HUE025801T2 - Amidin funkciós csoporttal rendelkezõ hatóanyagok bioelérhetõségének javítása gyógyszerkészítményben - Google Patents
Amidin funkciós csoporttal rendelkezõ hatóanyagok bioelérhetõségének javítása gyógyszerkészítményben Download PDFInfo
- Publication number
- HUE025801T2 HUE025801T2 HUE07785614A HUE07785614A HUE025801T2 HU E025801 T2 HUE025801 T2 HU E025801T2 HU E07785614 A HUE07785614 A HU E07785614A HU E07785614 A HUE07785614 A HU E07785614A HU E025801 T2 HUE025801 T2 HU E025801T2
- Authority
- HU
- Hungary
- Prior art keywords
- inhibitor
- use according
- inhibitors
- bioavailability
- medicaments
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/08—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis for Pneumocystis carinii
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
- C07C259/12—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
- C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- AIDS & HIV (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Claims (6)
- Szíthatta 1mi igénvpomok ί. Az tt) képlesÊ N,Nmdihidrevktmídín alkalmazásam gÿ'ôgyhaîàsd anyag tmtldin hmkcios csoportjának heiyePexkejeként gyógyszerekben a gyógyhatású aovs'g bioaléthetoségènek javasára.
- 2. Az 1. Igénypont szerinti alkalmazás, azzal jellemezve, hogy a gyógyhatású anyag a kdve-kezok csoportjából válaszloti: pcoteáz Inhibitorok, DNS- & RNS-mterkaláió vegy8kt«k, viráiis enzimek inhibitora; és N-teetil-ö-aszpartát receptor aníagogiaták.
- 3 A 2. igénypont szerűm aikahuazús, azzal jeliofuezYe, hogy a proteáz inhibitor egy írotnbsn inhibitor, Xa Dktör inhibitora. Vii iakto< inhibitora vagy a kongóidéiba kaszkátl mindegyik proieázának inhibitora vagy mairigiáz inhibitor.
- 4. a 2. igénypont szerinti alkalmazás, azzal jellemezve, hogy a proteáz inhibitor egy nrokináz jnhMor,
- 5. A 2. igénypont szerinti alkalmazás, azzal jellemezve, hogy a DNS- és RNS-Iznerknláló vegyidet a peaiamiáin, dirmnazéo vagy ixommatnidlnet.
- 6. A 2. igénypont szerinti alkalmazás, azzal jellemezve, hogy a viráiis enzimek inhibitora egy nearaminiááz inhibitor. ?. A 2. igénypont szerűm alkalmazás az mi jellemezve. hogy a gyógyhatású anyag egy N-metll-D-axzpatíáz receptor atbagonista.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102006034256A DE102006034256A1 (de) | 2006-07-21 | 2006-07-21 | Verbesserung der Bioverfügbarkeit von Wirkstoffen mit Amidinfunktion in Arzneimitteln |
Publications (1)
Publication Number | Publication Date |
---|---|
HUE025801T2 true HUE025801T2 (hu) | 2016-04-28 |
Family
ID=38721771
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HUE07785614A HUE025801T2 (hu) | 2006-07-21 | 2007-07-10 | Amidin funkciós csoporttal rendelkezõ hatóanyagok bioelérhetõségének javítása gyógyszerkészítményben |
Country Status (19)
Country | Link |
---|---|
US (1) | US20090270440A1 (hu) |
EP (2) | EP2987784A1 (hu) |
JP (1) | JP2009544588A (hu) |
KR (1) | KR20090075792A (hu) |
CN (2) | CN101506151A (hu) |
AU (1) | AU2007276526B2 (hu) |
CA (2) | CA2658434C (hu) |
CY (1) | CY1116941T1 (hu) |
DE (1) | DE102006034256A1 (hu) |
DK (1) | DK2046732T5 (hu) |
ES (1) | ES2555778T3 (hu) |
HK (2) | HK1210694A1 (hu) |
HU (1) | HUE025801T2 (hu) |
PL (1) | PL2046732T3 (hu) |
PT (1) | PT2046732E (hu) |
SG (1) | SG173401A1 (hu) |
SI (1) | SI2046732T1 (hu) |
WO (1) | WO2008009264A1 (hu) |
ZA (1) | ZA200901212B (hu) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9662308B2 (en) | 2008-02-01 | 2017-05-30 | Dritte Patentportfolio Beteiligungsgesellschaft Mbh & Co. Kg | Orally bioavailable pentamidine prodrugs for the treatment of diseases |
DE102008007440A1 (de) | 2008-02-01 | 2009-08-13 | Dritte Patentportfolio Beteiligungsgesellschaft Mbh & Co.Kg | Aminosäurederivate als Arzneistoffe |
DE102008007381A1 (de) * | 2008-02-01 | 2009-08-13 | Dritte Patentportfolio Beteiligungsgesellschaft Mbh & Co.Kg | Amidine und Guanidine und deren Derivate zur Behandlung von Krankheiten |
DE102008061247A1 (de) | 2008-12-10 | 2010-06-24 | Christian-Albrechts-Universität Zu Kiel | Inhibitoren der Dimethylarginin Dimethylaminohydrolase |
