ID17504A - Mesilat trihidrat 5-(2-(4-1,2-benzisotiazol-3-il)-1-piperazinil)-etil)-6-kloro-1,3-dihidro-2h-indol-2-on - Google Patents

Mesilat trihidrat 5-(2-(4-1,2-benzisotiazol-3-il)-1-piperazinil)-etil)-6-kloro-1,3-dihidro-2h-indol-2-on

Info

Publication number
ID17504A
ID17504A IDP971490A ID971490A ID17504A ID 17504 A ID17504 A ID 17504A ID P971490 A IDP971490 A ID P971490A ID 971490 A ID971490 A ID 971490A ID 17504 A ID17504 A ID 17504A
Authority
ID
Indonesia
Prior art keywords
trihidrat
mesilat
benzisotiazol
piperazinil
etyl
Prior art date
Application number
IDP971490A
Other languages
English (en)
Indonesian (id)
Inventor
Frank R Busch
Carol A Rose
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ID17504A publication Critical patent/ID17504A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IDP971490A 1996-05-07 1997-05-05 Mesilat trihidrat 5-(2-(4-1,2-benzisotiazol-3-il)-1-piperazinil)-etil)-6-kloro-1,3-dihidro-2h-indol-2-on ID17504A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1653796P 1996-05-07 1996-05-07

Publications (1)

Publication Number Publication Date
ID17504A true ID17504A (id) 1998-01-08

Family

ID=21777622

Family Applications (1)

Application Number Title Priority Date Filing Date
IDP971490A ID17504A (id) 1996-05-07 1997-05-05 Mesilat trihidrat 5-(2-(4-1,2-benzisotiazol-3-il)-1-piperazinil)-etil)-6-kloro-1,3-dihidro-2h-indol-2-on

Country Status (45)

Country Link
US (1) US6110918A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0904273B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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KR (1) KR100333214B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1092658C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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HU (1) HU229057B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ID (1) ID17504A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL126590A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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ZA (1) ZA973875B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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HN1996000101A (es) * 1996-02-28 1997-06-26 Inc Pfizer Terapia combinada para la osteoporosis
UA57734C2 (uk) 1996-05-07 2003-07-15 Пфайзер Інк. Комплекси включення арилгетероциклічних солей
TW491847B (en) 1996-05-07 2002-06-21 Pfizer Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2h-indol-2-one
IL127497A (en) * 1997-12-18 2002-07-25 Pfizer Prod Inc Medicinal products containing piperazinyl-heterocyclic compounds for the treatment of psychiatric disorders
DE69910706T2 (de) * 1998-05-26 2004-07-08 Pfizer Products Inc., Groton Medikament zur Behandlung von Glaukoma und ischämischer Retinopathie
US20080113025A1 (en) * 1998-11-02 2008-05-15 Elan Pharma International Limited Compositions comprising nanoparticulate naproxen and controlled release hydrocodone
IL149186A0 (en) 1999-12-23 2002-11-10 Pfizer Prod Inc Pharmaceutical compositions providing enhanced drug concentrations
CN1431901A (zh) * 2000-06-02 2003-07-23 辉瑞产品公司 用于治疗精神病和眼科疾病的s-甲基-二氢一齐拉昔酮
AR032641A1 (es) * 2001-01-29 2003-11-19 Otsuka Pharma Co Ltd Agonista de subtipo de receptor 5-ht 1a.
US7053092B2 (en) 2001-01-29 2006-05-30 Otsuka Pharmaceutical Co., Ltd. 5-HT1a receptor subtype agonist
US8703772B2 (en) 2001-09-25 2014-04-22 Otsuka Pharmaceutical Co., Ltd. Low hygroscopic aripiprazole drug substance and processes for the preparation thereof
AR033485A1 (es) 2001-09-25 2003-12-26 Otsuka Pharma Co Ltd Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma
US20040048876A1 (en) * 2002-02-20 2004-03-11 Pfizer Inc. Ziprasidone composition and synthetic controls
UY27668A1 (es) * 2002-02-20 2003-10-31 Pfizer Prod Inc Composición de ziprasidona y controles sintéticos
AU2003300814A1 (en) 2002-12-04 2004-06-23 Dr. Reddy's Laboratories Inc. Polymorphic forms of ziprasidone and its hydrochloride
WO2004050655A1 (en) * 2002-12-04 2004-06-17 Dr. Reddy's Laboratories Limited Polymorphic forms of ziprasidone and its hydrochloride
MXPA05012325A (es) * 2003-05-16 2006-01-30 Pfizer Prod Inc Procedimiento para potenciar la cognicion usando zipirasidona.
MXPA05012392A (es) * 2003-05-16 2006-02-02 Pfizer Prod Inc Tratamientos de ansiedad con ziprasidona.
CA2525866A1 (en) * 2003-05-16 2004-11-25 Pfizer Products Inc. Treatment of psychotic and depressive disorders
EP1546146A1 (en) * 2003-06-03 2005-06-29 Teva Pharmaceutical Industries Limited POLYMORPHIC FORMS OF ZIPRASIDONE HCl AND PROCESSES FOR THEIR PREPARATION
CA2537413A1 (en) * 2003-09-02 2005-03-10 Imran Ahmed Sustained release dosage forms of ziprasidone
CA2543805A1 (en) * 2003-10-24 2005-05-06 Gideon Pilarsky Processes for preparation of ziprasidone
EP1592688A2 (en) * 2003-12-18 2005-11-09 Teva Pharmaceutical Industries Ltd. Polymorphic form b2 of ziprasidone base
CA2552126A1 (en) * 2003-12-31 2005-07-21 Actavis Group Hf Ziprasidone formulations
PT1720867E (pt) * 2004-02-27 2010-01-28 Ranbaxy Lab Ltd Processo para a preparação de ziprasidona
WO2006026426A2 (en) * 2004-08-27 2006-03-09 University Of Kentucky Research Foundation Amyloid peptide inactivating enzyme to treat alzheimer’s disease peripherally
ES2250001B1 (es) * 2004-09-29 2007-06-01 Medichem, S.A. Proceso para la purificacion de ziprasidona.
US7777037B2 (en) * 2004-10-27 2010-08-17 Dr. Reddy's Laboratories Limited Ziprasidone process
CA2587710C (en) * 2004-11-16 2014-10-21 Elan Pharma International Ltd. Injectable nanoparticulate olanzapine formulations
EP1863806A1 (en) * 2005-02-11 2007-12-12 Teva Pharmaceutical Industries Ltd Amorphous ziprasidone mesylate
CA2598288A1 (en) * 2005-03-03 2006-09-14 Elan Pharma International Limited Nanoparticulate compositions of heterocyclic amide derivatives
ITMI20050346A1 (it) 2005-03-07 2006-09-08 Dipharma Spa Forma solida di ziprasidone cloridrato
EP1858892A1 (en) * 2005-03-14 2007-11-28 Teva Pharmaceutical Industries Ltd Anhydrous ziprasidone mesylate and a process for its preparation
US20060270684A1 (en) * 2005-03-14 2006-11-30 Judith Aronhime Crystalline forms of ziprasidone mesylate
JP2010527925A (ja) * 2007-05-18 2010-08-19 サイドース・エルエルシー ジプラシドン製剤
KR100948126B1 (ko) * 2007-12-10 2010-03-18 씨제이제일제당 (주) 결정형의 지프라시돈 술폰산염, 그 제조방법, 및 그것를포함하는 약제학적 조성물
CN102234273B (zh) * 2010-04-21 2015-08-05 上海医药工业研究院 甲磺酸齐拉西酮半水合物及其制备方法
SI23610A (sl) 2011-01-13 2012-07-31 Diagen@d@o@o Nove adicijske soli ziprasidona postopek za njihovo pripravo in njihova uporaba v terapiji
CA2891122C (en) 2012-11-14 2021-07-20 The Johns Hopkins University Methods and compositions for treating schizophrenia

