HUP0003555A2 - Gombaellenes hatású triazolszármazékok, ezeket tartalmazó gyógyszerkészítmények és intermedierjük - Google Patents

Gombaellenes hatású triazolszármazékok, ezeket tartalmazó gyógyszerkészítmények és intermedierjük

Info

Publication number
HUP0003555A2
HUP0003555A2 HU0003555A HUP0003555A HUP0003555A2 HU P0003555 A2 HUP0003555 A2 HU P0003555A2 HU 0003555 A HU0003555 A HU 0003555A HU P0003555 A HUP0003555 A HU P0003555A HU P0003555 A2 HUP0003555 A2 HU P0003555A2
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
triazole derivatives
antifugal
activity
Prior art date
Application number
HU0003555A
Other languages
English (en)
Inventor
Toshiyuki Konosu
Makoto Mori
Satoshi Ohya
Sadao Oida
Takuya Uchida
Original Assignee
Sankyo Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co., Ltd. filed Critical Sankyo Co., Ltd.
Publication of HU0003555D0 publication Critical patent/HU0003555D0/hu
Publication of HUP0003555A2 publication Critical patent/HUP0003555A2/hu
Publication of HU224699B1 publication Critical patent/HU224699B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/56—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and doubly-bound oxygen atoms bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

A találmány tárgya (I) általános képletű vegyület vagy gyógyászatilagelfogadható sója vagy észterszármazéka, ahol Ar jelentésefenilcsoport, mely adott esetben 1-3 szubsztituenssel helyettesített ahalogénatomok és a trifluormetilcsoportok közül választva. A találmánytárgyát képezi továbbá a fenti vegyületek gyógyászati készítménybenvaló alkalmazása, (II) képletű intermedierjük, illetve maguk agyógyászati készítmények is. Ó
HU0003555A 1999-09-09 2000-09-08 Triazole derivatives having antifugal activity, pharmaceutical compositions containing them and their use for producing medicaments HU224699B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP25570299 1999-09-09
JP2000103826 2000-04-05

Publications (3)

Publication Number Publication Date
HU0003555D0 HU0003555D0 (en) 2000-09-08
HUP0003555A2 true HUP0003555A2 (hu) 2002-05-29
HU224699B1 HU224699B1 (en) 2006-01-30

Family

ID=26542380

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0003555A HU224699B1 (en) 1999-09-09 2000-09-08 Triazole derivatives having antifugal activity, pharmaceutical compositions containing them and their use for producing medicaments

Country Status (23)

Country Link
US (3) US6391903B1 (hu)
EP (1) EP1083175B1 (hu)
KR (1) KR100592201B1 (hu)
CN (1) CN1167700C (hu)
AR (1) AR025610A1 (hu)
AT (1) ATE244238T1 (hu)
AU (1) AU778073B2 (hu)
BR (1) BR0004066A (hu)
CA (1) CA2317691C (hu)
DE (1) DE60003618T2 (hu)
DK (1) DK1083175T3 (hu)
ES (1) ES2200786T3 (hu)
HK (1) HK1034259A1 (hu)
HU (1) HU224699B1 (hu)
ID (1) ID27234A (hu)
IL (1) IL138329A0 (hu)
NO (1) NO318352B1 (hu)
NZ (1) NZ506818A (hu)
PT (1) PT1083175E (hu)
RU (1) RU2203280C2 (hu)
SA (1) SA00210602B1 (hu)
TR (1) TR200002610A3 (hu)
TW (1) TW530057B (hu)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI334866B (en) 2002-05-29 2010-12-21 Mercian Corp Novel physiologically active substances
TW200503697A (en) * 2003-06-06 2005-02-01 Sankyo Co Medicinal compositions containing triazole compounds
EP1954264B1 (en) 2005-12-01 2009-10-07 Basilea Pharmaceutica AG Process for the manufacture of epoxybutanol intermediates
AU2008211950A1 (en) 2007-01-29 2008-08-07 Eisai R & D Management Co., Ltd. Solid of macrolide compound, method for production thereof, and pharmaceutical composition comprising the same

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8322983D0 (en) * 1983-08-26 1983-09-28 Pfizer Ltd Triazole antifungal agents
US4483863A (en) * 1984-01-20 1984-11-20 Pfizer Inc. Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
TW198027B (hu) * 1990-08-26 1993-01-11 Sankyo Co
JP2902345B2 (ja) 1995-04-06 1999-06-07 三共株式会社 トリアゾール抗真菌剤
CN1151138C (zh) 1995-04-06 2004-05-26 三共株式会社 三唑抗真菌剂
EP0780380B1 (en) * 1995-12-22 2001-06-13 Ss Pharmaceutical Co., Ltd. Triazole derivatives with antimycotic action and intermediates
JP3622882B2 (ja) 1996-10-04 2005-02-23 三共株式会社 トリアゾール誘導体を含有する医薬
AU5779598A (en) 1997-02-04 1998-08-25 Sankyo Company Limited Triazole derivatives
JPH1180135A (ja) 1997-07-08 1999-03-26 Sankyo Co Ltd 抗真菌トリアゾール化合物
WO1999002524A1 (fr) 1997-07-08 1999-01-21 Sankyo Company, Limited Composes antifongiques a base de triazole
US6303728B1 (en) 1997-07-08 2001-10-16 Kaneka Corporation Hydrosilylation process and polymers produced by the process

Also Published As

Publication number Publication date
KR20010067169A (ko) 2001-07-12
DK1083175T3 (da) 2003-10-06
EP1083175A3 (en) 2001-04-11
US6391903B1 (en) 2002-05-21
HU0003555D0 (en) 2000-09-08
TR200002610A2 (tr) 2001-06-21
KR100592201B1 (ko) 2006-06-23
RU2203280C2 (ru) 2003-04-27
NZ506818A (en) 2001-07-27
CA2317691A1 (en) 2001-03-09
PT1083175E (pt) 2003-09-30
CN1167700C (zh) 2004-09-22
TR200002610A3 (tr) 2001-06-21
CN1291610A (zh) 2001-04-18
SA00210602B1 (ar) 2006-06-04
ID27234A (id) 2001-03-15
CA2317691C (en) 2009-02-17
ES2200786T3 (es) 2004-03-16
AU5657500A (en) 2001-03-15
NO20004511D0 (no) 2000-09-08
US6392082B1 (en) 2002-05-21
EP1083175B1 (en) 2003-07-02
DE60003618T2 (de) 2004-04-15
NO318352B1 (no) 2005-03-07
HU224699B1 (en) 2006-01-30
TW530057B (en) 2003-05-01
DE60003618D1 (de) 2003-08-07
US6337403B1 (en) 2002-01-08
NO20004511L (no) 2001-03-12
EP1083175A2 (en) 2001-03-14
AR025610A1 (es) 2002-12-04
BR0004066A (pt) 2001-04-17
AU778073B2 (en) 2004-11-11
ATE244238T1 (de) 2003-07-15
HK1034259A1 (en) 2001-10-19
IL138329A0 (en) 2001-10-31

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Legal Events

Date Code Title Description
HFG4 Patent granted, date of granting

Effective date: 20051123

MM4A Lapse of definitive patent protection due to non-payment of fees