FI69453C - Saett att framstaella en ny polymorf form av terapeutiskt anvaendbar 2-(4-klorfenyl)-alfa-metyl-5-bensoxazolylaettiksyra - Google Patents

Saett att framstaella en ny polymorf form av terapeutiskt anvaendbar 2-(4-klorfenyl)-alfa-metyl-5-bensoxazolylaettiksyra Download PDF

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Publication number
FI69453C
FI69453C FI782043A FI782043A FI69453C FI 69453 C FI69453 C FI 69453C FI 782043 A FI782043 A FI 782043A FI 782043 A FI782043 A FI 782043A FI 69453 C FI69453 C FI 69453C
Authority
FI
Finland
Prior art keywords
methyl
chlorophenyl
polymorf
benzozazolyl
alphate
Prior art date
Application number
FI782043A
Other languages
English (en)
Finnish (fi)
Other versions
FI782043A (fi
FI69453B (fi
Inventor
Roy Sherlock
Terence Alan Hicks
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of FI782043A publication Critical patent/FI782043A/fi
Priority to FI831930A priority Critical patent/FI69454C/fi
Application granted granted Critical
Publication of FI69453B publication Critical patent/FI69453B/fi
Publication of FI69453C publication Critical patent/FI69453C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57Aryl or substituted aryl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI782043A 1977-06-28 1978-06-27 Saett att framstaella en ny polymorf form av terapeutiskt anvaendbar 2-(4-klorfenyl)-alfa-metyl-5-bensoxazolylaettiksyra FI69453C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI831930A FI69454C (fi) 1977-06-28 1983-05-30 Saett att framstaella en termodynamiskt stabil ny polymorf form av terapeutiskt anvaendbar 2-(4-klorfenyl)-alfa-metyl-5-bensoxazolylaettiksyra

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB26907/77A GB1590587A (en) 1977-06-28 1977-06-28 Benoxaprofen
GB2690777 1977-06-28

Publications (3)

Publication Number Publication Date
FI782043A FI782043A (fi) 1978-12-29
FI69453B FI69453B (fi) 1985-10-31
FI69453C true FI69453C (fi) 1986-02-10

Family

ID=10251100

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782043A FI69453C (fi) 1977-06-28 1978-06-27 Saett att framstaella en ny polymorf form av terapeutiskt anvaendbar 2-(4-klorfenyl)-alfa-metyl-5-bensoxazolylaettiksyra

Country Status (17)

Country Link
EP (1) EP0000276B1 (xx)
JP (1) JPS5411224A (xx)
AT (1) AT360008B (xx)
AU (1) AU518403B2 (xx)
BE (1) BE868522A (xx)
CH (1) CH631449A5 (xx)
DE (2) DE2828074A1 (xx)
DK (1) DK145419C (xx)
FI (1) FI69453C (xx)
FR (1) FR2396004A1 (xx)
GB (1) GB1590587A (xx)
IE (1) IE47009B1 (xx)
IL (1) IL55015A (xx)
IT (1) IT1105065B (xx)
LU (1) LU79879A1 (xx)
NZ (1) NZ187674A (xx)
ZA (1) ZA783660B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1435721A (en) * 1972-05-18 1976-05-12 Lilly Industries Ltd Benzoxazole derivatives
US3888864A (en) 1973-06-29 1975-06-10 Hoffmann La Roche Amino lower alkyl ether derivatives of opium alkaloids
GB1495488A (en) * 1976-06-23 1977-12-21 Ippco Int Pharma Patents Co Es Optically active 2-(2-phenyl-5-benzoxazolyl)propionic acids
IT1099589B (it) * 1978-08-04 1985-09-18 Ravizza Spa Processo per la preparazione di derivati dell'acido benzoxazolil propionico
IT1157295B (it) * 1982-07-19 1987-02-11 Ravizza Spa Processo perfezionato per la preparazione di derivati dell'acido benzoxazolil propionico
UA83620C2 (ru) 2001-12-05 2008-08-11 Уайт Замещенные бензоксазолы и их аналоги как эстрогенные агенты
WO2021116820A1 (en) * 2019-12-10 2021-06-17 Aurobindo Pharma Limited An improved process for the preparation of benoxaprofen
DE102022117931A1 (de) 2022-07-18 2024-01-18 HUECK System GmbH & Co. KG Profilanordnung mit wärmedämmung
US11981645B1 (en) 2023-10-10 2024-05-14 King Faisal University N′-(2-naphthoyloxy)-2-(benzo[d]oxazol-2-yl)acetimidamide as antimicrobial compound

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1435721A (en) * 1972-05-18 1976-05-12 Lilly Industries Ltd Benzoxazole derivatives
GB1488003A (en) * 1973-10-23 1977-10-05 Lilly Industries Ltd 1,2-benzisoxazole derivatives processes for their preparation and their use as pharmaceuticals
US4087437A (en) * 1976-09-07 1978-05-02 Eli Lilly And Company 2-Phenyl-5-benzoxazolylalkanoic acid purification process

Also Published As

Publication number Publication date
DK145419C (da) 1983-04-18
EP0000276B1 (en) 1982-09-01
DE2862013D1 (en) 1982-10-28
BE868522A (fr) 1978-12-27
IT7850048A0 (it) 1978-06-27
IL55015A0 (en) 1978-08-31
IE47009B1 (en) 1983-11-30
IL55015A (en) 1981-11-30
FI782043A (fi) 1978-12-29
FR2396004B1 (xx) 1981-09-18
CH631449A5 (fr) 1982-08-13
FI69453B (fi) 1985-10-31
JPS6231714B2 (xx) 1987-07-09
IE781277L (en) 1978-12-28
DK287578A (da) 1978-12-29
LU79879A1 (xx) 1978-12-07
JPS5411224A (en) 1979-01-27
AT360008B (de) 1980-12-10
EP0000276A1 (en) 1979-01-10
AU518403B2 (en) 1981-10-01
DK145419B (da) 1982-11-15
ATA466178A (de) 1980-05-15
GB1590587A (en) 1981-06-03
DE2828074A1 (de) 1979-01-11
NZ187674A (en) 1980-11-14
ZA783660B (en) 1979-06-27
IT1105065B (it) 1985-10-28
FR2396004A1 (fr) 1979-01-26
AU3750178A (en) 1980-01-03

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Owner name: LILLY INDUSTRIES LIMITED