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US5312925A (en) 1992-09-01 1994-05-17 Pfizer Inc. Monohydrate of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one-hydrochloride
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Also Published As

Publication number Publication date
PL188164B1 (pl) 2004-12-31
AR007003A1 (es) 1999-10-13
HK1017893A1 (en) 1999-12-03
US6110918A (en) 2000-08-29
DZ2221A1 (fr) 2002-12-03
HN1997000040A (es) 1997-06-05
CA2252895A1 (en) 1997-11-13
NZ508303A (en) 2001-07-27
MA26427A1 (fr) 2004-12-20
DE69720719T2 (de) 2003-11-06
HUP9902808A2 (hu) 2000-03-28
EG24401A (en) 2009-04-29
EP0904273A1 (en) 1999-03-31
JPH11509865A (ja) 1999-08-31
IL126590A0 (en) 1999-08-17
NO985193L (no) 1998-11-06
CA2252895C (en) 2002-08-20
EP0904273B1 (en) 2003-04-09
CO4940465A1 (es) 2000-07-24
SI0904273T1 (en) 2003-08-31
WO1997042190A1 (en) 1997-11-13
TW427989B (en) 2001-04-01
KR20000010822A (ko) 2000-02-25
UA47467C2 (uk) 2002-07-15
OA10908A (en) 2001-10-26
IL126590A (en) 2001-11-25
YU49398B (sh) 2005-11-28
EA001180B1 (ru) 2000-10-30
EA199800909A1 (ru) 1999-04-29
CN1216990A (zh) 1999-05-19
AU730856C (en) 2001-11-15
IS2301B (is) 2007-10-15
NO985193D0 (no) 1998-11-06
AU1936897A (en) 1997-11-26
SK150598A3 (en) 2000-03-13
MY128051A (en) 2007-01-31
ES2192264T3 (es) 2003-10-01
PL329880A1 (en) 1999-04-12
PT904273E (pt) 2003-06-30
TNSN97073A1 (fr) 2005-03-15
ME00901B (me) 2005-11-28
KR100333214B1 (ko) 2002-06-20
GT199700042A (es) 1998-10-02
UY24543A1 (es) 2000-09-29
IS4878A (is) 1998-10-23
AP9700978A0 (en) 1997-07-31
CN1092658C (zh) 2002-10-16
ZA973875B (en) 1998-11-06
AU730856B2 (en) 2001-03-15
HU229057B1 (en) 2013-07-29
NZ332219A (en) 2005-02-25
DE69720719D1 (de) 2003-05-15
BR9708932A (pt) 1999-08-03
SK282674B6 (sk) 2002-11-06
HRP970235B1 (en) 2002-08-31
JP3102896B2 (ja) 2000-10-23
BG63601B1 (bg) 2002-06-28
BG102893A (en) 1999-09-30
YU17397A (sh) 2000-10-30
DK0904273T3 (da) 2003-07-07
CZ349498A3 (cs) 1999-09-15
TR199802241T2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1999-02-22
AP838A (en) 2000-05-03
ATE236902T1 (de) 2003-04-15
HUP9902808A3 (en) 2000-04-28
NO312513B1 (no) 2002-05-21
HRP970235A2 (en) 1998-06-30
CZ289216B6 (cs) 2001-12-12

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