ZA200403967B - Crystalline form of a ribofuranosyluronamide derivative, a humen adenosine A2A receptor agonist - Google Patents
Crystalline form of a ribofuranosyluronamide derivative, a humen adenosine A2A receptor agonist Download PDFInfo
- Publication number
- ZA200403967B ZA200403967B ZA200403967A ZA200403967A ZA200403967B ZA 200403967 B ZA200403967 B ZA 200403967B ZA 200403967 A ZA200403967 A ZA 200403967A ZA 200403967 A ZA200403967 A ZA 200403967A ZA 200403967 B ZA200403967 B ZA 200403967B
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- ZA
- South Africa
- Prior art keywords
- ethyl
- ribofuranosyluronamide
- purine
- amino
- pyridyl
- Prior art date
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0129273.9A GB0129273D0 (en) | 2001-12-06 | 2001-12-06 | Crystalline drug form |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200403967B true ZA200403967B (en) | 2006-05-31 |
Family
ID=9927165
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200403967A ZA200403967B (en) | 2001-12-06 | 2004-05-21 | Crystalline form of a ribofuranosyluronamide derivative, a humen adenosine A2A receptor agonist |
Country Status (41)
| Country | Link |
|---|---|
| US (3) | US6852746B2 (pt) |
| EP (1) | EP1456219B1 (pt) |
| JP (1) | JP4184279B2 (pt) |
| KR (1) | KR100554333B1 (pt) |
| CN (1) | CN100381454C (pt) |
| AP (1) | AP2004003056A0 (pt) |
| AR (2) | AR038547A1 (pt) |
| AT (1) | ATE364615T1 (pt) |
| AU (2) | AU2002347509B2 (pt) |
| BR (1) | BR0214747A (pt) |
| CA (1) | CA2468847C (pt) |
| CY (1) | CY1106822T1 (pt) |
| DE (1) | DE60220713T2 (pt) |
| DK (1) | DK1456219T3 (pt) |
| EA (1) | EA006857B1 (pt) |
| EC (1) | ECSP045141A (pt) |
| ES (1) | ES2286303T3 (pt) |
| GB (1) | GB0129273D0 (pt) |
| GT (2) | GT200200256A (pt) |
| HK (1) | HK1071143A1 (pt) |
| HN (1) | HN2002000352A (pt) |
| HR (1) | HRP20040516A2 (pt) |
| HU (1) | HUP0700046A2 (pt) |
| IL (2) | IL162101A0 (pt) |
| IS (1) | IS7279A (pt) |
| MA (1) | MA27151A1 (pt) |
| MX (1) | MXPA04005505A (pt) |
| NO (1) | NO20042837L (pt) |
| NZ (1) | NZ533053A (pt) |
| OA (1) | OA12737A (pt) |
| PA (2) | PA8560501A1 (pt) |
| PE (2) | PE20030822A1 (pt) |
| PL (1) | PL370971A1 (pt) |
| PT (1) | PT1456219E (pt) |
| RS (1) | RS49504A (pt) |
| SV (1) | SV2004001425A (pt) |
| TN (1) | TNSN04103A1 (pt) |
| TW (2) | TW200301130A (pt) |
| UY (1) | UY27568A1 (pt) |
| WO (2) | WO2003048180A1 (pt) |
| ZA (1) | ZA200403967B (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030225089A1 (en) * | 2002-04-10 | 2003-12-04 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pharmaceutical compositions based on anticholinergics and p38 kinase inhibitors |
| DE10345065A1 (de) * | 2003-09-26 | 2005-04-14 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Aerosolformulierung für die Inhalation enthaltend ein Anticholinergikum |
| AR049384A1 (es) | 2004-05-24 | 2006-07-26 | Glaxo Group Ltd | Derivados de purina |
| GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
| JPWO2021084791A1 (pt) * | 2019-10-28 | 2021-05-06 | ||
| CN115400140B (zh) * | 2022-01-27 | 2024-02-20 | 宁波熙健医药科技有限公司 | 呋喃核糖基吡啶衍生物用于预防或治疗癫痫或惊厥的用途 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5376645A (en) | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| KR0166088B1 (ko) | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
| IT1254915B (it) * | 1992-04-24 | 1995-10-11 | Gloria Cristalli | Derivati di adenosina ad attivita' a2 agonista |
| GB9711643D0 (en) | 1997-06-05 | 1997-07-30 | Janssen Pharmaceutica Nv | Glass thermoplastic systems |
| GB9913932D0 (en) * | 1999-06-15 | 1999-08-18 | Pfizer Ltd | Purine derivatives |
| WO2001020089A1 (fr) | 1999-09-10 | 2001-03-22 | Maeda Corporation | Structure de beton et procede de construction |
| GB0003960D0 (en) * | 2000-02-18 | 2000-04-12 | Pfizer Ltd | Purine derivatives |
| GB0009592D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory combinations |
| GB0009606D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Therapeutic combinations |
| GB0009583D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory formulations |
| GB0009605D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Medicaments |
| TWI227240B (en) * | 2000-06-06 | 2005-02-01 | Pfizer | 2-aminocarbonyl-9H-purine derivatives |
