HUT65132A - Process for producing esters of bi- and tricyclic amino-alcohols and pharmaceutical compositions containing them - Google Patents

Process for producing esters of bi- and tricyclic amino-alcohols and pharmaceutical compositions containing them

Info

Publication number
HUT65132A
HUT65132A HU9302611A HU9302611A HUT65132A HU T65132 A HUT65132 A HU T65132A HU 9302611 A HU9302611 A HU 9302611A HU 9302611 A HU9302611 A HU 9302611A HU T65132 A HUT65132 A HU T65132A
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
alcohols
compositions containing
producing esters
tricyclic amino
Prior art date
Application number
HU9302611A
Other languages
English (en)
Other versions
HU224210B1 (hu
HU9302611D0 (en
Inventor
Rolf Banholzer
Rudolf Bauer
Richard Reichl
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of HU9302611D0 publication Critical patent/HU9302611D0/hu
Publication of HUT65132A publication Critical patent/HUT65132A/hu
Publication of HU224210B1 publication Critical patent/HU224210B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
HU9302611A 1991-03-15 1992-03-05 Eljárás bi- és triciklikus amino-alkoholok észterei és ezeket hatóanyagként tartalmazó gyógyszerkészítmények előállítására HU224210B1 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4108393A DE4108393A1 (de) 1991-03-15 1991-03-15 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln
PCT/EP1992/000489 WO1992016528A1 (de) 1991-03-15 1992-03-05 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln

Publications (3)

Publication Number Publication Date
HU9302611D0 HU9302611D0 (en) 1993-12-28
HUT65132A true HUT65132A (en) 1994-04-28
HU224210B1 HU224210B1 (hu) 2005-06-28

Family

ID=6427349

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9302611A HU224210B1 (hu) 1991-03-15 1992-03-05 Eljárás bi- és triciklikus amino-alkoholok észterei és ezeket hatóanyagként tartalmazó gyógyszerkészítmények előállítására

Country Status (26)

Country Link
US (1) US5654314A (hu)
EP (1) EP0579615B1 (hu)
JP (1) JP3352684B2 (hu)
KR (1) KR100307274B1 (hu)
AT (1) ATE202778T1 (hu)
AU (1) AU662128B2 (hu)
CA (1) CA2105575C (hu)
CZ (1) CZ281509B6 (hu)
DE (2) DE4108393A1 (hu)
DK (1) DK0579615T3 (hu)
ES (1) ES2160577T3 (hu)
FI (1) FI120235B (hu)
GR (1) GR3036792T3 (hu)
HU (1) HU224210B1 (hu)
IE (1) IE920815A1 (hu)
IL (1) IL101225A (hu)
MX (1) MX9201139A (hu)
NO (1) NO304266B1 (hu)
NZ (1) NZ241961A (hu)
PL (1) PL179673B1 (hu)
PT (1) PT100234B (hu)
SG (1) SG43037A1 (hu)
SK (1) SK281511B6 (hu)
UA (1) UA29406C2 (hu)
WO (1) WO1992016528A1 (hu)
ZA (1) ZA921875B (hu)

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US7214687B2 (en) * 1999-07-14 2007-05-08 Almirall Ag Quinuclidine derivatives and medicinal compositions containing the same
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US20020137764A1 (en) * 2000-10-31 2002-09-26 Karin Drechsel Inhalable formulation of a solution containing a tiotropium salt
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US7405224B2 (en) 2002-01-31 2008-07-29 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthenecarboxylates, processes for preparing them, and their use as pharmaceutical compositions
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US6696462B2 (en) 2002-01-31 2004-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Anticholinergics, processes for the preparation thereof, and pharmaceutical compositions
DE10211700A1 (de) * 2002-03-16 2003-09-25 Boehringer Ingelheim Pharma Neue Difurylglykolsäureester, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel
US20030229227A1 (en) * 2002-03-16 2003-12-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg New difurylglycolic acid esters, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions
US7309707B2 (en) * 2002-03-20 2007-12-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Crystalline micronisate, process for the manufacture thereof and use thereof for the preparation of a medicament
US7311894B2 (en) * 2002-03-28 2007-12-25 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations containing an anticholinergic
US7244415B2 (en) * 2002-03-28 2007-07-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations of an anhydrate
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TWI695723B (zh) 2009-05-29 2020-06-11 美商沛爾醫療股份有限公司 用於經由呼吸道輸送活性劑的組成物以及相關方法與系統
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Also Published As

Publication number Publication date
NZ241961A (en) 1995-07-26
IL101225A0 (en) 1992-11-15
FI934000A0 (fi) 1993-09-13
SK94993A3 (en) 1994-04-06
US5654314A (en) 1997-08-05
WO1992016528A1 (de) 1992-10-01
ES2160577T3 (es) 2001-11-16
IL101225A (en) 1996-05-14
NO933274D0 (no) 1993-09-14
JPH06505718A (ja) 1994-06-30
CA2105575A1 (en) 1992-09-16
CA2105575C (en) 2000-04-25
ATE202778T1 (de) 2001-07-15
HU224210B1 (hu) 2005-06-28
SG43037A1 (en) 1997-10-17
GR3036792T3 (en) 2002-01-31
FI120235B (fi) 2009-08-14
AU1345792A (en) 1992-10-21
PT100234A (pt) 1993-07-30
DE4108393A1 (de) 1992-09-17
FI934000A (fi) 1993-09-13
SK281511B6 (sk) 2001-04-09
JP3352684B2 (ja) 2002-12-03
KR100307274B1 (ko) 2001-12-05
EP0579615B1 (de) 2001-07-04
ZA921875B (en) 1993-09-13
NO933274L (no) 1993-11-12
HU9302611D0 (en) 1993-12-28
EP0579615A1 (de) 1994-01-26
DE59209907D1 (de) 2001-08-09
AU662128B2 (en) 1995-08-24
MX9201139A (es) 1992-10-01
PT100234B (pt) 1999-06-30
UA29406C2 (uk) 2000-11-15
DK0579615T3 (da) 2001-09-17
IE920815A1 (en) 1992-09-23
NO304266B1 (no) 1998-11-23
CZ191793A3 (en) 1994-05-18
PL179673B1 (pl) 2000-10-31
CZ281509B6 (cs) 1996-10-16

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