HRP20201621T1 - Derivati indola za uporabu u medicini - Google Patents

Derivati indola za uporabu u medicini Download PDF

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Publication number
HRP20201621T1
HRP20201621T1 HRP20201621TT HRP20201621T HRP20201621T1 HR P20201621 T1 HRP20201621 T1 HR P20201621T1 HR P20201621T T HRP20201621T T HR P20201621TT HR P20201621 T HRP20201621 T HR P20201621T HR P20201621 T1 HRP20201621 T1 HR P20201621T1
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HR
Croatia
Prior art keywords
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cancer
lymphoma
leukemia
cell
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HRP20201621TT
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English (en)
Croatian (hr)
Inventor
Phillip Cowley
Alan Wise
Susan Davis
Michael Kiczun
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Iomet Pharma Ltd.
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Priority claimed from GB201406154A external-priority patent/GB201406154D0/en
Priority claimed from GB201502156A external-priority patent/GB201502156D0/en
Application filed by Iomet Pharma Ltd. filed Critical Iomet Pharma Ltd.
Publication of HRP20201621T1 publication Critical patent/HRP20201621T1/hr

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    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/42—Oxazoles
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