HRP20040516A2 - Crystalline form of a ribofuranosyluronamide derivative; a human adenosine a2a receptor agonist - Google Patents
Crystalline form of a ribofuranosyluronamide derivative; a human adenosine a2a receptor agonist Download PDFInfo
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- HRP20040516A2 HRP20040516A2 HR20040516A HRP20040516A HRP20040516A2 HR P20040516 A2 HRP20040516 A2 HR P20040516A2 HR 20040516 A HR20040516 A HR 20040516A HR P20040516 A HRP20040516 A HR P20040516A HR P20040516 A2 HRP20040516 A2 HR P20040516A2
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- HR
- Croatia
- Prior art keywords
- ethyl
- ribofuranosyluronamide
- diphenylethyl
- purine
- carboxamide
- Prior art date
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Applications Claiming Priority (2)
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GBGB0129273.9A GB0129273D0 (en) | 2001-12-06 | 2001-12-06 | Crystalline drug form |
PCT/IB2002/004979 WO2003048180A1 (en) | 2001-12-06 | 2002-11-27 | Crystalline form of a ribofuranosyluronamide derivative; a human adenosine a2a receptor agonist |
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HR20040516A HRP20040516A2 (en) | 2001-12-06 | 2004-06-07 | Crystalline form of a ribofuranosyluronamide derivative; a human adenosine a2a receptor agonist |
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US20030225089A1 (en) * | 2002-04-10 | 2003-12-04 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pharmaceutical compositions based on anticholinergics and p38 kinase inhibitors |
DE10345065A1 (de) * | 2003-09-26 | 2005-04-14 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Aerosolformulierung für die Inhalation enthaltend ein Anticholinergikum |
PE20060272A1 (es) | 2004-05-24 | 2006-05-22 | Glaxo Group Ltd | (2r,3r,4s,5r,2'r,3'r,4's,5's)-2,2'-{trans-1,4-ciclohexanodiilbis-[imino(2-{[2-(1-metil-1h-imidazol-4-il)etil]amino}-9h-purin-6,9-diil)]}bis[5-(2-etil-2h-tetrazol-5-il)tetrahidro-3,4-furanodiol] como agonista a2a |
GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
WO2021084791A1 (ja) * | 2019-10-28 | 2021-05-06 | 有限会社イムノ | アデノシンa2a受容体を標的とする組成物 |
CN115400140B (zh) * | 2022-01-27 | 2024-02-20 | 宁波熙健医药科技有限公司 | 呋喃核糖基吡啶衍生物用于预防或治疗癫痫或惊厥的用途 |
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US5376645A (en) | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
KR0166088B1 (ko) | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
IT1254915B (it) * | 1992-04-24 | 1995-10-11 | Gloria Cristalli | Derivati di adenosina ad attivita' a2 agonista |
GB9711643D0 (en) | 1997-06-05 | 1997-07-30 | Janssen Pharmaceutica Nv | Glass thermoplastic systems |
GB9913932D0 (en) * | 1999-06-15 | 1999-08-18 | Pfizer Ltd | Purine derivatives |
WO2001020089A1 (fr) | 1999-09-10 | 2001-03-22 | Maeda Corporation | Structure de beton et procede de construction |
GB0003960D0 (en) * | 2000-02-18 | 2000-04-12 | Pfizer Ltd | Purine derivatives |
GB0009606D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Therapeutic combinations |
GB0009605D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Medicaments |
GB0009592D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory combinations |
GB0009583D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory formulations |
TWI227240B (en) * | 2000-06-06 | 2005-02-01 | Pfizer | 2-aminocarbonyl-9H-purine derivatives |
AU5800800A (en) | 2000-07-26 | 2002-02-05 | Swisscom Mobile Ag | Method for the assembly of a mobile radio network base station and connection ofthe base station to the network |
WO2002096462A1 (en) * | 2001-05-25 | 2002-12-05 | Pfizer Inc. | An adenosine a2a receptor agonist and an anticholinergic agent in combination for treating obstructive airways diseases |
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