FI910126A0 - Menetelmä farmaseuttisesti käyttökelpoisen 4-(5,6,7,8-tetrahydroimidatso/1,5-a/pyridin-5-yyli)-bentsonitriilin hydrokloridin valmistamiseksi kiteisessä hemihydraattimuodossa - Google Patents

Menetelmä farmaseuttisesti käyttökelpoisen 4-(5,6,7,8-tetrahydroimidatso/1,5-a/pyridin-5-yyli)-bentsonitriilin hydrokloridin valmistamiseksi kiteisessä hemihydraattimuodossa

Info

Publication number
FI910126A0
FI910126A0 FI910126A FI910126A FI910126A0 FI 910126 A0 FI910126 A0 FI 910126A0 FI 910126 A FI910126 A FI 910126A FI 910126 A FI910126 A FI 910126A FI 910126 A0 FI910126 A0 FI 910126A0
Authority
FI
Finland
Prior art keywords
pyridin
preparation
benzonitrile
tetrahydroimidazo
pharmaceutically useful
Prior art date
Application number
FI910126A
Other languages
English (en)
Swedish (sv)
Other versions
FI94528B (fi
FI910126A (fi
FI94528C (fi
Inventor
Jutta Ibrahim
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of FI910126A0 publication Critical patent/FI910126A0/fi
Publication of FI910126A publication Critical patent/FI910126A/fi
Publication of FI94528B publication Critical patent/FI94528B/fi
Application granted granted Critical
Publication of FI94528C publication Critical patent/FI94528C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Lubricants (AREA)
  • Compounds Of Alkaline-Earth Elements, Aluminum Or Rare-Earth Metals (AREA)
  • Liquid Crystal Substances (AREA)
  • Pyridine Compounds (AREA)
  • Photoreceptors In Electrophotography (AREA)
FI910126A 1990-01-12 1991-01-09 Menetelmä farmaseuttisesti käyttökelpoisen 4-(5,6,7,8-tetrahydroimidatso/1,5-a/pyridin-5-yyli)-bentsonitriilin hydrokloridin valmistamiseksi kiteisessä hemihydraattimuodossa FI94528C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH10090 1990-01-12
CH10090 1990-01-12

Publications (4)

Publication Number Publication Date
FI910126A0 true FI910126A0 (fi) 1991-01-09
FI910126A FI910126A (fi) 1991-07-13
FI94528B FI94528B (fi) 1995-06-15
FI94528C FI94528C (fi) 1995-09-25

Family

ID=4179261

Family Applications (1)

Application Number Title Priority Date Filing Date
FI910126A FI94528C (fi) 1990-01-12 1991-01-09 Menetelmä farmaseuttisesti käyttökelpoisen 4-(5,6,7,8-tetrahydroimidatso/1,5-a/pyridin-5-yyli)-bentsonitriilin hydrokloridin valmistamiseksi kiteisessä hemihydraattimuodossa

Country Status (33)

Country Link
US (1) US5098911A (fi)
EP (1) EP0437415B1 (fi)
JP (1) JP2694186B2 (fi)
KR (1) KR100191360B1 (fi)
CN (1) CN1037966C (fi)
AT (1) ATE125809T1 (fi)
AU (1) AU638085B2 (fi)
BG (2) BG60033A3 (fi)
CA (1) CA2033937C (fi)
CZ (1) CZ279823B6 (fi)
DE (1) DE59106101D1 (fi)
DK (1) DK0437415T3 (fi)
DZ (1) DZ1482A1 (fi)
ES (1) ES2075399T3 (fi)
FI (1) FI94528C (fi)
GR (1) GR3017027T3 (fi)
HK (1) HK1000663A1 (fi)
HU (1) HU216192B (fi)
ID (1) ID964B (fi)
IE (1) IE67512B1 (fi)
IL (1) IL96879A (fi)
MA (1) MA22040A1 (fi)
MT (1) MTP1076B (fi)
NO (1) NO175747C (fi)
NZ (1) NZ236735A (fi)
PH (1) PH27601A (fi)
PL (3) PL166500B1 (fi)
PT (1) PT96447B (fi)
RO (1) RO107408B1 (fi)
RU (2) RU2021271C1 (fi)
SA (1) SA93140021B1 (fi)
TN (1) TNSN91001A1 (fi)
ZA (1) ZA91229B (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW208013B (fi) * 1990-03-01 1993-06-21 Daiichi Co Ltd
EP0457716A1 (de) * 1990-04-20 1991-11-21 Ciba-Geigy Ag Naphthalinderivate
TW224461B (fi) * 1990-09-18 1994-06-01 Ciba Geigy Ag
CH683151A5 (de) * 1991-04-24 1994-01-31 Ciba Geigy Ag Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.
JP2914324B2 (ja) * 1995-10-23 1999-06-28 味の素株式会社 ピペリジン誘導体の結晶並びにその製造中間体及び製造方法
KR101913442B1 (ko) 2010-09-01 2018-10-30 에자이 알앤드디 매니지먼트 가부시키가이샤 체중 관리에 유용한 5-ht2c 작동제의 변형-방출 투여 형태
WO2012030939A1 (en) 2010-09-01 2012-03-08 Arena Pharmaceuticals, Inc. Administration of lorcaserin to individuals with renal impairment
AP2014007762A0 (en) 2012-01-17 2014-07-31 Novartis Ag New forms and salts of a dihydropyrrolo[1,2C]imidazolyl aldosterone synthase or aromatase inhibitor
WO2018078049A1 (en) 2016-10-27 2018-05-03 Damian Pharma Ag Aldosterone synthase inhibitor
CN114853755A (zh) 2016-10-27 2022-08-05 达米安制药股份公司 醛固酮合酶抑制剂
BR112020022173A2 (pt) 2018-05-03 2021-02-02 Damian Pharma Ag r-fadrozol para uso no tratamento de aldostonerismo

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4617307A (en) * 1984-06-20 1986-10-14 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridine derivatives as aromatase inhibitors
US4588732A (en) * 1982-12-21 1986-05-13 Ciba-Geigy Corporation Certain imidazo(1,5-a)pyridine derivatives and their use as thromboxane synthetase inhibitors

Also Published As

Publication number Publication date
ES2075399T3 (es) 1995-10-01
KR100191360B1 (ko) 1999-06-15
DK0437415T3 (da) 1995-09-18
ATE125809T1 (de) 1995-08-15
BG61489B2 (bg) 1997-09-30
DZ1482A1 (fr) 2004-09-13
PL166157B1 (pl) 1995-04-28
HK1000663A1 (en) 1998-04-17
FI94528B (fi) 1995-06-15
RO107408B1 (ro) 1993-11-30
IE910103A1 (en) 1991-07-17
HU910084D0 (en) 1991-08-28
IE67512B1 (en) 1996-04-03
PH27601A (en) 1993-08-31
IL96879A0 (en) 1992-03-29
AU638085B2 (en) 1993-06-17
PT96447A (pt) 1991-10-15
SA93140021B1 (ar) 2006-07-11
JP2694186B2 (ja) 1997-12-24
TNSN91001A1 (en) 1992-10-25
NO910137D0 (no) 1991-01-11
RU2021271C1 (ru) 1994-10-15
PL288653A1 (en) 1991-12-16
CN1037966C (zh) 1998-04-08
CA2033937C (en) 2001-03-13
NO175747B (no) 1994-08-22
CN1055739A (zh) 1991-10-30
MTP1076B (en) 1991-09-30
EP0437415A3 (en) 1992-01-22
GR3017027T3 (en) 1995-11-30
CZ279823B6 (cs) 1995-07-12
IL96879A (en) 1995-06-29
DE59106101D1 (de) 1995-09-07
EP0437415A2 (de) 1991-07-17
EP0437415B1 (de) 1995-08-02
NO175747C (no) 1994-11-30
PL166500B1 (pl) 1995-05-31
US5098911A (en) 1992-03-24
AU6928091A (en) 1991-07-18
NZ236735A (en) 1992-10-28
ID964B (id) 1996-09-30
PT96447B (pt) 1998-09-30
CA2033937A1 (en) 1991-07-13
CS9100055A2 (en) 1991-08-13
NO910137L (no) 1991-07-15
FI910126A (fi) 1991-07-13
BG60033A3 (en) 1993-07-15
RU2088584C1 (ru) 1997-08-27
PL167164B1 (pl) 1995-08-31
HUT56568A (en) 1991-09-30
HU216192B (en) 2001-03-28
JPH04210982A (ja) 1992-08-03
ZA91229B (en) 1991-08-28
KR910014376A (ko) 1991-08-31
FI94528C (fi) 1995-09-25
MA22040A1 (fr) 1991-10-01

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Owner name: NOVARTIS AG