HU222015B1 - Benzopiránvegyületek előállítási eljárásaiban felhasználható intermedierek és eljárás a köztitermékek előállítására - Google Patents

Benzopiránvegyületek előállítási eljárásaiban felhasználható intermedierek és eljárás a köztitermékek előállítására Download PDF

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Publication number
HU222015B1
HU222015B1 HU9503137A HU9503137A HU222015B1 HU 222015 B1 HU222015 B1 HU 222015B1 HU 9503137 A HU9503137 A HU 9503137A HU 9503137 A HU9503137 A HU 9503137A HU 222015 B1 HU222015 B1 HU 222015B1
Authority
HU
Hungary
Prior art keywords
formula
alkyl
compound
group
hydrogen
Prior art date
Application number
HU9503137A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9503137D0 (en
HUT72660A (en
Inventor
Richard Gramam Geen
Graham Johnson
Inderjit Singh Mann
Vance Novack
Neil Smith
Original Assignee
Smithkline Beecham Plc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc. filed Critical Smithkline Beecham Plc.
Publication of HU9503137D0 publication Critical patent/HU9503137D0/hu
Publication of HUT72660A publication Critical patent/HUT72660A/hu
Publication of HU222015B1 publication Critical patent/HU222015B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HU9503137A 1992-11-27 1993-11-19 Benzopiránvegyületek előállítási eljárásaiban felhasználható intermedierek és eljárás a köztitermékek előállítására HU222015B1 (hu)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB929224922A GB9224922D0 (en) 1992-11-27 1992-11-27 Process
HU9501553A HU222017B1 (hu) 1992-11-27 1993-11-19 Eljárás benzopiránszármazékok előállítására
PCT/EP1993/003257 WO1994012492A1 (en) 1992-11-27 1993-11-19 Process for preparing benzopyran compounds

Publications (3)

Publication Number Publication Date
HU9503137D0 HU9503137D0 (en) 1995-12-28
HUT72660A HUT72660A (en) 1996-05-28
HU222015B1 true HU222015B1 (hu) 2003-03-28

Family

ID=10725801

Family Applications (2)

Application Number Title Priority Date Filing Date
HU9501553A HU222017B1 (hu) 1992-11-27 1993-11-19 Eljárás benzopiránszármazékok előállítására
HU9503137A HU222015B1 (hu) 1992-11-27 1993-11-19 Benzopiránvegyületek előállítási eljárásaiban felhasználható intermedierek és eljárás a köztitermékek előállítására

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HU9501553A HU222017B1 (hu) 1992-11-27 1993-11-19 Eljárás benzopiránszármazékok előállítására

Country Status (33)

Country Link
US (3) US5616721A (cs)
EP (1) EP0670835B1 (cs)
JP (2) JP3505179B2 (cs)
KR (1) KR100305150B1 (cs)
CN (1) CN1049657C (cs)
AP (1) AP428A (cs)
AT (1) ATE234297T1 (cs)
AU (1) AU673704B2 (cs)
BR (1) BR9307539A (cs)
CA (1) CA2149886C (cs)
CZ (2) CZ282991B6 (cs)
DE (1) DE69332761T2 (cs)
DK (1) DK0670835T3 (cs)
ES (1) ES2194023T3 (cs)
FI (1) FI952585L (cs)
GB (1) GB9224922D0 (cs)
HU (2) HU222017B1 (cs)
IL (3) IL119366A (cs)
MA (1) MA23041A1 (cs)
MX (1) MX9307406A (cs)
MY (1) MY109573A (cs)
NO (2) NO307967B1 (cs)
NZ (1) NZ257857A (cs)
PH (1) PH31585A (cs)
PL (1) PL175039B1 (cs)
RU (1) RU2094428C1 (cs)
SG (1) SG48341A1 (cs)
SI (1) SI9300613A (cs)
SK (1) SK281083B6 (cs)
TW (1) TW376384B (cs)
UA (1) UA41904C2 (cs)
WO (1) WO1994012492A1 (cs)
ZA (1) ZA938826B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2167384A1 (en) 1994-05-16 1995-11-23 Hideki Ushio Process for producing tetrazole compound and intermediate therefor
GB9410207D0 (en) * 1994-05-21 1994-07-06 Smithkline Beecham Plc Process
EP0716088B1 (en) * 1994-06-23 2004-02-18 Sumitomo Chemical Company, Limited Process for producing 2-(tetrazol-5-yl)-4-oxo-4h-benzopyrans
CH691301A5 (de) * 1995-06-29 2001-06-29 Sumitomo Chemical Co Verfahren zur Herstellung von 2-Acetyl-6-(4-(4-phenylbutoxy)benzoyl)aminophenol.
FR2742753B1 (fr) * 1995-12-22 1998-01-30 Rhone Poulenc Rorer Sa Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
DK0814804T3 (da) * 1996-01-04 2002-11-11 Smithkline Beecham Corp Substituerede benzopyraner
GB9700331D0 (en) * 1997-01-09 1997-02-26 Smithkline Beecham Plc Process
KR100683274B1 (ko) 2004-02-12 2007-02-15 에스케이케미칼주식회사 치환된 벤조피란 화합물의 제조방법
US7511171B2 (en) * 2004-04-01 2009-03-31 Sumitomo Chemical Company, Limited Method for producing carboxylic acid compound
KR100716274B1 (ko) 2006-10-02 2007-05-09 에스케이케미칼주식회사 치환된 벤조피란 화합물 합성용 화합물
KR100760015B1 (ko) * 2006-10-02 2007-09-19 에스케이케미칼주식회사 벤조피란 화합물 합성용 중간체
WO2010002075A1 (en) * 2008-07-02 2010-01-07 Pharmacostech Co., Ltd. Methods for preparing amide derivatives
CN101450943B (zh) * 2008-11-10 2012-11-07 河北科技大学 一种从四氢呋喃途径合成药物普仑司特的方法
CN104402711A (zh) * 2014-11-12 2015-03-11 平湖优康药物研发有限公司 一种抗哮喘药物普伦斯特中间体的合成工艺
CN108912100A (zh) * 2018-08-20 2018-11-30 浙江三门恒康制药有限公司 一种普仑斯特的制备方法
CN108947984B (zh) * 2018-09-17 2020-07-07 烟台万润药业有限公司 一种普仑司特的制备方法
CN110423206B (zh) * 2019-07-17 2022-07-08 天津大学 从氨肟化反应产物中分离环己酮肟、环己酮与甲苯的方法
CN111943899B (zh) * 2020-09-08 2023-04-21 河北凯诺中星科技有限公司 一种5-甲酸乙酯四氮唑的合成方法
CN113620937A (zh) * 2021-08-03 2021-11-09 湖南复瑞生物医药技术有限责任公司 一种高纯度小粒径普仑司特的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1362782A (en) * 1970-08-26 1974-08-07 Fisons Ltd Tetrazole derivatives
GB8402577D0 (en) * 1984-02-01 1984-03-07 Fisons Plc Nitrogen heterocyclic compounds
CA1261835A (en) * 1984-08-20 1989-09-26 Masaaki Toda (fused) benz(thio)amides
JPH0395144A (ja) * 1989-08-04 1991-04-19 Ono Pharmaceut Co Ltd アミノフェノール誘導体の製造方法
JP3095144B1 (ja) * 1999-05-10 2000-10-03 工業技術院長 生分解性ポリウレタン複合体及びその製造方法

