HK1072432A1 - Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands - Google Patents

Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands

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Publication number
HK1072432A1
HK1072432A1 HK05105957.5A HK05105957A HK1072432A1 HK 1072432 A1 HK1072432 A1 HK 1072432A1 HK 05105957 A HK05105957 A HK 05105957A HK 1072432 A1 HK1072432 A1 HK 1072432A1
Authority
HK
Hong Kong
Prior art keywords
thiadiazoleoxides
thiadiazoledioxides
cxc
chemokine receptor
receptor ligands
Prior art date
Application number
HK05105957.5A
Other languages
English (en)
Inventor
Arthur G Taveras
Cynthia J Aki
John J Baldwin
Ge Li
J Robert Merritt
Jianhua Chao
Younong Yu
Jay S Fine
Gaifa Lai
Minglang Wu
Purakkattle J Biju
William Hipkin
Evan A Hecker
Original Assignee
Pharmacopeia Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacopeia Inc filed Critical Pharmacopeia Inc
Publication of HK1072432A1 publication Critical patent/HK1072432A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
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HK05105957.5A 2002-10-09 2005-07-13 Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands HK1072432A1 (en)

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PE20040570A1 (es) 2004-08-30
ATE422203T1 (de) 2009-02-15
MY139601A (en) 2009-10-30
US7691856B2 (en) 2010-04-06
WO2004033440A1 (fr) 2004-04-22
WO2004033440A8 (fr) 2005-06-02
CN1720240B (zh) 2010-10-27
TW200413342A (en) 2004-08-01
US20040186142A1 (en) 2004-09-23
CN1720240A (zh) 2006-01-11
US20070264230A1 (en) 2007-11-15
CA2501535A1 (fr) 2004-04-22
JP2010270151A (ja) 2010-12-02
JP4664074B2 (ja) 2011-04-06
EP1551818A1 (fr) 2005-07-13
ES2321186T3 (es) 2009-06-03
AU2003288922A1 (en) 2004-05-04
EP1551818B1 (fr) 2009-02-04
DE60326080D1 (en) 2009-03-19
MXPA05003867A (es) 2005-11-23
JP2006508079A (ja) 2006-03-09
AR043052A1 (es) 2005-07-13

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