FI951593A0 - Uusi menetelmä bakkatiini-III:n ja 10-desasetyylibakkatiini-III:n esteröimiseksi - Google Patents

Uusi menetelmä bakkatiini-III:n ja 10-desasetyylibakkatiini-III:n esteröimiseksi

Info

Publication number
FI951593A0
FI951593A0 FI951593A FI951593A FI951593A0 FI 951593 A0 FI951593 A0 FI 951593A0 FI 951593 A FI951593 A FI 951593A FI 951593 A FI951593 A FI 951593A FI 951593 A0 FI951593 A0 FI 951593A0
Authority
FI
Finland
Prior art keywords
iii
radical
pct
formula
image
Prior art date
Application number
FI951593A
Other languages
English (en)
Swedish (sv)
Other versions
FI951593A (fi
FI115909B (fi
Inventor
Jean-Noel Denis
Andrew Greene
Jean Manuel Mas
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of FI951593A publication Critical patent/FI951593A/fi
Publication of FI951593A0 publication Critical patent/FI951593A0/fi
Application granted granted Critical
Publication of FI115909B publication Critical patent/FI115909B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epoxy Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
FI951593A 1992-10-05 1995-04-04 Uusi menetelmä bakkatiini-III:n ja 10-desasetyylibakkatiini-III:n esteröimiseksi FI115909B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9211739 1992-10-05
FR9211739A FR2696464B1 (fr) 1992-10-05 1992-10-05 Nouveau procédé d'estérification de la baccatine III et de la désacétyl-10 baccatine III.
FR9300965 1993-10-04
PCT/FR1993/000965 WO1994007876A1 (fr) 1992-10-05 1993-10-04 Nouveau procede d'esterification de la baccatine iii et de la desacetyl-10 baccatine iii

Publications (3)

Publication Number Publication Date
FI951593A FI951593A (fi) 1995-04-04
FI951593A0 true FI951593A0 (fi) 1995-04-04
FI115909B FI115909B (fi) 2005-08-15

Family

ID=9434116

Family Applications (1)

Application Number Title Priority Date Filing Date
FI951593A FI115909B (fi) 1992-10-05 1995-04-04 Uusi menetelmä bakkatiini-III:n ja 10-desasetyylibakkatiini-III:n esteröimiseksi

Country Status (24)

Country Link
US (2) US5717103A (fi)
EP (1) EP0663905B1 (fi)
JP (1) JP3064419B2 (fi)
KR (1) KR100290663B1 (fi)
AT (1) ATE147734T1 (fi)
AU (1) AU689446B2 (fi)
CA (1) CA2146372C (fi)
CZ (1) CZ284818B6 (fi)
DE (1) DE69307526T2 (fi)
DK (1) DK0663905T3 (fi)
ES (1) ES2096328T3 (fi)
FI (1) FI115909B (fi)
FR (1) FR2696464B1 (fi)
GR (1) GR3022286T3 (fi)
HU (1) HU225973B1 (fi)
MX (1) MX9305764A (fi)
NO (1) NO313141B1 (fi)
NZ (1) NZ256443A (fi)
PL (1) PL178090B1 (fi)
RU (1) RU2123493C1 (fi)
SK (1) SK281035B6 (fi)
TW (1) TW372234B (fi)
WO (1) WO1994007876A1 (fi)
ZA (1) ZA937316B (fi)

