HK1051039A1 - Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase. - Google Patents

Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase.

Info

Publication number
HK1051039A1
HK1051039A1 HK03103208A HK03103208A HK1051039A1 HK 1051039 A1 HK1051039 A1 HK 1051039A1 HK 03103208 A HK03103208 A HK 03103208A HK 03103208 A HK03103208 A HK 03103208A HK 1051039 A1 HK1051039 A1 HK 1051039A1
Authority
HK
Hong Kong
Prior art keywords
heteroalkylamino
inhibitors
protein kinase
substituted bicyclic
nitrogen heterocycles
Prior art date
Application number
HK03103208A
Other languages
English (en)
Inventor
James Patrick Dunn
Lawrence Emerson Fisher
David Michael Goldstein
William Harris
Christopher Huw Hill
Ian Edward David Smith
Teresa Rosanne Welch
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HK1051039A1 publication Critical patent/HK1051039A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
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HK03103208A 1999-10-21 2003-05-06 Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase. HK1051039A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16080399P 1999-10-21 1999-10-21
US21374300P 2000-06-22 2000-06-22
PCT/EP2000/010088 WO2001029042A1 (en) 1999-10-21 2000-10-13 Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase

Publications (1)

Publication Number Publication Date
HK1051039A1 true HK1051039A1 (en) 2003-07-18

Family

ID=26857240

Family Applications (1)

Application Number Title Priority Date Filing Date
HK03103208A HK1051039A1 (en) 1999-10-21 2003-05-06 Heteroalkylamino-substituted bicyclic nitrogen heterocycles as inhibitors of p38 protein kinase.

Country Status (27)

Country Link
US (1) US6451804B1 (pl)
EP (1) EP1228070B1 (pl)
JP (1) JP3961830B2 (pl)
KR (1) KR100523120B1 (pl)
CN (1) CN1171889C (pl)
AR (1) AR026084A1 (pl)
AT (1) ATE353329T1 (pl)
AU (1) AU776250B2 (pl)
BR (1) BR0015243A (pl)
CA (1) CA2388142C (pl)
CZ (1) CZ20021744A3 (pl)
DE (1) DE60033307T2 (pl)
ES (1) ES2280247T3 (pl)
HK (1) HK1051039A1 (pl)
HR (1) HRP20020328A2 (pl)
HU (1) HUP0203564A3 (pl)
IL (1) IL149100A0 (pl)
MA (1) MA26837A1 (pl)
MX (1) MXPA02003950A (pl)
NO (1) NO20021781L (pl)
NZ (1) NZ518119A (pl)
PE (1) PE20010758A1 (pl)
PL (1) PL357502A1 (pl)
RU (1) RU2265606C2 (pl)
TR (1) TR200201057T2 (pl)
WO (1) WO2001029042A1 (pl)
YU (1) YU29102A (pl)

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GB2452696B (en) * 2007-08-02 2009-09-23 Cambridge Entpr Ltd 3-(2',2'-dimethylpropanoylamino)-tetrahydropyridin-2-one and its use in pharmaceutical compositions
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EP2113503A1 (en) 2008-04-28 2009-11-04 Laboratorios Almirall, S.A. New substituted indolin-2-one derivatives and their use as p39 mitogen-activated kinase inhibitors
CA2774040C (en) 2009-09-30 2014-09-09 Toray Industries, Inc. 2, 3-dihydro-1h-inden-2-yl urea derivatives and medical uses thereof
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