GEP201706780B - Substituted 2-aza-bicyclo [2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin c - Google Patents

Substituted 2-aza-bicyclo [2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin c

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Publication number
GEP201706780B
GEP201706780B GEAP201413959A GEAP2014013959A GEP201706780B GE P201706780 B GEP201706780 B GE P201706780B GE AP201413959 A GEAP201413959 A GE AP201413959A GE AP2014013959 A GEAP2014013959 A GE AP2014013959A GE P201706780 B GEP201706780 B GE P201706780B
Authority
GE
Georgia
Prior art keywords
cathepsin
aza
bicyclo
heptane
cyano
Prior art date
Application number
GEAP201413959A
Other languages
English (en)
Inventor
Ralf Anderskewitz
Matthias Grauert
Marc Grauert
Peter Wilhelm Haebel
Thorsten Oost
Alexander Pautsch
Stefan Peters
Florian Binder
Viktor Vintonyak
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of GEP201706780B publication Critical patent/GEP201706780B/en

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    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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