Family

ID=27121201

Family Applications (2)

Application Number Title Priority Date Filing Date
IE842/78A IE47271B1 (en) 1977-04-28 1978-04-27 Process for the preparation of 1-n-acyl-aminoglycosides
IE841/78A IE46945B1 (en) 1977-04-28 1978-04-27 Process for the preparation of kanamycin derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
IE841/78A IE46945B1 (en) 1977-04-28 1978-04-27 Process for the preparation of kanamycin derivatives

Country Status (27)

Country Link
JP (1) JPS53149951A (ja)
AR (1) AR218910A1 (ja)
AT (1) AT357675B (ja)
CA (2) CA1100953A (ja)
CH (1) CH639104A5 (ja)
CS (1) CS207607B2 (ja)
CY (1) CY1241A (ja)
DE (2) DE2818992A1 (ja)
DK (2) DK172543B1 (ja)
EG (1) EG13710A (ja)
ES (1) ES469303A1 (ja)
FI (1) FI781288A (ja)
FR (2) FR2388827A1 (ja)
GB (1) GB1598294A (ja)
HK (1) HK51484A (ja)
IE (2) IE47271B1 (ja)
IT (2) IT1156718B (ja)
KE (1) KE3398A (ja)
LU (1) LU79541A1 (ja)
MY (1) MY8500528A (ja)
NL (1) NL178790C (ja)
NO (2) NO149635C (ja)
PL (1) PL117307B1 (ja)
PT (1) PT67959B (ja)
SE (2) SE447259B (ja)
SG (1) SG22884G (ja)
YU (2) YU102578A (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55306A (en) * 1978-04-28 1980-01-05 Bristol Myers Co Manufacture of 11nn*omegaaaminooalphaahydroxy alkanoyl**aminoglycoside antibiotic
EP1484317A4 (en) * 2002-02-19 2006-08-30 Amato Pharm Prod Ltd LACTIC ACID DERIVATIVE
CN103360440B (zh) 2007-11-21 2016-08-31 尔察祯有限公司 抗菌性氨基糖苷类似物
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin
WO2010132757A2 (en) * 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132765A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs

Also Published As

Publication number Publication date
CS207607B2 (en) 1981-08-31
DK172543B1 (da) 1998-12-07
NO149635C (no) 1984-05-23
DE2818992C2 (ja) 1988-03-17
FR2388826B1 (ja) 1982-12-10
IE780842L (en) 1978-10-28
JPS53149951A (en) 1978-12-27
NO154697B (no) 1986-08-25
YU41590B (en) 1987-12-31
CY1241A (en) 1984-06-29
CA1100953A (en) 1981-05-12
NO154697C (no) 1986-12-03
NL178790B (nl) 1985-12-16
NO781437L (no) 1978-10-31
DE2818822A1 (de) 1978-11-09
NO831197L (no) 1978-10-31
DK182978A (da) 1978-10-29
IE780841L (en) 1978-10-28
FR2388827B1 (ja) 1982-07-09
NO149635B (no) 1984-02-13
PT67959B (en) 1980-03-05
SG22884G (en) 1985-01-04
SE447259B (sv) 1986-11-03
YU102578A (en) 1983-01-21
CH639104A5 (en) 1983-10-31
DK183078A (da) 1978-10-29
DK165450C (da) 1993-04-13
SE7804973L (sv) 1978-10-29
HK51484A (en) 1984-06-22
ES469303A1 (es) 1979-09-16
CA1105454A (en) 1981-07-21
MY8500528A (en) 1985-12-31
GB1598294A (en) 1981-09-16
IT1105500B (it) 1985-11-04
EG13710A (en) 1982-09-30
SE8305538L (sv) 1983-10-07
PL206457A1 (ja) 1980-03-24
LU79541A1 (fr) 1978-11-28
FI781288A (fi) 1978-10-29
DE2818822C2 (ja) 1989-01-26
FR2388827A1 (fr) 1978-11-24
YU102478A (en) 1982-10-31
SE8305538D0 (sv) 1983-10-07
IT1156718B (it) 1987-02-04
NL178790C (nl) 1986-05-16
NL7804503A (nl) 1978-10-31
IT7849137A0 (it) 1978-04-28
PL117307B1 (en) 1981-07-31
AT357675B (de) 1980-07-25
FR2388826A1 (fr) 1978-11-24
DK165450B (da) 1992-11-30
KE3398A (en) 1984-06-08
PT67959A (en) 1978-05-01
IE46945B1 (en) 1983-11-16
IT7849136A0 (it) 1978-04-28
JPS5721277B2 (ja) 1982-05-06
DE2818992A1 (de) 1978-11-23
ATA312778A (de) 1979-12-15
AR218910A1 (es) 1980-07-15
SE461148B (sv) 1990-01-15

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Legal Events

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MK9A Patent expired