HUP9902955A3 - Water-soluble 20 (s)-camptothecin derivatives substituted at position-5, process for their preparation, their use and pharmaceutical compositions containing the same compounds - Google Patents
Water-soluble 20 (s)-camptothecin derivatives substituted at position-5, process for their preparation, their use and pharmaceutical compositions containing the same compoundsInfo
- Publication number
- HUP9902955A3 HUP9902955A3 HU9902955A HUP9902955A HUP9902955A3 HU P9902955 A3 HUP9902955 A3 HU P9902955A3 HU 9902955 A HU9902955 A HU 9902955A HU P9902955 A HUP9902955 A HU P9902955A HU P9902955 A3 HUP9902955 A3 HU P9902955A3
- Authority
- HU
- Hungary
- Prior art keywords
- soluble
- preparation
- water
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
- VSJKWCGYPAHWDS-FQEVSTJZSA-N camptothecin Chemical group C1=CC=C2C=C(CN3C4=CC5=C(C3=O)COC(=O)[C@]5(O)CC)C4=NC2=C1 VSJKWCGYPAHWDS-FQEVSTJZSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US65525996A | 1996-06-05 | 1996-06-05 | |
US65525896A | 1996-06-05 | 1996-06-05 | |
US08/771,391 US6177439B1 (en) | 1995-06-06 | 1996-12-19 | Water soluble analogues of 20(S)-camptothecin |
PCT/US1997/006962 WO1997046563A1 (en) | 1996-06-05 | 1997-04-22 | Novel water-soluble c-ring analogues of 20 (s)-camptothecin |
Publications (3)
Publication Number | Publication Date |
---|---|
HUP9902955A2 HUP9902955A2 (hu) | 2000-02-28 |
HUP9902955A3 true HUP9902955A3 (en) | 2000-04-28 |
HU225989B1 HU225989B1 (en) | 2008-02-28 |
Family
ID=27417940
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9902955A HU225989B1 (en) | 1996-06-05 | 1997-04-22 | 20-(s)-camptothecin derivatives substituted at position 5, process for their preparation, their use and pharmaceutical compositions containing the same compounds |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP0847397B1 (hu) |
JP (1) | JP3600248B2 (hu) |
KR (1) | KR100295238B1 (hu) |
CN (1) | CN1101818C (hu) |
AR (1) | AR006926A1 (hu) |
AU (1) | AU718060C (hu) |
BR (1) | BR9702285A (hu) |
CA (1) | CA2228595C (hu) |
CZ (1) | CZ293421B6 (hu) |
DK (1) | DK0847397T3 (hu) |
HU (1) | HU225989B1 (hu) |
IL (1) | IL123201A (hu) |
MX (1) | MX9800993A (hu) |
NO (1) | NO313998B1 (hu) |
NZ (1) | NZ329896A (hu) |
PL (1) | PL188075B1 (hu) |
TW (1) | TW502037B (hu) |
UA (1) | UA51666C2 (hu) |
WO (1) | WO1997046563A1 (hu) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5972955A (en) * | 1995-06-06 | 1999-10-26 | Dr. Reddy's Research Foundation | Water soluble C-ring analogues of 20(S)-camptothecin |
US6177439B1 (en) * | 1995-06-06 | 2001-01-23 | Reddy's Research Foundation | Water soluble analogues of 20(S)-camptothecin |
ITMI20061475A1 (it) * | 2006-07-26 | 2008-01-27 | Indena Spa | Derivati della camptotecina ad attivita antitumorale |
CN102453036B (zh) * | 2010-10-27 | 2015-12-02 | 李红玉 | 一种喜树碱类化合物及其制备方法和在农药中的用途 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4399282A (en) * | 1979-07-10 | 1983-08-16 | Kabushiki Kaisha Yakult Honsha | Camptothecin derivatives |
