GT200400248A - Proceso para la preparacion de inhibidores de tubulina - Google Patents
Proceso para la preparacion de inhibidores de tubulinaInfo
- Publication number
- GT200400248A GT200400248A GT200400248A GT200400248A GT200400248A GT 200400248 A GT200400248 A GT 200400248A GT 200400248 A GT200400248 A GT 200400248A GT 200400248 A GT200400248 A GT 200400248A GT 200400248 A GT200400248 A GT 200400248A
- Authority
- GT
- Guatemala
- Prior art keywords
- preparation
- tubulin inhibitors
- tubulin
- inhibitors
- pictures
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A UN COMPUESTO DE FORMULA GENERAL I EN LA QUE R1,R2,R3,R4,X, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON INHIBIDORES DE TUBULINA POR LO QUE SON DE UTILIDAD EN CUADROS DE CANCER.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52793103P | 2003-12-08 | 2003-12-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200400248A true GT200400248A (es) | 2005-09-14 |
Family
ID=34676796
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200400248A GT200400248A (es) | 2003-12-08 | 2004-12-03 | Proceso para la preparacion de inhibidores de tubulina |
Country Status (29)
Country | Link |
---|---|
US (1) | US7396835B2 (es) |
EP (1) | EP1692137B1 (es) |
JP (1) | JP2007513185A (es) |
KR (1) | KR20060094984A (es) |
CN (1) | CN1890245A (es) |
AR (1) | AR046939A1 (es) |
AT (1) | ATE356128T1 (es) |
AU (1) | AU2004297244A1 (es) |
BR (1) | BRPI0417422A (es) |
CA (1) | CA2546899A1 (es) |
CO (1) | CO5700827A2 (es) |
CR (1) | CR8435A (es) |
DE (1) | DE602004005239T2 (es) |
DK (1) | DK1692137T3 (es) |
EC (1) | ECSP066606A (es) |
ES (1) | ES2281850T3 (es) |
GT (1) | GT200400248A (es) |
HK (1) | HK1090377A1 (es) |
IL (1) | IL175775A0 (es) |
MY (1) | MY179926A (es) |
NO (1) | NO20062492L (es) |
NZ (1) | NZ547471A (es) |
PA (1) | PA8619401A1 (es) |
PE (1) | PE20050593A1 (es) |
PL (1) | PL1692137T3 (es) |
RU (1) | RU2006117023A (es) |
TW (1) | TW200522963A (es) |
WO (1) | WO2005056560A1 (es) |
ZA (1) | ZA200604680B (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6255309B1 (en) * | 1999-03-19 | 2001-07-03 | American Cyanomid Co. | Fungicidal trifluoromethylalkylamino-triazolopyrimidines |
US7419982B2 (en) * | 2003-09-24 | 2008-09-02 | Wyeth Holdings Corporation | Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts |
TW200800959A (en) | 2005-06-10 | 2008-01-01 | Wyeth Corp | Piperazine-piperidine antagonists and agonists of the 5-HT1a receptor |
TW200808730A (en) * | 2006-06-09 | 2008-02-16 | Wyeth Corp | Process for synthesizing piperazine-piperidine compounds |
US20100056371A1 (en) * | 2007-01-08 | 2010-03-04 | Basf Se | Use of Azolopyrimidines for Controlling Phytopathogenic Harmful Fungi |
US9649317B2 (en) | 2012-09-19 | 2017-05-16 | The Trustees Of The University Of Pennsylvania | Heterocyclic compounds and their use for the treatment of neurodegenerative tauopathies |
US11623927B2 (en) | 2018-03-02 | 2023-04-11 | The Trustees Of The University Of Pennsylvania | Substituted [1,2,4]triazolo[1,5-a]pyrimidines for stabilizing microtubules |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW224044B (es) | 1991-12-30 | 1994-05-21 | Shell Internat Res Schappej B V | |
