HK1096673A1 - Compositions useful as inhibitors of protein kinases - Google Patents
Compositions useful as inhibitors of protein kinasesInfo
- Publication number
- HK1096673A1 HK1096673A1 HK07101507.7A HK07101507A HK1096673A1 HK 1096673 A1 HK1096673 A1 HK 1096673A1 HK 07101507 A HK07101507 A HK 07101507A HK 1096673 A1 HK1096673 A1 HK 1096673A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- inhibitors
- protein kinases
- compositions useful
- compounds
- compositions
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 3
- 102000001253 Protein Kinase Human genes 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 108060006633 protein kinase Proteins 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 4
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 1
Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
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- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurosurgery (AREA)
- Virology (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Communicable Diseases (AREA)
- Psychiatry (AREA)
- Molecular Biology (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Otolaryngology (AREA)
- Biotechnology (AREA)
- Pain & Pain Management (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US51088103P | 2003-10-14 | 2003-10-14 | |
PCT/US2004/033749 WO2005037843A1 (en) | 2003-10-14 | 2004-10-14 | Compositions useful as inhibitors of protein kinases |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1096673A1 true HK1096673A1 (en) | 2007-06-08 |
Family
ID=36585960
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK07101507.7A HK1096673A1 (en) | 2003-10-14 | 2007-02-08 | Compositions useful as inhibitors of protein kinases |
Country Status (12)
Country | Link |
---|---|
US (3) | US7700609B2 (ja) |
EP (1) | EP1692140B1 (ja) |
JP (2) | JP2007509848A (ja) |
CN (3) | CN1897950A (ja) |
AT (1) | ATE451376T1 (ja) |
AU (1) | AU2004282172B2 (ja) |
CA (1) | CA2542113A1 (ja) |
DE (1) | DE602004024572D1 (ja) |
ES (1) | ES2338234T3 (ja) |
HK (1) | HK1096673A1 (ja) |
TW (1) | TW200530251A (ja) |
WO (1) | WO2005037843A1 (ja) |
Families Citing this family (180)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1897950A (zh) | 2003-10-14 | 2007-01-17 | 惠氏公司 | 稠合芳基和杂芳基衍生物及其使用方法 |
KR101372783B1 (ko) | 2004-01-22 | 2014-03-11 | 유니버시티 오브 마이애미 | 국소용 코-엔자임 큐10 제형 및 그의 사용 방법 |
US7772232B2 (en) * | 2004-04-15 | 2010-08-10 | Bristol-Myers Squibb Company | Quinazolinyl compounds as inhibitors of potassium channel function |
US8057815B2 (en) * | 2004-04-19 | 2011-11-15 | Portola Pharmaceuticals, Inc. | Methods of treatment with Syk inhibitors |
WO2005111039A2 (en) | 2004-05-14 | 2005-11-24 | Millennium Pharmaceuticals, Inc. | Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase |
MY147767A (en) * | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
WO2006023861A1 (en) * | 2004-08-24 | 2006-03-02 | Janssen Pharmaceutica N.V. | Novel benzo-fused heteroaryl sulfamide derivatives useful as anticonvulsant agents |
US20060276528A1 (en) * | 2004-08-24 | 2006-12-07 | Abdel-Magid Ahmed F | Novel benzo-fused heteroaryl sulfamide derivatives useful as anticonvulsant agents |
US7459448B2 (en) | 2004-10-04 | 2008-12-02 | Millennium Pharmaceuticals, Inc. | Lactam compounds useful as protein kinase inhibitors |
ATE479687T1 (de) | 2004-10-15 | 2010-09-15 | Takeda Pharmaceutical | Kinaseinhibitoren |
CN101754947A (zh) * | 2005-05-20 | 2010-06-23 | 詹森药业有限公司 | 磺酰胺衍生物的制备方法 |
US8058231B2 (en) * | 2005-09-20 | 2011-11-15 | Nihon University | Transcriptional regulation of high affinity IgE receptor γ-chain |
US8119655B2 (en) | 2005-10-07 | 2012-02-21 | Takeda Pharmaceutical Company Limited | Kinase inhibitors |
US20070155824A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives for disease modification / epileptogenesis |
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- 2004-10-14 ES ES04794973T patent/ES2338234T3/es active Active
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- 2004-10-14 EP EP04794973A patent/EP1692140B1/en active Active
- 2004-10-14 CN CN201010166197A patent/CN101824043A/zh active Pending
- 2004-10-14 AT AT04794973T patent/ATE451376T1/de not_active IP Right Cessation
- 2004-10-14 WO PCT/US2004/033749 patent/WO2005037843A1/en active Application Filing
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- 2004-10-14 TW TW093131191A patent/TW200530251A/zh unknown
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CN1894258A (zh) | 2007-01-10 |
CN1894258B (zh) | 2010-06-16 |
TW200530251A (en) | 2005-09-16 |
JP2007509848A (ja) | 2007-04-19 |
US20120183577A1 (en) | 2012-07-19 |
US8017619B2 (en) | 2011-09-13 |
DE602004024572D1 (de) | 2010-01-21 |
CN1897950A (zh) | 2007-01-17 |
CN101824043A (zh) | 2010-09-08 |
WO2005037843A1 (en) | 2005-04-28 |
US20100280026A1 (en) | 2010-11-04 |
JP2011241231A (ja) | 2011-12-01 |
ATE451376T1 (de) | 2009-12-15 |
US7700609B2 (en) | 2010-04-20 |
US20050148603A1 (en) | 2005-07-07 |
AU2004282172A1 (en) | 2005-04-28 |
ES2338234T3 (es) | 2010-05-05 |
US8288400B2 (en) | 2012-10-16 |
EP1692140B1 (en) | 2009-12-09 |
EP1692140A1 (en) | 2006-08-23 |
CA2542113A1 (en) | 2005-04-28 |
AU2004282172B2 (en) | 2011-03-10 |
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