HUP0203332A3 - Cyclothiocarbamate derivatives, their use as progesterone receptor modulators and pharmaceutical compositions containing them - Google Patents

Cyclothiocarbamate derivatives, their use as progesterone receptor modulators and pharmaceutical compositions containing them

Info

Publication number
HUP0203332A3
HUP0203332A3 HU0203332A HUP0203332A HUP0203332A3 HU P0203332 A3 HUP0203332 A3 HU P0203332A3 HU 0203332 A HU0203332 A HU 0203332A HU P0203332 A HUP0203332 A HU P0203332A HU P0203332 A3 HUP0203332 A3 HU P0203332A3
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
receptor modulators
progesterone receptor
cyclothiocarbamate
Prior art date
Application number
HU0203332A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/552,354 external-priority patent/US6436929B1/en
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of HUP0203332A2 publication Critical patent/HUP0203332A2/hu
Publication of HUP0203332A3 publication Critical patent/HUP0203332A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Chemical Or Physical Treatment Of Fibers (AREA)
  • Detergent Compositions (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HU0203332A 1999-05-04 2000-05-01 Cyclothiocarbamate derivatives, their use as progesterone receptor modulators and pharmaceutical compositions containing them HUP0203332A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18301399P 1999-05-04 1999-05-04
US09/552,354 US6436929B1 (en) 1999-05-04 2000-04-19 Cyclothiocarbamate derivatives as progesterone receptor modulators
PCT/US2000/011749 WO2000066570A1 (en) 1999-05-04 2000-05-01 Cyclothiocarbamate derivatives as progesterone receptor modulators

Publications (2)

Publication Number Publication Date
HUP0203332A2 HUP0203332A2 (hu) 2003-01-28
HUP0203332A3 true HUP0203332A3 (en) 2004-12-28

Family

ID=26878649

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203332A HUP0203332A3 (en) 1999-05-04 2000-05-01 Cyclothiocarbamate derivatives, their use as progesterone receptor modulators and pharmaceutical compositions containing them

Country Status (24)

Country Link
EP (1) EP1175411B1 (https=)
JP (2) JP4958338B2 (https=)
KR (1) KR100732692B1 (https=)
CN (1) CN1131856C (https=)
AT (1) ATE386729T1 (https=)
AU (1) AU766801B2 (https=)
BG (1) BG65277B1 (https=)
BR (1) BR0010214A (https=)
CA (1) CA2371712C (https=)
CZ (1) CZ20013952A3 (https=)
DE (1) DE60038108T2 (https=)
DK (1) DK1175411T3 (https=)
EA (1) EA004511B1 (https=)
ES (1) ES2301482T3 (https=)
GE (1) GEP20043181B (https=)
HU (1) HUP0203332A3 (https=)
IL (1) IL146298A0 (https=)
MX (1) MXPA01011287A (https=)
NO (1) NO321370B1 (https=)
NZ (1) NZ515353A (https=)
PL (1) PL351083A1 (https=)
SG (1) SG120970A1 (https=)
SK (1) SK15922001A3 (https=)
TR (1) TR200103285T2 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG120970A1 (en) * 1999-05-04 2006-04-26 Ligand Pharm Inc Cyclothiocarbamate derivatives as progesterone receptor modulators
US6407101B1 (en) * 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
ES2317223T3 (es) * 2004-04-08 2009-04-16 Wyeth Derivados de tioamida como moduladores del receptor de progesterona.
JP4950027B2 (ja) * 2004-04-08 2012-06-13 ワイス・エルエルシー チオアミド不純物を最小限に抑えるための方法
BRPI0510278A (pt) * 2004-04-27 2007-10-30 Wyeth Corp método para produzir compostos, produto, e, composto
MXPA06012403A (es) 2004-04-27 2007-01-17 Wyeth Corp Purificacion de moduladores de receptor progesterona.
US20060009428A1 (en) * 2004-07-07 2006-01-12 Wyeth Cyclic progestin regimens and kits
MX2007001812A (es) * 2004-08-13 2007-03-26 Wyeth Corp Derivados de tanaproget, metabolitos, y usos de los mismos.
CN101166532B (zh) 2005-04-28 2011-06-22 惠氏公司 微粒化的他那普戈特、组合物及其制备方法
CN101166521A (zh) * 2005-04-28 2008-04-23 惠氏公司 通过湿制粒法制备包含微粒化他那普戈特的组合物
CN101166736B (zh) * 2005-04-28 2013-02-06 惠氏公司 他那普戈特的多晶型ⅱ
AU2006241189B2 (en) * 2005-04-28 2012-01-19 Wyeth Llc Purified form of tanaproget
MX2007013467A (es) 2005-04-28 2008-01-21 Wyeth Corp Tanaproget micronizado y composiciones que contienen el mismo.
CA2610767C (en) * 2005-06-09 2014-09-23 Wyeth Tanaproget compositions containing ethinyl estradiol