DE102009004204A1 (de) * | 2009-01-09 | 2010-07-15 | Christian-Albrechts-Universität Zu Kiel | Verfahren zur verbesserten Bioaktivierung von Arzneistoffen |
CN103420994B (zh) * | 2012-05-24 | 2016-04-06 | 天津药物研究院 | 作为前药的达比加群酯衍生物及其制备方法和用途 |
CN103864710B (zh) * | 2014-03-24 | 2016-05-25 | 西安近代化学研究所 | 一种3-(3-氨基呋咱-4-基)-5-甲基-5-取代-4-羟基-4h,5h-1,2,4-恶二唑化合物的合成方法 |
CN103951660B (zh) * | 2014-03-24 | 2016-07-06 | 西安近代化学研究所 | 一种恶二唑化合物的合成方法 |
GB201615693D0 (en) | 2016-09-15 | 2016-11-02 | Combinatorx Infection Ltd | Combinations |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4321444A1 (de) * | 1993-06-28 | 1995-01-05 | Bernd Prof Dr Clement | Pharmazeutische Zubereitung |
US5723495A (en) * | 1995-11-16 | 1998-03-03 | The University Of North Carolina At Chapel Hill | Benzamidoxime prodrugs as antipneumocystic agents |
US6740682B2 (en) * | 1997-08-29 | 2004-05-25 | Tularik Limited | Meta-benzamidine derivatives as serine protease inhibitors |
US6291514B1 (en) * | 1998-02-09 | 2001-09-18 | 3-Dimensional Pharmaceuticals, Inc. | Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors |
US7157596B2 (en) * | 2000-09-08 | 2007-01-02 | Dendreon Corporation | Inhibitors of serine protease activity of matriptase or MTSP1 |
US20040082585A1 (en) * | 2001-10-03 | 2004-04-29 | Pharmacia Corporation | Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
-
2006
- 2006-07-21 DE DE102006034256A patent/DE102006034256A1/de not_active Withdrawn
-
2007
- 2007-07-10 CN CNA2007800275303A patent/CN101506151A/zh active Pending
- 2007-07-10 CA CA2658434A patent/CA2658434C/en not_active Expired - Fee Related
- 2007-07-10 SG SG2011052545A patent/SG173401A1/en unknown
- 2007-07-10 EP EP15184167.3A patent/EP2987784A1/de not_active Withdrawn
- 2007-07-10 CA CA2777173A patent/CA2777173A1/en not_active Abandoned
- 2007-07-10 ES ES07785614.4T patent/ES2555778T3/es active Active
- 2007-07-10 PT PT77856144T patent/PT2046732E/pt unknown
- 2007-07-10 DK DK07785614.4T patent/DK2046732T5/en active
- 2007-07-10 US US12/374,300 patent/US20090270440A1/en not_active Abandoned
- 2007-07-10 KR KR1020097002587A patent/KR20090075792A/ko not_active Application Discontinuation
- 2007-07-10 JP JP2009519786A patent/JP2009544588A/ja active Pending
- 2007-07-10 PL PL07785614T patent/PL2046732T3/pl unknown
- 2007-07-10 CN CN201510045378.8A patent/CN104644619A/zh active Pending
- 2007-07-10 SI SI200731707T patent/SI2046732T1/sl unknown
- 2007-07-10 WO PCT/DE2007/001216 patent/WO2008009264A1/de active Application Filing
- 2007-07-10 AU AU2007276526A patent/AU2007276526B2/en not_active Ceased
- 2007-07-10 HU HUE07785614A patent/HUE025801T2/hu unknown
- 2007-07-10 EP EP07785614.4A patent/EP2046732B1/de not_active Not-in-force
-
2009
- 2009-02-20 ZA ZA2009/01212A patent/ZA200901212B/en unknown
-
2015
- 2015-11-17 CY CY20151101033T patent/CY1116941T1/el unknown
- 2015-11-19 HK HK15111410.2A patent/HK1210694A1/xx unknown
-
2016
- 2016-08-10 HK HK16109558.7A patent/HK1221455A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
EP2046732A1 (de) | 2009-04-15 |
CA2658434C (en) | 2012-08-14 |
HK1210694A1 (en) | 2016-05-06 |
SG173401A1 (en) | 2011-08-29 |
AU2007276526A1 (en) | 2008-01-24 |
DK2046732T5 (en) | 2016-01-04 |
WO2008009264A1 (de) | 2008-01-24 |
CN104644619A (zh) | 2015-05-27 |
EP2046732B1 (de) | 2015-09-09 |
US20090270440A1 (en) | 2009-10-29 |
DE102006034256A1 (de) | 2008-01-31 |
CY1116941T1 (el) | 2017-04-05 |
ES2555778T3 (es) | 2016-01-08 |
HK1221455A1 (zh) | 2017-06-02 |
ZA200901212B (en) | 2010-02-24 |
PL2046732T3 (pl) | 2016-02-29 |
EP2987784A1 (de) | 2016-02-24 |
PT2046732E (pt) | 2016-01-06 |
CA2658434E (en) | 2008-01-24 |
CA2777173A1 (en) | 2008-01-24 |
CA2658434A1 (en) | 2008-01-24 |
KR20090075792A (ko) | 2009-07-09 |
AU2007276526B2 (en) | 2011-08-11 |
DK2046732T3 (en) | 2015-11-16 |
CN101506151A (zh) | 2009-08-12 |
JP2009544588A (ja) | 2009-12-17 |
SI2046732T1 (sl) | 2016-02-29 |
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