| EP1304005B1 (de) | 2000-07-26 | 2004-09-15 | Swisscom Mobile AG | Verfahren zum errichten einer basisstation eines mobilfunknetzes und verbinden der basisstation mit dem mobilfunknetz |
| EP1395287A1 (en) * | 2001-05-25 | 2004-03-10 | Pfizer Inc. | An adenosine a2a receptor agonist and an anticholinergic agent in combination for treating obstructive airways diseases |
-
2001
- 2001-12-06 GB GBGB0129273.9A patent/GB0129273D0/en not_active Ceased
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2002
- 2002-11-27 EA EA200400638A patent/EA006857B1/ru not_active IP Right Cessation
- 2002-11-27 CA CA002468847A patent/CA2468847C/en not_active Expired - Fee Related
- 2002-11-27 AP APAP/P/2004/003056A patent/AP2004003056A0/en unknown
- 2002-11-27 RS YU49504A patent/RS49504A/sr unknown
- 2002-11-27 HU HU0700046A patent/HUP0700046A2/hu unknown
- 2002-11-27 JP JP2003549368A patent/JP4184279B2/ja not_active Expired - Fee Related
- 2002-11-27 PL PL02370971A patent/PL370971A1/xx not_active Application Discontinuation
- 2002-11-27 AU AU2002347509A patent/AU2002347509B2/en not_active Ceased
- 2002-11-27 BR BR0214747-5A patent/BR0214747A/pt not_active IP Right Cessation
- 2002-11-27 NZ NZ533053A patent/NZ533053A/en unknown
- 2002-11-27 OA OA1200400163A patent/OA12737A/en unknown
- 2002-11-27 WO PCT/IB2002/004979 patent/WO2003048180A1/en active IP Right Grant
- 2002-11-27 AT AT02783443T patent/ATE364615T1/de not_active IP Right Cessation
- 2002-11-27 KR KR1020047008594A patent/KR100554333B1/ko not_active IP Right Cessation
- 2002-11-27 CN CNB028244117A patent/CN100381454C/zh not_active Expired - Fee Related
- 2002-11-27 IL IL16210102A patent/IL162101A0/xx unknown
- 2002-11-27 WO PCT/IB2002/005038 patent/WO2003047597A1/en not_active Application Discontinuation
- 2002-11-27 MX MXPA04005505A patent/MXPA04005505A/es active IP Right Grant
- 2002-11-27 ES ES02783443T patent/ES2286303T3/es not_active Expired - Lifetime
- 2002-11-27 EP EP02783443A patent/EP1456219B1/en not_active Expired - Lifetime
- 2002-11-27 DE DE60220713T patent/DE60220713T2/de not_active Expired - Lifetime
- 2002-11-27 PT PT02783443T patent/PT1456219E/pt unknown
- 2002-11-27 AU AU2002351056A patent/AU2002351056A1/en not_active Abandoned
- 2002-11-27 DK DK02783443T patent/DK1456219T3/da active
- 2002-12-02 PE PE2002001155A patent/PE20030822A1/es not_active Application Discontinuation
- 2002-12-02 PE PE2002001154A patent/PE20030722A1/es not_active Application Discontinuation
- 2002-12-03 HN HN2002000352A patent/HN2002000352A/es unknown
- 2002-12-03 US US10/308,805 patent/US6852746B2/en not_active Expired - Fee Related
- 2002-12-03 US US10/308,829 patent/US20030144243A1/en not_active Abandoned
- 2002-12-04 AR ARP020104683A patent/AR038547A1/es unknown
- 2002-12-04 AR ARP020104684A patent/AR037633A1/es not_active Application Discontinuation
- 2002-12-05 GT GT200200256A patent/GT200200256A/es unknown
- 2002-12-05 TW TW091135302A patent/TW200301130A/zh unknown
- 2002-12-05 UY UY27568A patent/UY27568A1/es not_active Application Discontinuation
- 2002-12-05 TW TW091135301A patent/TW200301129A/zh unknown
- 2002-12-05 GT GT200200257A patent/GT200200257A/es unknown
- 2002-12-05 SV SV2002001425A patent/SV2004001425A/es not_active Application Discontinuation
- 2002-12-06 PA PA20028560501A patent/PA8560501A1/es unknown
- 2002-12-06 PA PA20028560301A patent/PA8560301A1/es unknown
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2004
- 2004-05-20 IL IL162101A patent/IL162101A/en not_active IP Right Cessation
- 2004-05-21 IS IS7279A patent/IS7279A/is unknown
- 2004-05-21 ZA ZA200403967A patent/ZA200403967B/en unknown
- 2004-06-02 MA MA27711A patent/MA27151A1/fr unknown
- 2004-06-04 EC EC2004005141A patent/ECSP045141A/es unknown
- 2004-06-04 TN TNP2004000103A patent/TNSN04103A1/fr unknown
- 2004-06-07 HR HR20040516A patent/HRP20040516A2/hr not_active Application Discontinuation
- 2004-07-05 NO NO20042837A patent/NO20042837L/no not_active Application Discontinuation
- 2004-09-03 US US10/934,903 patent/US7022727B2/en not_active Expired - Fee Related
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2005
- 2005-05-06 HK HK05103825A patent/HK1071143A1/xx not_active IP Right Cessation
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2007
- 2007-08-27 CY CY20071101103T patent/CY1106822T1/el unknown
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