HRP970273A2 - Vitamin d3 analogs - Google Patents

Vitamin d3 analogs

Info

Publication number
HRP970273A2
HRP970273A2 HR60/039,900A HRP970273A HRP970273A2 HR P970273 A2 HRP970273 A2 HR P970273A2 HR P970273 A HRP970273 A HR P970273A HR P970273 A2 HRP970273 A2 HR P970273A2
Authority
HR
Croatia
Prior art keywords
analogs
vitamin
Prior art date
Application number
HR60/039,900A
Other languages
English (en)
Inventor
Andrew David Batcho
Graeme Findlay Bryce
Bernard Michael Hennessy
Jerome Anthony Iacobelli
Milan Radoje Uskokovic
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HRP970273A2 publication Critical patent/HRP970273A2/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HR60/039,900A 1996-05-23 1997-05-20 Vitamin d3 analogs HRP970273A2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1818696P 1996-05-23 1996-05-23
US1815396P 1996-05-23 1996-05-23
US3990097P 1997-03-19 1997-03-19

Publications (1)

Publication Number Publication Date
HRP970273A2 true HRP970273A2 (en) 1998-04-30

Family

ID=27360973

Family Applications (1)

Application Number Title Priority Date Filing Date
HR60/039,900A HRP970273A2 (en) 1996-05-23 1997-05-20 Vitamin d3 analogs

Country Status (29)

Country Link
EP (2) EP1464640A3 (de)
JP (1) JP2859247B2 (de)
KR (1) KR100783856B1 (de)
CN (1) CN1176072C (de)
AR (1) AR007241A1 (de)
AT (1) ATE277008T1 (de)
AU (1) AU723929B2 (de)
BR (1) BR9703384A (de)
CA (1) CA2205275C (de)
CO (1) CO4950531A1 (de)
CZ (1) CZ157897A3 (de)
DE (1) DE69730774T2 (de)
DK (1) DK0808833T3 (de)
ES (1) ES2227635T3 (de)
HR (1) HRP970273A2 (de)
HU (1) HUP9700926A3 (de)
IL (1) IL120843A0 (de)
MA (1) MA24251A1 (de)
NO (1) NO972304L (de)
NZ (1) NZ314839A (de)
PE (1) PE70198A1 (de)
PL (1) PL320132A1 (de)
PT (1) PT808833E (de)
SG (1) SG70009A1 (de)
TR (1) TR199700415A2 (de)
TW (1) TW445252B (de)
UY (1) UY24561A1 (de)
YU (1) YU20197A (de)
ZA (1) ZA974336B (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5939408A (en) 1996-05-23 1999-08-17 Hoffman-La Roche Inc. Vitamin D3 analogs
JP2002515898A (ja) * 1997-02-25 2002-05-28 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン ヒトの皮膚での経時老化を防止および治療するための方法および組成物
EP0981514B1 (de) * 1997-05-16 2006-04-05 Woman & Infants Hospital 3-epi-vitamin d2 verbindungen und ihre anwendungen
CA2289209C (en) 1997-05-16 2006-07-25 Women & Infants Hospital Cyclic ether vitamin d3 compounds, 1.alpha. (oh) 3-epi-vitamin d3 compounds and uses thereof
EP0957098A1 (de) * 1998-05-14 1999-11-17 F. Hoffmann-La Roche Ag Zwischenprodukte zur Synthese von 3-epi Vitamin D3 Metaboliten und Analogen
US6603030B1 (en) 1999-04-22 2003-08-05 Hoffman-La Roche Inc. Process for producing phosphineoxide vitamin D precursors
CA2370565C (en) * 1999-04-23 2008-11-25 Leo Pharma A/S Dermally applicable vitamin d-containing pharmaceutical compositions
US6255501B1 (en) * 1999-04-26 2001-07-03 Hoffman-La Roche Inc. Process for preparing antiosteoporotic agents
US20020045606A1 (en) * 1999-12-02 2002-04-18 Reddy Satyanarayana G. Esters of vitamin D3 and uses thereof
US7332482B2 (en) 2003-09-24 2008-02-19 Bioxell S.P.A. Method for treating benign prostatic hyperplasia
GB2407499B (en) * 2003-11-03 2008-02-27 Bioxell Spa Vitamin D3 analogue for use in the treatment of BPH
BRPI0404050A (pt) * 2003-09-24 2005-06-14 Bioxell Spa Uso de um composto ou de um seu sal ou éster farmaceuticamente aceitável, formulação farmacêutica, formulação acondicionada, composto, e, método para prevenir e/ou tratar hiperplasia benigna da próstata em pacientes em necessidade de tal prevenção ou tratamento
JP2007525533A (ja) 2004-03-01 2007-09-06 ビオエクセル エスピーエー 間質性膀胱炎の治療方法、並びに関連化合物及び組成物
CA2586679A1 (en) 2004-11-12 2006-05-18 Bioxell Spa Combined use of vitamin d derivatives and anti-proliferative agents for treating bladder cancer
CA2605815A1 (en) * 2005-04-25 2006-11-02 Cytochroma Inc. Low-calcemic 16,23-diene 25-oxime analogs of 1alpha,25-dihydroxy vitamin d3
BRPI0614894A2 (pt) * 2005-08-18 2016-08-30 Bioxell Spa método para produzir um composto, e, composto
TW200838544A (en) * 2007-01-25 2008-10-01 Bioxell Spa Synthesis of 1 α-fluoro-25-hydroxy-16-23E-diene-26, 27-bishomo-20-epi-cholecalciferol
ES2544819T3 (es) 2007-05-30 2015-09-04 Opko IP Holdings II, Inc. Proceso para la producción de precursores de la vitamina D de óxido de fosfina
ES2366077B2 (es) * 2010-03-30 2012-06-25 Universidade De Vigo Compuestos quirales, procedimientos de obtención y uso.
US9006220B2 (en) * 2010-10-25 2015-04-14 Teijin Pharma Limited 23-yne-vitamin D3 derivative
WO2014074601A2 (en) * 2012-11-07 2014-05-15 Vid Scale, Inc Temporal filter for denoising a high dynamic range video
CN105348164B (zh) * 2015-10-29 2017-03-29 无锡福祈制药有限公司 一种1α‑羟基维生素D2的制备方法
CN106748942B (zh) * 2016-11-28 2018-06-29 无锡福祈制药有限公司 度骨化醇类似物wxfq-65及其合成方法
ES2731558B2 (es) * 2018-05-15 2020-03-18 Univ Santiago Compostela Compuestos de interés farmacéutico
CN109738252B (zh) * 2019-01-23 2021-03-09 深圳天辰医疗科技有限公司 25-羟基-维生素d解离液
CN109696435B (zh) * 2019-01-25 2021-03-09 深圳天辰医疗科技有限公司 维生素d的测定方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA8923B (en) * 1988-01-20 1989-09-27 Hoffmann La Roche 16-dehydro-vitamin d3-derivatives
GB8914963D0 (en) * 1989-06-29 1989-08-23 Leo Pharm Prod Ltd Chemical compounds
GB9017890D0 (en) * 1990-08-15 1990-09-26 Leo Pharm Prod Ltd Chemical compounds i
GB9206648D0 (en) * 1992-03-26 1992-05-06 Leo Pharm Prod Ltd Chemical compounds
ATE141914T1 (de) * 1992-05-20 1996-09-15 Hoffmann La Roche Fluorierte analoge vitamins d3
US5428029A (en) * 1993-11-24 1995-06-27 Hoffmann-La Roche Inc. Vitamin D3 fluorinated analogs
JP3228488B2 (ja) * 1993-12-24 2001-11-12 株式会社クラレ 20−エピステロイド誘導体およびその製造方法