US5593996A (en) | 1991-12-30 | 1997-01-14 | American Cyanamid Company | Triazolopyrimidine derivatives |
JP2794510B2 (ja) | 1992-03-27 | 1998-09-10 | 富士写真フイルム株式会社 | ハロゲン化銀写真感光材料 |
IL108731A (en) | 1993-03-04 | 1997-03-18 | Shell Int Research | 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES |
IL108747A (en) | 1993-03-04 | 1999-03-12 | Shell Int Research | Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation |
RU2147584C1 (ru) | 1995-10-27 | 2000-04-20 | Американ Цианамид Компани | Способ получения дигалоидазолопиримидинов и способ получения дигидроксиазолопиримидинов |
US5817663A (en) | 1996-10-07 | 1998-10-06 | American Cyanamid Company | Pentafluorophenylazolopyrimidines |
US5750766A (en) | 1997-03-18 | 1998-05-12 | American Cyanamid Company | Process for the preparation of arylmalonates |
AU6558498A (en) | 1997-03-18 | 1998-10-12 | American Cyanamid Company | Process for the preparation of arylmalonates |
US5948783A (en) | 1997-04-14 | 1999-09-07 | American Cyanamid Company | Fungicidal trifluoromethylalkylamino-triazolopyrimidines |
TWI252231B (en) | 1997-04-14 | 2006-04-01 | American Cyanamid Co | Fungicidal trifluorophenyl-triazolopyrimidines |
TW460476B (en) | 1997-04-14 | 2001-10-21 | American Cyanamid Co | Fungicidal trifluoromethylalkylamino-triazolopyrimidines |
US6117876A (en) * | 1997-04-14 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
US5994360A (en) | 1997-07-14 | 1999-11-30 | American Cyanamid Company | Fungicidal 5-alkyl-triazolopyrimidines |
US5986153A (en) | 1997-09-30 | 1999-11-16 | Phillips Petroleum Company | Olefin color stabilization |
US6020338A (en) | 1998-02-11 | 2000-02-01 | American Cyanamid Company | Fungicidal 7-alkyl-triazolopyrimidines |
WO1999048893A1 (en) * | 1998-03-23 | 1999-09-30 | American Cyanamid Company | Fungicidal 6-(2-halo-4-alkoxyphenyl)-triazolopyrimidines |
US5981534A (en) | 1998-09-25 | 1999-11-09 | American Cyanamid Company | Fungicidal 6-(2,6-difluoro-4-alkoxyphenyl)-triazolopyrimidines |
US5985883A (en) | 1998-09-25 | 1999-11-16 | American Cyanamid Company | Fungicidal trichlorophenyl-triazolopyrimidines |
JP2000103790A (ja) | 1998-09-25 | 2000-04-11 | American Cyanamid Co | 殺菌・殺カビ性のトリハロフェニル―トリアゾロピリミジン類 |
US6242451B1 (en) | 1998-09-25 | 2001-06-05 | Klaus-Juergen Pees | Fungicidal trihalophenyl-triazolopyrimidines |
US5986135A (en) | 1998-09-25 | 1999-11-16 | American Cyanamid Company | Fungicidal trifluoromethylalkylamino-triazolopyrimidines |
NZ523807A (en) | 2000-06-30 | 2004-09-24 | Wyeth Corp | Substituted-triazolopyrimidines as anticancer agents |
SI1680425T1 (sl) * | 2003-09-24 | 2007-04-30 | Wyeth Corp | 6-((substituirani)fenil)triazolopirimidini kot sredstva proti raku |
CN101193884A (zh) * | 2005-06-13 | 2008-06-04 | 惠氏公司 | 微管蛋白抑制剂和其制备方法 |
-
2004
- 2004-12-02 MY MYPI20044999A patent/MY179926A/en unknown
- 2004-12-03 TW TW093137287A patent/TW200522963A/zh unknown
- 2004-12-03 GT GT200400248A patent/GT200400248A/es unknown
