FI925767A0 - Dialkoxi-pyridinyl-bensimidazolderivater, foerfaranden foer deras framstaellning och deras farmaceutiska anvaendning - Google Patents

Dialkoxi-pyridinyl-bensimidazolderivater, foerfaranden foer deras framstaellning och deras farmaceutiska anvaendning

Info

Publication number
FI925767A0
FI925767A0 FI925767A FI925767A FI925767A0 FI 925767 A0 FI925767 A0 FI 925767A0 FI 925767 A FI925767 A FI 925767A FI 925767 A FI925767 A FI 925767A FI 925767 A0 FI925767 A0 FI 925767A0
Authority
FI
Finland
Prior art keywords
deras
pharmaceutiska
benzenimidazolderivater
anvaendning
dialkoxy
Prior art date
Application number
FI925767A
Other languages
English (en)
Finnish (fi)
Other versions
FI925767A (fi
Inventor
Arne Elof Braendstroem
Per Lennart Lindberg
Gunnel Elisabeth Sunden
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9002206A external-priority patent/SE9002206D0/xx
Priority claimed from SE9002207A external-priority patent/SE9002207D0/xx
Application filed by Astra Ab filed Critical Astra Ab
Publication of FI925767A publication Critical patent/FI925767A/fi
Publication of FI925767A0 publication Critical patent/FI925767A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI925767A 1990-06-20 1992-12-18 Dialkoxi-pyridinyl-bensimidazolderivater, foerfaranden foer deras framstaellning och deras farmaceutiska anvaendning FI925767A0 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9002206A SE9002206D0 (sv) 1990-06-20 1990-06-20 New compounds
SE9002207A SE9002207D0 (sv) 1990-06-20 1990-06-20 New compounds i
PCT/SE1991/000416 WO1991019712A1 (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use

Publications (2)

Publication Number Publication Date
FI925767A FI925767A (fi) 1992-12-18
FI925767A0 true FI925767A0 (fi) 1992-12-18

Family

ID=26660803

Family Applications (1)

Application Number Title Priority Date Filing Date
FI925767A FI925767A0 (fi) 1990-06-20 1992-12-18 Dialkoxi-pyridinyl-bensimidazolderivater, foerfaranden foer deras framstaellning och deras farmaceutiska anvaendning

Country Status (29)

Country Link
US (1) US5430042A (no)
EP (1) EP0593463B1 (no)
JP (1) JP3049367B2 (no)
CN (1) CN1058213A (no)
AP (1) AP253A (no)
AT (1) ATE184602T1 (no)
AU (1) AU649456B2 (no)
BG (1) BG97198A (no)
CA (1) CA2083606C (no)
CZ (1) CZ279434B6 (no)
DE (1) DE69131627T2 (no)
EG (1) EG19752A (no)
ES (1) ES2140391T3 (no)
FI (1) FI925767A0 (no)
HU (1) HUT62882A (no)
IE (1) IE912026A1 (no)
IL (1) IL98472A (no)
IS (1) IS3720A7 (no)
LV (1) LV10269B (no)
MA (1) MA22198A1 (no)
NO (1) NO924650D0 (no)
NZ (1) NZ238545A (no)
OA (1) OA09683A (no)
PL (2) PL165898B1 (no)
PT (1) PT98036A (no)
RO (1) RO110497B1 (no)
TN (1) TNSN91050A1 (no)
WO (1) WO1991019712A1 (no)
YU (1) YU104091A (no)