Also Published As

Publication number Publication date
IL120843A0 (en) 1997-09-30
AR007241A1 (es) 1999-10-27
EP0808833B1 (de) 2004-09-22
SG70009A1 (en) 2000-01-25
CA2205275A1 (en) 1997-11-23
HU9700926D0 (en) 1997-07-28
HUP9700926A3 (en) 1999-05-28
YU20197A (sh) 1999-09-27
EP1464640A2 (de) 2004-10-06
NO972304D0 (no) 1997-05-21
CA2205275C (en) 2007-04-03
CN1176072C (zh) 2004-11-17
UY24561A1 (es) 2000-12-29
AU2357797A (en) 1997-11-27
ZA974336B (en) 1997-11-24
HUP9700926A2 (hu) 1998-01-28
JP2859247B2 (ja) 1999-02-17
ATE277008T1 (de) 2004-10-15
EP0808833A3 (de) 1998-11-25
PE70198A1 (es) 1998-11-26
CN1175573A (zh) 1998-03-11
PL320132A1 (en) 1997-11-24
DE69730774T2 (de) 2005-09-29
TW445252B (en) 2001-07-11
EP0808833A2 (de) 1997-11-26
MA24251A1 (fr) 1998-04-01
MX9703774A (es) 1998-06-30
KR100783856B1 (ko) 2008-05-09
KR970074765A (ko) 1997-12-10
EP1464640A3 (de) 2005-01-12
ES2227635T3 (es) 2005-04-01
AU723929B2 (en) 2000-09-07
NZ314839A (en) 2000-01-28
DK0808833T3 (da) 2005-01-31
TR199700415A3 (tr) 1997-12-21
NO972304L (no) 1997-11-24
BR9703384A (pt) 1998-09-15
CO4950531A1 (es) 2000-09-01
JPH1045713A (ja) 1998-02-17
TR199700415A2 (xx) 1997-12-21
DE69730774D1 (de) 2004-10-28
CZ157897A3 (en) 1997-12-17
PT808833E (pt) 2004-11-30

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Legal Events

Date Code Title Description
A1OB Publication of a patent application
AIPI Request for the grant of a patent on the basis of a substantive examination of a patent application
ODBC Application rejected