HK1176054A1 - Fused heteroaromatic pyrrolidinones as syk inhibitors syk - Google Patents

Fused heteroaromatic pyrrolidinones as syk inhibitors syk

Info

Publication number
HK1176054A1
HK1176054A1 HK13102881.3A HK13102881A HK1176054A1 HK 1176054 A1 HK1176054 A1 HK 1176054A1 HK 13102881 A HK13102881 A HK 13102881A HK 1176054 A1 HK1176054 A1 HK 1176054A1
Authority
HK
Hong Kong
Prior art keywords
syk
fused heteroaromatic
inhibitors
pyrrolidinones
heteroaromatic pyrrolidinones
Prior art date
Application number
HK13102881.3A
Other languages
English (en)
Chinese (zh)
Inventor
Yasuyoshi Arikawa
Benjamin Jones
Betty Lam
Zhe Nie
Christopher Smith
Masashi Takahashi
Qing Dong
Victoria Feher
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43618073&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1176054(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of HK1176054A1 publication Critical patent/HK1176054A1/xx

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Veterinary Medicine (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Diabetes (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
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  • Endocrinology (AREA)
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  • Obesity (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
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HK13102881.3A 2009-12-23 2013-03-07 Fused heteroaromatic pyrrolidinones as syk inhibitors syk HK1176054A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28996909P 2009-12-23 2009-12-23
US38696410P 2010-09-27 2010-09-27
PCT/US2010/061146 WO2011079051A1 (en) 2009-12-23 2010-12-17 Fused heteroaromatic pyrrolidinones as syk inhibitors

Publications (1)

Publication Number Publication Date
HK1176054A1 true HK1176054A1 (en) 2013-07-19

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Family Applications (1)

Application Number Title Priority Date Filing Date
HK13102881.3A HK1176054A1 (en) 2009-12-23 2013-03-07 Fused heteroaromatic pyrrolidinones as syk inhibitors syk

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US (7) US8440689B2 (ar)
EP (4) EP3825316A1 (ar)
JP (7) JP5658274B2 (ar)
KR (1) KR101790255B1 (ar)
CN (1) CN102753548B (ar)
AR (1) AR081797A1 (ar)
AU (1) AU2010333804B2 (ar)
BR (1) BR112012015651B1 (ar)
CA (1) CA2786950C (ar)
CL (1) CL2012001745A1 (ar)
CO (1) CO6592058A2 (ar)
CR (1) CR20120392A (ar)
CY (1) CY1116736T1 (ar)
DK (1) DK2516434T3 (ar)
DO (1) DOP2012000180A (ar)
EA (1) EA021568B1 (ar)
EC (1) ECSP12012057A (ar)
ES (1) ES2545616T3 (ar)
GE (1) GEP20156243B (ar)
HK (1) HK1176054A1 (ar)
HR (1) HRP20150878T1 (ar)
HU (1) HUE025177T2 (ar)
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MA (1) MA33909B1 (ar)
ME (1) ME02186B (ar)
MX (1) MX2012007402A (ar)
MY (1) MY159257A (ar)
NZ (1) NZ601267A (ar)
PE (1) PE20130188A1 (ar)
PL (1) PL2516434T3 (ar)
PT (1) PT2516434E (ar)
RS (1) RS54180B1 (ar)
SG (1) SG181857A1 (ar)
SI (1) SI2516434T1 (ar)
SM (1) SMT201500199B (ar)
TN (1) TN2012000316A1 (ar)
TW (1) TWI457339B (ar)
UA (1) UA107100C2 (ar)
UY (1) UY33151A (ar)
WO (1) WO2011079051A1 (ar)
ZA (1) ZA201205428B (ar)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2516434T3 (pl) 2009-12-23 2015-11-30 Takeda Pharmaceuticals Co Skondensowane heteroaromatyczne pirolidynony jako inhibitory SYK
ES2588680T3 (es) * 2011-03-28 2016-11-04 F. Hoffmann-La Roche Ag Compuestos de tiazolopirimidina
EP2723739B1 (en) * 2011-06-22 2016-08-24 Takeda Pharmaceutical Company Limited Substituted 6-aza-isoindolin-1-one derivatives
US9469654B2 (en) 2012-09-27 2016-10-18 Portola Pharmaceuticals, Inc. Bicyclic oxa-lactam kinase inhibitors
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