- 2004-12-07 PE PE2004001201A patent/PE20050593A1/es not_active Application Discontinuation
- 2004-12-07 DE DE602004005239T patent/DE602004005239T2/de not_active Expired - Fee Related
- 2004-12-07 EP EP04813203A patent/EP1692137B1/en active Active
- 2004-12-07 KR KR1020067012134A patent/KR20060094984A/ko not_active Application Discontinuation
- 2004-12-07 RU RU2006117023/04A patent/RU2006117023A/ru not_active Application Discontinuation
- 2004-12-07 PA PA20048619401A patent/PA8619401A1/es unknown
- 2004-12-07 ES ES04813203T patent/ES2281850T3/es active Active
- 2004-12-07 AU AU2004297244A patent/AU2004297244A1/en not_active Withdrawn
- 2004-12-07 BR BRPI0417422-4A patent/BRPI0417422A/pt not_active IP Right Cessation
- 2004-12-07 AR ARP040104569A patent/AR046939A1/es not_active Application Discontinuation
- 2004-12-07 JP JP2006542867A patent/JP2007513185A/ja not_active Withdrawn
- 2004-12-07 PL PL04813203T patent/PL1692137T3/pl unknown
- 2004-12-07 WO PCT/US2004/040854 patent/WO2005056560A1/en active IP Right Grant
- 2004-12-07 DK DK04813203T patent/DK1692137T3/da active
- 2004-12-07 CA CA002546899A patent/CA2546899A1/en not_active Abandoned
- 2004-12-07 CN CNA2004800362897A patent/CN1890245A/zh active Pending
- 2004-12-07 NZ NZ547471A patent/NZ547471A/en unknown
- 2004-12-07 AT AT04813203T patent/ATE356128T1/de not_active IP Right Cessation
- 2004-12-08 US US11/007,839 patent/US7396835B2/en not_active Expired - Fee Related
-
2006
- 2006-05-18 IL IL175775A patent/IL175775A0/en unknown
- 2006-05-31 NO NO20062492A patent/NO20062492L/no not_active Application Discontinuation
- 2006-06-05 EC EC2006006606A patent/ECSP066606A/es unknown
- 2006-06-06 CR CR8435A patent/CR8435A/es not_active Application Discontinuation
- 2006-06-07 ZA ZA200604680A patent/ZA200604680B/xx unknown
- 2006-06-08 CO CO06055468A patent/CO5700827A2/es not_active Application Discontinuation
- 2006-11-02 HK HK06112063A patent/HK1090377A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ES2281850T3 (es) | 2007-10-01 |
DE602004005239T2 (de) | 2007-12-20 |
CN1890245A (zh) | 2007-01-03 |
CR8435A (es) | 2007-06-08 |
ZA200604680B (en) | 2009-04-29 |
PA8619401A1 (es) | 2005-08-04 |
US7396835B2 (en) | 2008-07-08 |
DK1692137T3 (da) | 2007-04-30 |
RU2006117023A (ru) | 2008-01-20 |
DE602004005239D1 (de) | 2007-04-19 |
AR046939A1 (es) | 2006-01-04 |
CO5700827A2 (es) | 2006-11-30 |
ECSP066606A (es) | 2006-10-25 |
TW200522963A (en) | 2005-07-16 |
US20050124635A1 (en) | 2005-06-09 |
MY179926A (en) | 2020-11-19 |
HK1090377A1 (en) | 2006-12-22 |
PE20050593A1 (es) | 2005-09-27 |
IL175775A0 (en) | 2006-09-05 |
KR20060094984A (ko) | 2006-08-30 |
AU2004297244A1 (en) | 2005-06-23 |
NO20062492L (no) | 2006-07-03 |
JP2007513185A (ja) | 2007-05-24 |
PL1692137T3 (pl) | 2007-06-29 |
BRPI0417422A (pt) | 2007-03-13 |
EP1692137B1 (en) | 2007-03-07 |
EP1692137A1 (en) | 2006-08-23 |
CA2546899A1 (en) | 2005-06-23 |
NZ547471A (en) | 2009-03-31 |
WO2005056560A1 (en) | 2005-06-23 |
ATE356128T1 (de) | 2007-03-15 |
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