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SE9500422D0 (sv) * 1995-02-06 1995-02-06 Astra Ab New oral pharmaceutical dosage forms
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US6699885B2 (en) * 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
US6645988B2 (en) 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
SE9600070D0 (sv) * 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
EP0983263A1 (en) * 1997-05-30 2000-03-08 Dr. Reddy's Research Foundation Novel benzimidazole derivatives as antiulcer agents, process for their preparation and pharmaceutical compositions containing them
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SE0101379D0 (sv) 2001-04-18 2001-04-18 Diabact Ab Komposition som hämmar utsöndring av magsyra
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CA2492718C (en) * 2002-07-19 2010-12-21 Michael E. Garst Prodrugs of proton pump inhibitors
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US20040248942A1 (en) * 2003-02-20 2004-12-09 Bonnie Hepburn Novel formulation, omeprazole antacid complex-immediate release for rapid and sustained suppression of gastric acid
US8802139B2 (en) 2003-06-26 2014-08-12 Intellipharmaceutics Corp. Proton pump-inhibitor-containing capsules which comprise subunits differently structured for a delayed release of the active ingredient
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US20070161679A1 (en) * 2004-02-18 2007-07-12 Allergan, Inc. Method and compositions for the intravenous administration of compounds related to proton pump inhibitors
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US8906940B2 (en) * 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8815916B2 (en) * 2004-05-25 2014-08-26 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8394409B2 (en) 2004-07-01 2013-03-12 Intellipharmaceutics Corp. Controlled extended drug release technology
JP3921497B2 (ja) * 2004-08-06 2007-05-30 エーザイ・アール・アンド・ディー・マネジメント株式会社 ベンズイミダゾール誘導体とアミンとの塩およびその製造方法
US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
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US20070015782A1 (en) * 2005-04-15 2007-01-18 Eisai Co., Ltd. Benzimidazole compound
US9040564B2 (en) 2005-04-28 2015-05-26 Eisai R&D Management Co., Ltd. Stabilized composition
US7981908B2 (en) 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
US7803817B2 (en) 2005-05-11 2010-09-28 Vecta, Ltd. Composition and methods for inhibiting gastric acid secretion
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CA2648280C (en) 2006-04-03 2014-03-11 Isa Odidi Controlled release delivery device comprising an organosol coat
WO2007122686A1 (ja) * 2006-04-14 2007-11-01 Eisai R & D Management Co., Ltd. ベンズイミダゾール化合物
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JP5492417B2 (ja) * 2006-10-13 2014-05-14 エーザイ・アール・アンド・ディー・マネジメント株式会社 胃酸分泌抑制作用を有するベンズイミダゾール化合物
JP2009196894A (ja) * 2006-10-13 2009-09-03 Eisai R & D Management Co Ltd スルフィニルベンズイミダゾール化合物またはその塩の製造方法
CA2667682A1 (en) 2006-10-27 2008-05-15 The Curators Of The University Of Missouri Compositions comprising acid labile proton pump inhibiting agents, at least one other pharmaceutically active agent and methods of using same
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WO2009105568A1 (en) 2008-02-20 2009-08-27 The Curators Of The University Of Missouri Composition comprising a combination of omeprazole and lansoprazole, and a buffering agent, and methods of using same
CN102209529A (zh) 2008-09-09 2011-10-05 阿斯利康(瑞典)有限公司 将药物组合物递送至有需要的患者的方法
KR20120030106A (ko) 2009-06-25 2012-03-27 아스트라제네카 아베 Nsaid-연관된 궤양의 발생 위험이 있는 환자의 치료 방법
WO2011080500A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
EP2519229A2 (en) 2009-12-29 2012-11-07 Novartis AG New pharmaceutical dosage form for the treatment of gastric acid-related disorders
WO2011080502A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
EP2601947A1 (en) 2011-12-05 2013-06-12 Abo Bakr Mohammed Ali Al-Mehdar Fixed-dose combination for treatment of helicobacter pylori associated diseases
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Also Published As

Publication number Publication date
NZ238545A (en) 1993-08-26
IL98472A (en) 1995-08-31
EP0593463B1 (en) 1999-09-15
US5430042A (en) 1995-07-04
FI925767A (fi) 1992-12-18
AU649456B2 (en) 1994-05-26
EP0593463A1 (en) 1994-04-27
PL297294A1 (no) 1992-07-13
BG97198A (bg) 1993-12-24
AP253A (en) 1993-05-03
CN1058213A (zh) 1992-01-29
JP3049367B2 (ja) 2000-06-05
HUT62882A (en) 1993-06-28
MA22198A1 (fr) 1992-04-01
ATE184602T1 (de) 1999-10-15
PL165898B1 (pl) 1995-02-28
PL297295A1 (no) 1992-07-13
IE912026A1 (en) 1992-01-01
CA2083606C (en) 2001-08-21
ES2140391T3 (es) 2000-03-01
NO924650L (no) 1992-12-02
AP9100286A0 (en) 1991-07-31
OA09683A (en) 1993-05-15
LV10269B (en) 1995-10-20
HU9204034D0 (en) 1993-03-29
TNSN91050A1 (fr) 1992-10-25
NO924650D0 (no) 1992-12-02
CS189391A3 (en) 1992-06-17
YU104091A (sh) 1994-01-20
AU8061791A (en) 1992-01-07
IL98472A0 (en) 1992-07-15
IS3720A7 (is) 1991-12-21
LV10269A (lv) 1994-10-20
RO110497B1 (ro) 1996-01-30
PL166209B1 (pl) 1995-04-28
CZ279434B6 (cs) 1995-04-12
PT98036A (pt) 1992-03-31
CA2083606A1 (en) 1991-12-21
DE69131627D1 (de) 1999-10-21
DE69131627T2 (de) 2000-04-27
WO1991019712A1 (en) 1991-12-26
JPH05507714A (ja) 1993-11-04
EG19752A (en) 1996-01-31

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