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0510235A1 (en) * 1991-04-26 1992-10-28 Dong-A Pharm. Co., Ltd. Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same
JPH0510235A (ja) * 1991-07-05 1993-01-19 Nippondenso Co Ltd 内燃機関の点火時期制御装置
AU1694295A (en) * 1994-01-28 1995-08-15 Merck & Co., Inc. Benzoxazinones as inhibitors of hiv reverse transcriptase
US5696127A (en) * 1994-12-22 1997-12-09 Ligand Pharmaceuticals Incorporated Steroid receptor modulator compounds and methods
EP1043325B1 (en) * 1994-12-22 2004-06-16 Ligand Pharmaceuticals Incorporated Steroid receptor modulator compounds and methods
DE69724630T2 (de) * 1996-10-02 2004-07-29 Bristol-Myers Squibb Pharma Co. 4,4-disubstituierte 1,4-dihydro-2h-3,1-benzoxazin-2-one die anwendbar sind als hiv-reverstranskriptase-inhibitoren, zwischenprodukte und verfahren zu ihrer herstellung
SG120970A1 (en) * 1999-05-04 2006-04-26 Ligand Pharm Inc Cyclothiocarbamate derivatives as progesterone receptor modulators
MX2007013467A (es) * 2005-04-28 2008-01-21 Wyeth Corp Tanaproget micronizado y composiciones que contienen el mismo.
CA2610767C (en) * 2005-06-09 2014-09-23 Wyeth Tanaproget compositions containing ethinyl estradiol

Also Published As

Publication number Publication date
CN1349516A (zh) 2002-05-15
BG106080A (en) 2002-05-31
CZ20013952A3 (cs) 2002-05-15
EA004511B1 (ru) 2004-04-29
JP5523430B2 (ja) 2014-06-18
HUP0203332A2 (hu) 2003-01-28
CA2371712A1 (en) 2000-11-09
JP2002543192A (ja) 2002-12-17
NO20015381D0 (no) 2001-11-02
BG65277B1 (bg) 2007-11-30
GEP20043181B (en) 2004-02-25
EP1175411A1 (en) 2002-01-30
JP2012087129A (ja) 2012-05-10
IL146298A0 (en) 2002-07-25
TR200103285T2 (tr) 2002-02-21
ES2301482T3 (es) 2008-07-01
NO20015381L (no) 2002-01-03
DE60038108D1 (de) 2008-04-03
KR20020000170A (ko) 2002-01-04
NZ515353A (en) 2004-03-26
SK15922001A3 (sk) 2002-09-10
ATE386729T1 (de) 2008-03-15
BR0010214A (pt) 2002-02-13
CN1131856C (zh) 2003-12-24
CA2371712C (en) 2009-12-22
NO321370B1 (no) 2006-05-02
JP4958338B2 (ja) 2012-06-20
PL351083A1 (en) 2003-03-10
AU4811900A (en) 2000-11-17
KR100732692B1 (ko) 2007-06-27
AU766801B2 (en) 2003-10-23
SG120970A1 (en) 2006-04-26
EA200101181A1 (ru) 2002-04-25
DK1175411T3 (da) 2008-06-09
EP1175411B1 (en) 2008-02-20
MXPA01011287A (es) 2003-07-14
DE60038108T2 (de) 2009-02-12

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Legal Events

Date Code Title Description
GB9A Succession in title

Owner name: WYETH, US

Free format text: FORMER OWNER(S): AMERICAN HOME PRODUCTS CO., US; LIGAND PHARMACEUTICALS, INC., US; WYETH, US

FD9A Lapse of provisional protection due to non-payment of fees