US4473692A (en) * | 1981-09-04 | 1984-09-25 | Kabushiki Kaisha Yakult Honsha | Camptothecin derivatives and process for preparing same |
JPS58154584A (ja) * | 1982-03-10 | 1983-09-14 | Yakult Honsha Co Ltd | 5位ヒドロキシ置換カンプトテシン誘導体の製造法 |
JPS58154583A (ja) * | 1982-03-10 | 1983-09-14 | Yakult Honsha Co Ltd | 新規なカンプトテシン誘導体 |
-
1997
- 1997-04-22 HU HU9902955A patent/HU225989B1/hu not_active IP Right Cessation
- 1997-04-22 BR BR9702285-3A patent/BR9702285A/pt not_active IP Right Cessation
- 1997-04-22 CA CA002228595A patent/CA2228595C/en not_active Expired - Fee Related
- 1997-04-22 JP JP50056898A patent/JP3600248B2/ja not_active Expired - Fee Related
- 1997-04-22 IL IL123201A patent/IL123201A/en not_active IP Right Cessation
- 1997-04-22 CZ CZ1998320A patent/CZ293421B6/cs not_active IP Right Cessation
- 1997-04-22 EP EP97936012A patent/EP0847397B1/en not_active Expired - Lifetime
- 1997-04-22 PL PL97324887A patent/PL188075B1/pl not_active IP Right Cessation
- 1997-04-22 DK DK97936012T patent/DK0847397T3/da active
- 1997-04-22 AU AU38781/97A patent/AU718060C/en not_active Ceased
- 1997-04-22 UA UA98031174A patent/UA51666C2/uk unknown
- 1997-04-22 KR KR1019980700862A patent/KR100295238B1/ko not_active IP Right Cessation
- 1997-04-22 WO PCT/US1997/006962 patent/WO1997046563A1/en active IP Right Grant
- 1997-04-22 CN CN97190978A patent/CN1101818C/zh not_active Expired - Fee Related
- 1997-04-22 NZ NZ329896A patent/NZ329896A/xx unknown
- 1997-04-24 TW TW086105385A patent/TW502037B/zh not_active IP Right Cessation
- 1997-04-30 AR ARP970101800A patent/AR006926A1/es active IP Right Grant
-
1998
- 1998-02-04 MX MX9800993A patent/MX9800993A/es not_active IP Right Cessation
- 1998-02-04 NO NO19980485A patent/NO313998B1/no not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
BR9702285A (pt) | 1999-12-28 |
KR19990036194A (ko) | 1999-05-25 |
MX9800993A (es) | 1998-09-30 |
NO980485L (no) | 1998-03-20 |
TW502037B (en) | 2002-09-11 |
UA51666C2 (uk) | 2002-12-16 |
AR006926A1 (es) | 1999-09-29 |
AU718060C (en) | 2002-08-29 |
NO313998B1 (no) | 2003-01-13 |
HUP9902955A2 (hu) | 2000-02-28 |
PL324887A1 (en) | 1998-06-22 |
IL123201A0 (en) | 1998-09-24 |
KR100295238B1 (ko) | 2001-09-17 |
NZ329896A (en) | 1999-09-29 |
CA2228595A1 (en) | 1997-12-11 |
JP3600248B2 (ja) | 2004-12-15 |
CA2228595C (en) | 2002-04-09 |
JPH11501679A (ja) | 1999-02-09 |
AU3878197A (en) | 1998-01-05 |
CN1101818C (zh) | 2003-02-19 |
PL188075B1 (pl) | 2004-12-31 |
EP0847397A1 (en) | 1998-06-17 |
AU718060B2 (en) | 2000-04-06 |
DK0847397T3 (da) | 2002-12-23 |
CZ293421B6 (cs) | 2004-04-14 |
WO1997046563A1 (en) | 1997-12-11 |
CN1198164A (zh) | 1998-11-04 |
IL123201A (en) | 2007-07-24 |
EP0847397B1 (en) | 2002-09-04 |
NO980485D0 (no) | 1998-02-04 |
CZ32098A3 (cs) | 1998-07-15 |
HU225989B1 (en) | 2008-02-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of definitive patent protection due to non-payment of fees |