FR2400511A1 - N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique - Google Patents
N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastriqueInfo
- Publication number
- FR2400511A1 FR2400511A1 FR7824138A FR7824138A FR2400511A1 FR 2400511 A1 FR2400511 A1 FR 2400511A1 FR 7824138 A FR7824138 A FR 7824138A FR 7824138 A FR7824138 A FR 7824138A FR 2400511 A1 FR2400511 A1 FR 2400511A1
- Authority
- FR
- France
- Prior art keywords
- benzamides
- pyrazolidinyl
- antiemetic
- presenting
- gastric emptying
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- -1 4-PYRAZOLIDINYL Chemical class 0.000 title 1
- 230000003474 anti-emetic effect Effects 0.000 title 1
- 239000002111 antiemetic agent Substances 0.000 title 1
- 229940054066 benzamide antipsychotics Drugs 0.000 title 1
- 150000003936 benzamides Chemical class 0.000 title 1
- 230000030136 gastric emptying Effects 0.000 title 1
- WSKUIBCWQOEKLC-UHFFFAOYSA-N 4-pyrazolidin-1-ylbenzamide Chemical class N1(NCCC1)C1=CC=C(C(=O)N)C=C1 WSKUIBCWQOEKLC-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Otolaryngology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82603177A | 1977-08-19 | 1977-08-19 | |
| US90036978A | 1978-04-26 | 1978-04-26 | |
| US93012578A | 1978-08-01 | 1978-08-01 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2400511A1 true FR2400511A1 (fr) | 1979-03-16 |
| FR2400511B1 FR2400511B1 (en17) | 1981-09-04 |
Family
ID=27420183
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7824138A Granted FR2400511A1 (fr) | 1977-08-19 | 1978-08-18 | N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique |
Country Status (21)
| Country | Link |
|---|---|
| JP (1) | JPS5441873A (en17) |
| AU (1) | AU521421B2 (en17) |
| BR (1) | BR7805288A (en17) |
| CA (1) | CA1105037A (en17) |
| CH (2) | CH639374A5 (en17) |
| DE (1) | DE2836062A1 (en17) |
| DK (1) | DK152361C (en17) |
| ES (1) | ES472686A1 (en17) |
| FI (1) | FI68044C (en17) |
| FR (1) | FR2400511A1 (en17) |
| GB (2) | GB2003153B (en17) |
| HK (1) | HK42282A (en17) |
| IE (1) | IE47430B1 (en17) |
| MX (1) | MX5469E (en17) |
| NL (1) | NL7808596A (en17) |
| NO (1) | NO149107C (en17) |
| NZ (1) | NZ188189A (en17) |
| PH (1) | PH13331A (en17) |
| PT (1) | PT68442A (en17) |
| SE (2) | SE444434B (en17) |
| YU (1) | YU41116B (en17) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2490639A1 (fr) * | 1980-08-07 | 1982-03-26 | Robins Co Inc A H | Nouveau procede pour la synthese de 4-amino-1,2-dihydrocarbylpyrazolidines par l'intermediaire des analogues 4-nitro |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5126343A (en) * | 1989-09-11 | 1992-06-30 | G. D. Searle & Co. | N-azabicyclo [3.3.0]octane amides of aromatic acids |
| JP3065506B2 (ja) * | 1995-04-03 | 2000-07-17 | 株式会社資生堂 | ピラゾリジン誘導体及びラジカルスカベンジャー、脳梗塞抑制剤、脳浮腫抑制剤 |
| AR086587A1 (es) | 2011-05-31 | 2014-01-08 | Syngenta Participations Ag | Compuestos insecticidas |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3966957A (en) * | 1972-04-03 | 1976-06-29 | A. H. Robins Company, Incorporated | Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides |
-
1976
- 1976-08-14 PH PH21489A patent/PH13331A/en unknown
-
1978
- 1978-08-15 CH CH867478A patent/CH639374A5/fr not_active IP Right Cessation
- 1978-08-16 FI FI782507A patent/FI68044C/fi not_active IP Right Cessation
- 1978-08-16 SE SE7808694A patent/SE444434B/sv not_active IP Right Cessation
- 1978-08-17 GB GB7833696A patent/GB2003153B/en not_active Expired
- 1978-08-17 BR BR7805288A patent/BR7805288A/pt unknown
- 1978-08-17 DE DE19782836062 patent/DE2836062A1/de not_active Withdrawn
- 1978-08-17 GB GB7901821A patent/GB2017678B/en not_active Expired
- 1978-08-18 IE IE1682/78A patent/IE47430B1/en unknown
- 1978-08-18 NZ NZ188189A patent/NZ188189A/en unknown
- 1978-08-18 PT PT68442A patent/PT68442A/pt unknown
- 1978-08-18 MX MX787322U patent/MX5469E/es unknown
- 1978-08-18 DK DK366978A patent/DK152361C/da not_active IP Right Cessation
- 1978-08-18 NL NL7808596A patent/NL7808596A/xx not_active Application Discontinuation
- 1978-08-18 YU YU1986/78A patent/YU41116B/xx unknown
- 1978-08-18 CA CA309,651A patent/CA1105037A/en not_active Expired
- 1978-08-18 FR FR7824138A patent/FR2400511A1/fr active Granted
- 1978-08-18 NO NO782812A patent/NO149107C/no unknown
- 1978-08-18 AU AU39061/78A patent/AU521421B2/en not_active Expired
- 1978-08-18 ES ES472686A patent/ES472686A1/es not_active Expired
- 1978-08-19 JP JP10136878A patent/JPS5441873A/ja active Granted
-
1982
- 1982-09-30 HK HK422/82A patent/HK42282A/xx unknown
-
1983
- 1983-04-28 CH CH228983A patent/CH645356A5/fr not_active IP Right Cessation
- 1983-06-21 SE SE8303564A patent/SE451723B/sv not_active IP Right Cessation
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2490639A1 (fr) * | 1980-08-07 | 1982-03-26 | Robins Co Inc A H | Nouveau procede pour la synthese de 4-amino-1,2-dihydrocarbylpyrazolidines par l'intermediaire des analogues 4-nitro |
| FR2491065A1 (fr) * | 1980-08-07 | 1982-04-02 | Robins Co Inc A H | Nouveau procede pour la synthese de 4-nitro-1,2-dihydrocarbyl-pyrazolidines, et produits obtenus |
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |