FI925309L - Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi Download PDF

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Publication number
FI925309L
FI925309L FI925309A FI925309A FI925309L FI 925309 L FI925309 L FI 925309L FI 925309 A FI925309 A FI 925309A FI 925309 A FI925309 A FI 925309A FI 925309 L FI925309 L FI 925309L
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FI
Finland
Prior art keywords
isopropylimidazo
pyrido
dihydro
oxo
preparation
Prior art date
Application number
FI925309A
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English (en)
Swedish (sv)
Other versions
FI925309A0 (fi
FI93836C (fi
FI93836B (fi
Inventor
Holger Claus Hansen
Frank Waetjen
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Novo Nordisk As
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Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of FI925309A0 publication Critical patent/FI925309A0/fi
Publication of FI925309L publication Critical patent/FI925309L/fi
Application granted granted Critical
Publication of FI93836B publication Critical patent/FI93836B/fi
Publication of FI93836C publication Critical patent/FI93836C/fi

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI925309A 1987-12-08 1992-11-23 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi FI93836C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DK642287A DK160876C (da) 1987-12-08 1987-12-08 Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
DK642287 1987-12-08
FI885518 1988-11-28
FI885518A FI90548C (fi) 1987-12-08 1988-11-28 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi

Publications (4)

Publication Number Publication Date
FI925309A0 FI925309A0 (fi) 1992-11-23
FI925309L true FI925309L (fi) 1992-11-23
FI93836B FI93836B (fi) 1995-02-28
FI93836C FI93836C (fi) 1995-06-12

Family

ID=8148726

Family Applications (2)

Application Number Title Priority Date Filing Date
FI885518A FI90548C (fi) 1987-12-08 1988-11-28 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
FI925309A FI93836C (fi) 1987-12-08 1992-11-23 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI885518A FI90548C (fi) 1987-12-08 1988-11-28 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi

Country Status (18)

Country Link
US (2) US4968682A (fi)
EP (1) EP0320136B1 (fi)
JP (1) JPH01190684A (fi)
KR (1) KR0133079B1 (fi)
AT (1) ATE109147T1 (fi)
AU (1) AU613125B2 (fi)
CA (1) CA1327797C (fi)
DE (1) DE3850861T2 (fi)
DK (1) DK160876C (fi)
ES (1) ES2056941T3 (fi)
FI (2) FI90548C (fi)
IE (1) IE66336B1 (fi)
IL (1) IL88313A (fi)
NO (1) NO169540C (fi)
NZ (1) NZ227212A (fi)
PH (1) PH24818A (fi)
PT (1) PT89170B (fi)
ZA (1) ZA888558B (fi)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them
DK626288D0 (da) * 1988-11-10 1988-11-10 Ferrosan As Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen
US5602252A (en) * 1989-11-17 1997-02-11 Berlex Laboratories, Inc. Tricyclic pteridinones and a process for their preparation
US5854419A (en) * 1989-11-17 1998-12-29 Schering Aktiengesellschaft Tricyclic pteridinones and a process for their preparation
DK588389D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
DK588489D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5276028A (en) * 1990-06-22 1994-01-04 Nordisk A/S Imidazoquinoxaline compounds
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
US5371080A (en) * 1990-06-22 1994-12-06 Novo Nordisk A/S Imidazoquinazoline compounds and their use
CA2110942A1 (en) * 1991-06-14 1992-12-23 Pharmacia & Upjohn Company Llc Imidazo¬1,5-a|quinoxalines
JPH0525037A (ja) * 1991-07-01 1993-02-02 Upjohn Co:The 経口投与酵素感受性腸溶製剤
JP3512110B2 (ja) * 1992-02-13 2004-03-29 ファルマシア・アンド・アップジョン・カンパニー ベンゾジアゼピン受容体結合剤として有用な4−オキソ−および4H−イミダゾ(5,1−c)(1,4)ベンゾオキサジン類
TW274550B (fi) * 1992-09-26 1996-04-21 Hoechst Ag
EP0743855A1 (en) * 1994-01-03 1996-11-27 Acea Pharmaceuticals, Inc. 8-aza, 6-aza and 6,8-diaza-1,4-dihydroquinoxaline-2,3-diones and the use thereof as antagonists for the glycine/nmda receptor
US5792766A (en) * 1996-03-13 1998-08-11 Neurogen Corporation Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands
MX2008009475A (es) * 2006-01-23 2008-10-20 Amira Pharmaceuticals Inc Inhibidores triciclicos de 5-lipoxigenasa.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
ZA825094B (en) * 1981-07-16 1983-04-27 Usv Pharma Corp Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK161148C (da) * 1988-06-14 1991-11-18 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne

Also Published As

Publication number Publication date
NO885442L (no) 1989-06-09
ES2056941T3 (es) 1994-10-16
DK160876B (da) 1991-04-29
NO169540B (no) 1992-03-30
NO169540C (no) 1992-07-08
DE3850861D1 (de) 1994-09-01
AU613125B2 (en) 1991-07-25
EP0320136A3 (en) 1990-12-19
NO885442D0 (no) 1988-12-07
PT89170B (pt) 1993-06-30
DE3850861T2 (de) 1994-11-10
AU2660288A (en) 1989-06-08
DK642287D0 (da) 1987-12-08
ATE109147T1 (de) 1994-08-15
FI90548C (fi) 1994-02-25
IE66336B1 (en) 1995-12-27
FI925309A0 (fi) 1992-11-23
US4999354A (en) 1991-03-12
IL88313A (en) 1993-06-10
IE883347L (en) 1989-06-08
PH24818A (en) 1990-10-30
PT89170A (pt) 1989-12-29
FI885518A7 (fi) 1989-06-09
CA1327797C (en) 1994-03-15
IL88313A0 (en) 1989-06-30
JPH01190684A (ja) 1989-07-31
FI93836C (fi) 1995-06-12
EP0320136B1 (en) 1994-07-27
EP0320136A2 (en) 1989-06-14
DK160876C (da) 1991-10-14
FI885518A0 (fi) 1988-11-28
KR0133079B1 (ko) 1998-04-17
ZA888558B (en) 1989-08-30
FI90548B (fi) 1993-11-15
NZ227212A (en) 1990-07-26
US4968682A (en) 1990-11-06
KR890009931A (ko) 1989-08-04
FI93836B (fi) 1995-02-28
DK642287A (da) 1989-06-09

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