FI941829A - (S)-4-(4-dimetylamino)-1-(4'-fluorfenyl)-1-(hydroxibutyl)bensonitrilderivat - Google Patents

(S)-4-(4-dimetylamino)-1-(4'-fluorfenyl)-1-(hydroxibutyl)bensonitrilderivat Download PDF

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Publication number
FI941829A
FI941829A FI941829A FI941829A FI941829A FI 941829 A FI941829 A FI 941829A FI 941829 A FI941829 A FI 941829A FI 941829 A FI941829 A FI 941829A FI 941829 A FI941829 A FI 941829A
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FI
Finland
Prior art keywords
fluorophenyl
benzonitrile
hydroxybutyl
dimethylamino
geriatrics
Prior art date
Application number
FI941829A
Other languages
English (en)
Finnish (fi)
Other versions
FI113762B1 (sv
FI941829A0 (sv
Inventor
Klaus Peter Boegesoe
Jens Perregaard
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10638616&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI941829(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of FI941829A publication Critical patent/FI941829A/sv
Publication of FI941829A0 publication Critical patent/FI941829A0/sv
Application granted granted Critical
Publication of FI113762B1 publication Critical patent/FI113762B1/sv

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Psychiatry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Silicon Compounds (AREA)
FI941829A 1988-06-14 1994-04-20 (S)-4-[4-dimetylamino-1-(4'-fluorfenyl)-1-hydroxibutyl]bensonitrilderivat FI113762B1 (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888814057A GB8814057D0 (en) 1988-06-14 1988-06-14 New enantiomers & their isolation

Publications (3)

Publication Number Publication Date
FI941829A true FI941829A (sv) 1994-04-20
FI941829A0 FI941829A0 (sv) 1994-04-20
FI113762B1 FI113762B1 (sv) 2004-06-15

Family

ID=10638616

Family Applications (4)

Application Number Title Priority Date Filing Date
FI892823A FI98627C (sv) 1988-06-14 1989-06-08 Förfarande för framställning av en terapeutiskt användbar (S)-1-(3-dimetylaminopropyl)-1-(4'-fluorfenyl)-1,3-dihydrobensofuran-5-karbonitril
FI941829A FI113762B1 (sv) 1988-06-14 1994-04-20 (S)-4-[4-dimetylamino-1-(4'-fluorfenyl)-1-hydroxibutyl]bensonitrilderivat
FI20000507A FI20000507A (sv) 1988-06-14 2000-03-06 (+)-1-(3-dimetylaminopropyl)-1-(4'-fluorfenyl)-1,3-dihydroisobensofuran-5-karbonitril och farmaceutisk komposition som innehåller detta
FI20041359A FI20041359A (sv) 1988-06-14 2004-10-20 Diasteromeriskt salt av 4-{4-dimetylamino-1-('-fluorfenyl)-1-hydroxibutyl]benzonitril

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI892823A FI98627C (sv) 1988-06-14 1989-06-08 Förfarande för framställning av en terapeutiskt användbar (S)-1-(3-dimetylaminopropyl)-1-(4'-fluorfenyl)-1,3-dihydrobensofuran-5-karbonitril

Family Applications After (2)

Application Number Title Priority Date Filing Date
FI20000507A FI20000507A (sv) 1988-06-14 2000-03-06 (+)-1-(3-dimetylaminopropyl)-1-(4'-fluorfenyl)-1,3-dihydroisobensofuran-5-karbonitril och farmaceutisk komposition som innehåller detta
FI20041359A FI20041359A (sv) 1988-06-14 2004-10-20 Diasteromeriskt salt av 4-{4-dimetylamino-1-('-fluorfenyl)-1-hydroxibutyl]benzonitril

Country Status (24)

Country Link
US (2) US4943590A (sv)
EP (1) EP0347066B1 (sv)
JP (2) JP3044253B2 (sv)
AT (1) ATE119896T1 (sv)
AU (1) AU623144B2 (sv)
CA (2) CA1339452C (sv)
CY (2) CY2081B1 (sv)
DE (2) DE10399030I2 (sv)
DK (2) DK259989A (sv)
ES (1) ES2068891T4 (sv)
FI (4) FI98627C (sv)
GB (1) GB8814057D0 (sv)
GR (1) GR3015889T3 (sv)
HK (1) HK139596A (sv)
HU (1) HU211460A9 (sv)
IE (1) IE65734B1 (sv)
IL (1) IL90465A (sv)
LU (1) LU90999I2 (sv)
MX (1) MX9203346A (sv)
NL (1) NL300155I2 (sv)
NO (2) NO172892C (sv)
NZ (1) NZ229426A (sv)
PT (1) PT90845B (sv)
ZA (1) ZA894476B (sv)

Families Citing this family (146)

* Cited by examiner, † Cited by third party
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US6403657B1 (en) 1999-10-04 2002-06-11 Martin C. Hinz Comprehensive pharmacologic therapy for treatment of obesity
US6759437B2 (en) 1999-10-04 2004-07-06 Martin C. Hinz Comprehensive pharmacologic therapy for treatment of obesity including cysteine
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AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
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TR200201783T2 (tr) * 2000-01-14 2002-12-23 H. Lundbeck A/S 5-Siyanofatalid hazırlamak için yöntem
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KR20020080476A (ko) 2000-03-14 2002-10-23 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
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JP3038204B2 (ja) 2000-05-08
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