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FR2698361B1 (fr) * 1992-11-20 1995-01-13 Rhone Poulenc Rorer Sa Procédé de préparation d'un acide oxazolidine-1,3 carboxylique-5.
MX9307777A (es) 1992-12-15 1994-07-29 Upjohn Co 7-HALO-Y 7ß, 8ß-METANO-TAXOLES, USO ANTINEOPLASTICO Y COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN.
DK0703909T3 (da) * 1993-06-11 2000-09-11 Upjohn Co Delta6,7-taxoler, antineoplastisk anvendelse og farmaceutiske præparater indeholdende dem
ATE420628T1 (de) 1993-07-19 2009-01-15 Angiotech Pharm Inc Anti-angiogene mittel und verfahren zu deren verwendung
WO1995013267A1 (en) * 1993-11-12 1995-05-18 The Upjohn Company Pyrimidine-thioalkyl and alkylether compounds
IL112412A (en) * 1994-01-28 2000-02-29 Upjohn Co Delta 12,13-iso-taxol analogs and antineoplastic pharmaceutical compositions containing them
CA2178541C (en) 1995-06-07 2009-11-24 Neal E. Fearnot Implantable medical device
CN1216039A (zh) * 1996-05-08 1999-05-05 法玛西雅厄普约翰美国公司 制备紫杉酚的方法
US6150537A (en) * 1997-12-12 2000-11-21 Emory University Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
JP4502338B2 (ja) * 1999-09-17 2010-07-14 株式会社横浜国際バイオ研究所 タキソイド化合物の製造法
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US7351542B2 (en) 2002-05-20 2008-04-01 The Regents Of The University Of California Methods of modulating tubulin deacetylase activity
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Family Cites Families (7)

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Publication number Priority date Publication date Assignee Title
US34277A (en) * 1862-01-28 Improvement in lamps
US4942184A (en) * 1988-03-07 1990-07-17 The United States Of America As Represented By The Department Of Health And Human Services Water soluble, antineoplastic derivatives of taxol
FR2629818B1 (fr) * 1988-04-06 1990-11-16 Centre Nat Rech Scient Procede de preparation du taxol
USRE34277E (en) * 1988-04-06 1993-06-08 Centre National De La Recherche Scientifique Process for preparing taxol
MX9102128A (es) * 1990-11-23 1992-07-08 Rhone Poulenc Rorer Sa Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene
FR2696460B1 (fr) * 1992-10-05 1994-11-25 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2696458B1 (fr) * 1992-10-05 1994-11-10 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.

Also Published As

Publication number Publication date
CZ284818B6 (cs) 1999-03-17
HUT72616A (en) 1996-05-28
MX9305764A (es) 1995-01-31
NZ256443A (en) 1996-07-26
KR100290663B1 (ko) 2001-09-17
EP0663905B1 (fr) 1997-01-15
CZ83995A3 (en) 1995-09-13
US5717103A (en) 1998-02-10
ATE147734T1 (de) 1997-02-15
FR2696464A1 (fr) 1994-04-08
EP0663905A1 (fr) 1995-07-26
DE69307526T2 (de) 1997-05-22
ZA937316B (en) 1994-04-22
KR950703545A (ko) 1995-09-20
HU9500970D0 (en) 1995-06-28
CA2146372C (fr) 2003-09-09
AU5114893A (en) 1994-04-26
FR2696464B1 (fr) 1994-11-10
FI951593A (fi) 1995-04-04
NO313141B1 (no) 2002-08-19
FI115909B (fi) 2005-08-15
PL178090B1 (pl) 2000-02-29
GR3022286T3 (en) 1997-04-30
HU225973B1 (en) 2008-02-28
RU95110766A (ru) 1996-12-27
RU2123493C1 (ru) 1998-12-20
TW372234B (en) 1999-10-21
WO1994007876A1 (fr) 1994-04-14
JP3064419B2 (ja) 2000-07-12
US5977375A (en) 1999-11-02
SK43895A3 (en) 1995-08-09
NO951200D0 (no) 1995-03-29
DK0663905T3 (da) 1997-02-03
DE69307526D1 (de) 1997-02-27
CA2146372A1 (fr) 1994-04-14
JPH08501787A (ja) 1996-02-27
NO951200L (no) 1995-03-29
PL308239A1 (en) 1995-07-24
ES2096328T3 (es) 1997-03-01
SK281035B6 (sk) 2000-11-07
AU689446B2 (en) 1998-04-02

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