GT200600341A - Inhibidores macrociclicos del virus de la hepatitis c - Google Patents

Inhibidores macrociclicos del virus de la hepatitis c

Info

Publication number
GT200600341A
GT200600341A GT200600341A GT200600341A GT200600341A GT 200600341 A GT200600341 A GT 200600341A GT 200600341 A GT200600341 A GT 200600341A GT 200600341 A GT200600341 A GT 200600341A GT 200600341 A GT200600341 A GT 200600341A
Authority
GT
Guatemala
Prior art keywords
inhibitors
macrociclic
hepatitis
virus
formula
Prior art date
Application number
GT200600341A
Other languages
English (en)
Inventor
Pierre Jean-Marie Raboisson
Kock Herman Augustinus De
Sandrine Marie Hele Vendeville
Lili Hu
Vreken Wim Van De
David Craig Mcgowan
Abdellah Thari
Dominique Louis Nestor Surleraux
Kenneth Alan Simmen
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37036843&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200600341(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of GT200600341A publication Critical patent/GT200600341A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • C07K5/06165Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof

Abstract

LA INVENCIÓN SE REFIERE A INHIBIDORES DEL VHC DE FÓRMULA (I), LOS N-ÓXIDOS, SALES Y FORMAS ESTEREOQUÌMICAMENTE ISOMÉRICAS DE ÉSTOS, COMPOSICIONES FARMACÉUTICAS QUE CONTIENEN COMPUESTOS (I) Y PROCESOS PARA PREPARAR LOS COMPUESTOS (I). TAMBIÉN SE PROPORCIONAN COMBINACIONES BIODISPONIBLES DE LOS INHIBIDORES DEL VHC DE FÓRMULA (I) CON RITONAVIR.
GT200600341A 2005-07-29 2006-07-28 Inhibidores macrociclicos del virus de la hepatitis c GT200600341A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05107067 2005-07-29
EP05107413 2005-08-11

Publications (1)

Publication Number Publication Date
GT200600341A true GT200600341A (es) 2007-02-26

Family

ID=37036843

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600341A GT200600341A (es) 2005-07-29 2006-07-28 Inhibidores macrociclicos del virus de la hepatitis c

Country Status (28)

Country Link
US (1) US7989471B2 (es)
EP (1) EP1912995B1 (es)
JP (1) JP5426163B2 (es)
KR (1) KR101074673B1 (es)
CN (1) CN101233137B (es)
AP (1) AP2473A (es)
AR (1) AR055104A1 (es)
AT (1) ATE517902T1 (es)
AU (1) AU2006274858B2 (es)
BR (1) BRPI0614670A2 (es)
CA (1) CA2617095C (es)
DK (1) DK1912995T3 (es)
EA (1) EA014646B1 (es)
GT (1) GT200600341A (es)
HK (1) HK1116772A1 (es)
IL (1) IL188283A (es)
JO (1) JO2768B1 (es)
MX (1) MX2008001395A (es)
MY (1) MY152153A (es)
NO (1) NO20081071L (es)
NZ (1) NZ564541A (es)
PE (1) PE20070221A1 (es)
SG (1) SG163613A1 (es)
SI (1) SI1912995T1 (es)
SV (1) SV2008002639A (es)
TW (1) TWI412534B (es)
UY (1) UY29705A1 (es)
WO (1) WO2007014919A1 (es)

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Also Published As

Publication number Publication date
CN101233137A (zh) 2008-07-30
CA2617095C (en) 2014-05-13
MY152153A (en) 2014-08-15
KR20080041651A (ko) 2008-05-13
ATE517902T1 (de) 2011-08-15
EA014646B1 (ru) 2010-12-30
CA2617095A1 (en) 2007-02-08
US7989471B2 (en) 2011-08-02
DK1912995T3 (da) 2011-10-24
AP2473A (en) 2012-09-24
PE20070221A1 (es) 2007-04-16
SV2008002639A (es) 2008-07-23
IL188283A (en) 2016-12-29
US20100240698A1 (en) 2010-09-23
SG163613A1 (en) 2010-08-30
JP5426163B2 (ja) 2014-02-26
NZ564541A (en) 2010-03-26
JP2009502882A (ja) 2009-01-29
CN101233137B (zh) 2014-05-07
JO2768B1 (en) 2014-03-15
BRPI0614670A2 (pt) 2011-04-12
TWI412534B (zh) 2013-10-21
IL188283A0 (en) 2008-04-13
KR101074673B1 (ko) 2011-10-19
SI1912995T1 (sl) 2011-11-30
HK1116772A1 (en) 2009-01-02
EP1912995A1 (en) 2008-04-23
AR055104A1 (es) 2007-08-08
AU2006274858B2 (en) 2012-05-24
EP1912995B1 (en) 2011-07-27
EA200800484A1 (ru) 2008-06-30
NO20081071L (no) 2008-04-25
AU2006274858A1 (en) 2007-02-08
WO2007014919A1 (en) 2007-02-08
UY29705A1 (es) 2007-05-31
MX2008001395A (es) 2008-04-16
TW200745165A (en) 2007-12-16

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