Also Published As

Publication number Publication date
CA2149886A1 (en) 1994-06-09
PL309228A1 (en) 1995-10-02
AU673704B2 (en) 1996-11-21
HU222017B1 (hu) 2003-03-28
DK0670835T3 (da) 2003-06-23
FI952585A7 (fi) 1995-05-26
JPH08503481A (ja) 1996-04-16
CZ135795A3 (en) 1995-11-15
SK69695A3 (en) 1995-11-08
US5587483A (en) 1996-12-24
SK281083B6 (sk) 2000-11-07
IL119366A0 (en) 1997-01-10
AP428A (en) 1995-11-09
ATE234297T1 (de) 2003-03-15
NO952090L (no) 1995-05-29
HU9503137D0 (en) 1995-12-28
CN1107153A (zh) 1995-08-23
RU95113433A (ru) 1997-02-20
NO996324D0 (no) 1999-12-20
CA2149886C (en) 2005-05-03
US5616721A (en) 1997-04-01
NZ257857A (en) 1996-11-26
NO996324L (no) 1995-05-29
TW376384B (en) 1999-12-11
GB9224922D0 (en) 1993-01-13
EP0670835B1 (en) 2003-03-12
DE69332761T2 (de) 2004-03-18
MY109573A (en) 1997-02-28
CZ58497A3 (en) 1997-08-13
FI952585A0 (fi) 1995-05-26
SI9300613A (en) 1994-06-30
FI952585L (fi) 1995-05-26
CZ283978B6 (cs) 1998-07-15
KR950704305A (ko) 1995-11-17
AU5466594A (en) 1994-06-22
UA41904C2 (uk) 2001-10-15
CZ282991B6 (cs) 1997-12-17
MA23041A1 (fr) 1994-07-01
HK1012393A1 (en) 1999-07-30
RU2094428C1 (ru) 1997-10-27
JP3505179B2 (ja) 2004-03-08
PH31585A (en) 1998-11-03
JP2004035570A (ja) 2004-02-05
PL175039B1 (pl) 1998-10-30
US5596103A (en) 1997-01-21
IL107759A (en) 1998-12-06
HU9501553D0 (en) 1995-07-28
DE69332761D1 (de) 2003-04-17
IL119366A (en) 2001-08-26
JP3763828B2 (ja) 2006-04-05
IL107759A0 (en) 1994-02-27
WO1994012492A1 (en) 1994-06-09
SG48341A1 (en) 1998-04-17
NO952090D0 (no) 1995-05-26
EP0670835A1 (en) 1995-09-13
NO307967B1 (no) 2000-06-26
ZA938826B (en) 1995-05-25
CN1049657C (zh) 2000-02-23
AP9300593A0 (en) 1994-01-31
HUT72660A (en) 1996-05-28
MX9307406A (es) 1994-07-29
NO309718B1 (no) 2001-03-19
ES2194023T3 (es) 2003-11-16
KR100305150B1 (ko) 2001-11-22
HUT74010A (en) 1996-10-28
BR9307539A (pt) 1999-05-25

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