IL172026A0 - Cannabinoid receptor ligands and uses thereof - Google Patents
Cannabinoid receptor ligands and uses thereofInfo
- Publication number
- IL172026A0 IL172026A0 IL172026A IL17202605A IL172026A0 IL 172026 A0 IL172026 A0 IL 172026A0 IL 172026 A IL172026 A IL 172026A IL 17202605 A IL17202605 A IL 17202605A IL 172026 A0 IL172026 A0 IL 172026A0
- Authority
- IL
- Israel
- Prior art keywords
- receptor ligands
- cannabinoid receptor
- cannabinoid
- ligands
- receptor
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/10—Antiepileptics; Anticonvulsants for petit-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Child & Adolescent Psychology (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Nutrition Science (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrane Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US47694203P | 2003-06-09 | 2003-06-09 | |
PCT/IB2004/001888 WO2004108728A1 (en) | 2003-06-09 | 2004-06-03 | Cannabinoid receptor ligands and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
IL172026A0 true IL172026A0 (en) | 2009-02-11 |
Family
ID=33511826
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL172026A IL172026A0 (en) | 2003-06-09 | 2005-11-17 | Cannabinoid receptor ligands and uses thereof |
Country Status (21)
Country | Link |
---|---|
US (1) | US7232823B2 (en) |
EP (1) | EP1636233A1 (en) |
JP (1) | JP3917647B2 (en) |
KR (1) | KR20060007058A (en) |
CN (1) | CN1805963A (en) |
AP (1) | AP2005003466A0 (en) |
AU (1) | AU2004245316A1 (en) |
BR (1) | BRPI0411078A (en) |
CA (1) | CA2525752A1 (en) |
CO (1) | CO5640138A2 (en) |
EA (1) | EA200501771A1 (en) |
EC (1) | ECSP056208A (en) |
IL (1) | IL172026A0 (en) |
IS (1) | IS8137A (en) |
MA (1) | MA27853A1 (en) |
MX (1) | MXPA05013294A (en) |
NO (1) | NO20055731L (en) |
OA (1) | OA13172A (en) |
TN (1) | TNSN05317A1 (en) |
WO (1) | WO2004108728A1 (en) |
ZA (1) | ZA200509899B (en) |
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CN1875021A (en) * | 2003-11-04 | 2006-12-06 | 默克公司 | Substituted naphthyridinone derivatives |
US7151097B2 (en) | 2003-11-07 | 2006-12-19 | Pfizer Inc. | Bicyclic pyrazolyl and imidazolyl compounds and uses thereof |
RU2006118139A (en) * | 2003-12-02 | 2008-01-10 | Пфайзер Продактс Инк. (Us) | METHOD FOR CONVERTING HETEROCYCLIC KETONS TO AMIDOSubstituted HETEROCYCLES |
SG158168A1 (en) | 2004-12-23 | 2010-01-29 | Arena Pharm Inc | 5ht2c receptor modulator compositions and methods of use |
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WO2007003960A1 (en) * | 2005-06-30 | 2007-01-11 | Prosidion Limited | Gpcr agonists |
WO2007003962A2 (en) | 2005-06-30 | 2007-01-11 | Prosidion Limited | Gpcr agonists |
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BRPI0715160A2 (en) | 2006-08-08 | 2013-06-11 | Sanofi Aventis | arylamimoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, drugs comprising these compounds, and their use |
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CA2674360A1 (en) | 2007-01-04 | 2008-07-10 | Prosidion Limited | Piperidine gpcr agonists |
AR064735A1 (en) | 2007-01-04 | 2009-04-22 | Prosidion Ltd | GPCR AGONISTS AND PHARMACEUTICAL COMPOSITION BASED ON THE COMPOUND |
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GB0720390D0 (en) | 2007-10-18 | 2007-11-28 | Prosidion Ltd | G-Protein coupled receptor agonists |
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US8822727B2 (en) * | 2008-03-04 | 2014-09-02 | Arena Pharmaceuticals, Inc. | Processes for the preparation of intermediates related to the 5-HT2C agonist (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine |
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2004
- 2004-05-25 US US10/853,993 patent/US7232823B2/en not_active Expired - Fee Related
- 2004-06-03 AP AP2005003466A patent/AP2005003466A0/en unknown
- 2004-06-03 EA EA200501771A patent/EA200501771A1/en unknown
- 2004-06-03 BR BRPI0411078-1A patent/BRPI0411078A/en not_active IP Right Cessation
- 2004-06-03 CN CNA2004800161597A patent/CN1805963A/en active Pending
- 2004-06-03 KR KR1020057023720A patent/KR20060007058A/en active IP Right Grant
- 2004-06-03 OA OA1200500337A patent/OA13172A/en unknown
- 2004-06-03 JP JP2006516518A patent/JP3917647B2/en not_active Expired - Fee Related
- 2004-06-03 WO PCT/IB2004/001888 patent/WO2004108728A1/en active Application Filing
- 2004-06-03 CA CA002525752A patent/CA2525752A1/en not_active Abandoned
- 2004-06-03 EP EP04735931A patent/EP1636233A1/en not_active Withdrawn
- 2004-06-03 MX MXPA05013294A patent/MXPA05013294A/en unknown
- 2004-06-03 AU AU2004245316A patent/AU2004245316A1/en not_active Abandoned
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2005
- 2005-11-17 IL IL172026A patent/IL172026A0/en unknown
- 2005-11-21 IS IS8137A patent/IS8137A/en unknown
- 2005-12-05 NO NO20055731A patent/NO20055731L/en not_active Application Discontinuation
- 2005-12-06 ZA ZA200509899A patent/ZA200509899B/en unknown
- 2005-12-07 CO CO05124315A patent/CO5640138A2/en not_active Application Discontinuation
- 2005-12-09 MA MA28651A patent/MA27853A1/en unknown
- 2005-12-09 TN TNP2005000317A patent/TNSN05317A1/en unknown
- 2005-12-09 EC EC2005006208A patent/ECSP056208A/en unknown
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ZA200509899B (en) | 2006-12-27 |
KR20060007058A (en) | 2006-01-23 |
NO20055731L (en) | 2006-02-06 |
EA200501771A1 (en) | 2006-06-30 |
CA2525752A1 (en) | 2004-12-16 |
MXPA05013294A (en) | 2006-03-09 |
CO5640138A2 (en) | 2006-05-31 |
CN1805963A (en) | 2006-07-19 |
OA13172A (en) | 2006-12-13 |
AU2004245316A1 (en) | 2004-12-16 |
WO2004108728A1 (en) | 2004-12-16 |
IS8137A (en) | 2005-11-21 |
NO20055731D0 (en) | 2005-12-05 |
BRPI0411078A (en) | 2006-07-25 |
TNSN05317A1 (en) | 2007-07-10 |
US20040248881A1 (en) | 2004-12-09 |
EP1636233A1 (en) | 2006-03-22 |
JP3917647B2 (en) | 2007-05-23 |
ECSP056208A (en) | 2006-04-19 |
JP2006527262A (en) | 2006-11-30 |
US7232823B2 (en) | 2007-06-19 |
AP2005003466A0 (en) | 2005-12-31 |
MA27853A1 (en) | 2006-04-03 |
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