MXPA01011287A - Derivados de ciclotiocarbamato como moduladores de receptor de progesterona. - Google Patents

Derivados de ciclotiocarbamato como moduladores de receptor de progesterona.

Info

Publication number
MXPA01011287A
MXPA01011287A MXPA01011287A MXPA01011287A MXPA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A
Authority
MX
Mexico
Prior art keywords
alkyl
optionally substituted
aryl
ring
groups
Prior art date
Application number
MXPA01011287A
Other languages
English (en)
Inventor
P Edwards James
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/552,354 external-priority patent/US6436929B1/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of MXPA01011287A publication Critical patent/MXPA01011287A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
MXPA01011287A 1999-05-04 2000-05-01 Derivados de ciclotiocarbamato como moduladores de receptor de progesterona. MXPA01011287A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18301399P 1999-05-04 1999-05-04
US09/552,354 US6436929B1 (en) 1999-05-04 2000-04-19 Cyclothiocarbamate derivatives as progesterone receptor modulators
PCT/US2000/011749 WO2000066570A1 (en) 1999-05-04 2000-05-01 Cyclothiocarbamate derivatives as progesterone receptor modulators

Publications (1)

Publication Number Publication Date
MXPA01011287A true MXPA01011287A (es) 2003-07-14

Family

ID=26878649

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA01011287A MXPA01011287A (es) 1999-05-04 2000-05-01 Derivados de ciclotiocarbamato como moduladores de receptor de progesterona.

Country Status (24)

Country Link
EP (1) EP1175411B1 (es)
JP (2) JP4958338B2 (es)
KR (1) KR100732692B1 (es)
CN (1) CN1131856C (es)
AT (1) ATE386729T1 (es)
AU (1) AU766801B2 (es)
BG (1) BG65277B1 (es)
BR (1) BR0010214A (es)
CA (1) CA2371712C (es)
CZ (1) CZ20013952A3 (es)
DE (1) DE60038108T2 (es)
DK (1) DK1175411T3 (es)
EA (1) EA004511B1 (es)
ES (1) ES2301482T3 (es)
GE (1) GEP20043181B (es)
HU (1) HUP0203332A3 (es)
IL (1) IL146298A0 (es)
MX (1) MXPA01011287A (es)
NO (1) NO321370B1 (es)
NZ (1) NZ515353A (es)
PL (1) PL351083A1 (es)
SG (1) SG120970A1 (es)
SK (1) SK15922001A3 (es)
TR (1) TR200103285T2 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6407101B1 (en) * 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
BR0010214A (pt) * 1999-05-04 2002-02-13 American Home Prod Derivados de ciclotiocarbamato como moduladores de receptores de progesterona
WO2005100346A1 (en) * 2004-04-08 2005-10-27 Wyeth Thioamide derivatives as progesterone receptor modulators
DK1732922T3 (da) * 2004-04-08 2009-01-12 Wyeth Corp Fremgangsmåde til minimering af thioamidurenheder
MXPA06012402A (es) * 2004-04-27 2007-01-17 Wyeth Corp Carbamato y tiocarbamato biarilos ciclicos que contienen cianopirrol y metodos para preparar los mismos.
AU2005237520B2 (en) 2004-04-27 2012-01-19 Wyeth Purification of progesterone receptor modulators
CN104208067A (zh) * 2004-07-07 2014-12-17 惠氏公司 周期性黄体酮方案及试剂盒
JP4980217B2 (ja) * 2004-08-13 2012-07-18 ワイス・エルエルシー タナプロゲト誘導体、代謝産物、及びそれらの使用
PL1874278T3 (pl) * 2005-04-28 2009-12-31 Wyeth Corp Kompozycje zawierające mikronizowany tanaproget
BRPI0610433A2 (pt) * 2005-04-28 2010-11-23 Wyeth Corp forma polimórfica ii de tanaproget, processos para preparar a mesma, e para preparar forma micronizada de um composto, composição farmacêutica, método de preparação de uma composição farmacêutica, e, uso da forma polimórfica ii de tanaproget ou da forma micronizada
PE20061322A1 (es) * 2005-04-28 2006-12-28 Wyeth Corp Forma purificada de tanaproget
WO2006116596A2 (en) * 2005-04-28 2006-11-02 Wyeth Micronized tanaproget and compostions containing same
WO2006116514A2 (en) 2005-04-28 2006-11-02 Wyeth Micronized tanaproget, compositions, and methods of preparing the same
JP5339903B2 (ja) * 2005-06-09 2013-11-13 ワイス・エルエルシー エチニルエストラジオールを含むタナプロゲット組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0510235A1 (en) * 1991-04-26 1992-10-28 Dong-A Pharm. Co., Ltd. Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same
JPH0510235A (ja) * 1991-07-05 1993-01-19 Nippondenso Co Ltd 内燃機関の点火時期制御装置
WO1995020389A1 (en) * 1994-01-28 1995-08-03 Merck & Co., Inc. Benzoxazinones as inhibitors of hiv reverse transcriptase
US5688808A (en) * 1994-12-22 1997-11-18 Ligand Pharmaceuticals Incorporated Steroid receptor modulator compounds and methods
DK0800519T3 (da) * 1994-12-22 2004-03-01 Ligand Pharm Inc Steroidreceptormodulatorforbindelser og fremgangsmåder
EP0929533B1 (en) * 1996-10-02 2003-09-03 Bristol-Myers Squibb Pharma Company 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same
BR0010214A (pt) * 1999-05-04 2002-02-13 American Home Prod Derivados de ciclotiocarbamato como moduladores de receptores de progesterona
WO2006116596A2 (en) * 2005-04-28 2006-11-02 Wyeth Micronized tanaproget and compostions containing same
JP5339903B2 (ja) * 2005-06-09 2013-11-13 ワイス・エルエルシー エチニルエストラジオールを含むタナプロゲット組成物

Also Published As

Publication number Publication date
EP1175411B1 (en) 2008-02-20
PL351083A1 (en) 2003-03-10
ES2301482T3 (es) 2008-07-01
CN1131856C (zh) 2003-12-24
DE60038108T2 (de) 2009-02-12
HUP0203332A3 (en) 2004-12-28
JP2002543192A (ja) 2002-12-17
BG106080A (en) 2002-05-31
BR0010214A (pt) 2002-02-13
DE60038108D1 (de) 2008-04-03
AU4811900A (en) 2000-11-17
IL146298A0 (en) 2002-07-25
GEP20043181B (en) 2004-02-25
JP5523430B2 (ja) 2014-06-18
CZ20013952A3 (cs) 2002-05-15
KR20020000170A (ko) 2002-01-04
CA2371712A1 (en) 2000-11-09
NZ515353A (en) 2004-03-26
EA200101181A1 (ru) 2002-04-25
NO20015381L (no) 2002-01-03
KR100732692B1 (ko) 2007-06-27
NO20015381D0 (no) 2001-11-02
ATE386729T1 (de) 2008-03-15
EP1175411A1 (en) 2002-01-30
JP2012087129A (ja) 2012-05-10
JP4958338B2 (ja) 2012-06-20
BG65277B1 (bg) 2007-11-30
SK15922001A3 (sk) 2002-09-10
EA004511B1 (ru) 2004-04-29
HUP0203332A2 (hu) 2003-01-28
AU766801B2 (en) 2003-10-23
CN1349516A (zh) 2002-05-15
SG120970A1 (en) 2006-04-26
TR200103285T2 (tr) 2002-02-21
CA2371712C (en) 2009-12-22
DK1175411T3 (da) 2008-06-09
NO321370B1 (no) 2006-05-02

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