FI68824C - Foerfarande foer framstaellning av terapeutiskt effektiva substituerade 2-etenyl-4-oxo-4h-pyrido(1,2-a)pyrimidiner - Google Patents

Foerfarande foer framstaellning av terapeutiskt effektiva substituerade 2-etenyl-4-oxo-4h-pyrido(1,2-a)pyrimidiner Download PDF

Info

Publication number
FI68824C
FI68824C FI801464A FI801464A FI68824C FI 68824 C FI68824 C FI 68824C FI 801464 A FI801464 A FI 801464A FI 801464 A FI801464 A FI 801464A FI 68824 C FI68824 C FI 68824C
Authority
FI
Finland
Prior art keywords
pyrido
oxo
trans
pyrimidine
carboxylic acid
Prior art date
Application number
FI801464A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI68824B (fi
FI801464A (fi
Inventor
Gianfederico Doria
Ciriaco Romeo
Piero Sberze
Marcellino Tibolla
Maria Luisa Corno
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI801464A publication Critical patent/FI801464A/fi
Application granted granted Critical
Publication of FI68824B publication Critical patent/FI68824B/fi
Publication of FI68824C publication Critical patent/FI68824C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI801464A 1979-05-08 1980-05-06 Foerfarande foer framstaellning av terapeutiskt effektiva substituerade 2-etenyl-4-oxo-4h-pyrido(1,2-a)pyrimidiner FI68824C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7915810 1979-05-08
GB7915810 1979-05-08

Publications (3)

Publication Number Publication Date
FI801464A FI801464A (fi) 1980-11-09
FI68824B FI68824B (fi) 1985-07-31
FI68824C true FI68824C (fi) 1985-11-11

Family

ID=10504995

Family Applications (1)

Application Number Title Priority Date Filing Date
FI801464A FI68824C (fi) 1979-05-08 1980-05-06 Foerfarande foer framstaellning av terapeutiskt effektiva substituerade 2-etenyl-4-oxo-4h-pyrido(1,2-a)pyrimidiner

Country Status (28)

Country Link
US (2) US4310526A (fr)
JP (1) JPS562983A (fr)
AT (1) AT375370B (fr)
AU (1) AU527931B2 (fr)
BE (1) BE883150A (fr)
CA (1) CA1134359A (fr)
CH (1) CH647777A5 (fr)
CS (2) CS528780A2 (fr)
DE (1) DE3015738A1 (fr)
DK (1) DK200280A (fr)
ES (1) ES8104287A1 (fr)
FI (1) FI68824C (fr)
FR (1) FR2456093A1 (fr)
GB (1) GB2050353B (fr)
GR (1) GR68075B (fr)
HU (1) HU181778B (fr)
IE (1) IE49787B1 (fr)
IL (1) IL59802A (fr)
IT (1) IT1209326B (fr)
LU (1) LU82419A1 (fr)
NL (1) NL8002656A (fr)
NO (1) NO153137C (fr)
NZ (1) NZ193579A (fr)
PH (1) PH16695A (fr)
PT (1) PT71197A (fr)
SE (1) SE437158B (fr)
SU (2) SU1217259A3 (fr)
ZA (1) ZA802390B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT377586B (de) 1981-06-30 1985-04-10 Erba Farmitalia Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
CA1211111A (fr) * 1982-02-15 1986-09-09 Isao Yanagisawa Methode de preparation de composes nouveau genre de pyrimidone
ES8406476A1 (es) * 1982-04-29 1984-07-01 Erba Farmitalia Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas.
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
GB8501015D0 (en) * 1985-01-16 1985-02-20 Riker Laboratories Inc Drug
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
JP5419894B2 (ja) * 2008-01-11 2014-02-19 グレンマーク ファーマシューティカルズ， エセ．アー． Ｔｒｐｖ３モジュレーターとしての縮合ピリミジン誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones
HU178910B (en) 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180701B (en) 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
HU184058B (en) 1977-12-29 1984-06-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing new compounds with nitrogen bridge head

Also Published As

Publication number Publication date
GR68075B (fr) 1981-10-30
IT1209326B (it) 1989-07-16
IE49787B1 (en) 1985-12-11
SE8003433L (sv) 1980-11-09
ES491238A0 (es) 1981-04-01
DK200280A (da) 1980-11-09
NO153137B (no) 1985-10-14
NL8002656A (nl) 1980-11-11
IE800945L (en) 1980-11-08
SE437158B (sv) 1985-02-11
GB2050353B (en) 1983-04-27
LU82419A1 (fr) 1980-07-31
FR2456093B1 (fr) 1984-02-03
DE3015738A1 (de) 1980-11-13
US4310526A (en) 1982-01-12
FR2456093A1 (fr) 1980-12-05
FI68824B (fi) 1985-07-31
ES8104287A1 (es) 1981-04-01
SU1217259A3 (ru) 1986-03-07
NO801342L (no) 1980-11-10
BE883150A (fr) 1980-11-07
AT375370B (de) 1984-07-25
CS321380A2 (en) 1984-12-14
JPS562983A (en) 1981-01-13
NO153137C (no) 1986-01-22
CS244107B2 (en) 1986-07-17
US4341780A (en) 1982-07-27
IT8021821A0 (it) 1980-05-06
AU527931B2 (en) 1983-03-31
PT71197A (en) 1980-06-01
HU181778B (en) 1983-11-28
ZA802390B (en) 1981-04-29
IL59802A0 (en) 1980-06-30
SU1158045A3 (ru) 1985-05-23
PH16695A (en) 1984-01-06
CH647777A5 (de) 1985-02-15
CA1134359A (fr) 1982-10-26
ATA245680A (de) 1983-12-15
CS528780A2 (en) 1985-09-17
IL59802A (en) 1983-07-31
FI801464A (fi) 1980-11-09
GB2050353A (en) 1981-01-07
NZ193579A (en) 1982-09-07
AU5731980A (en) 1980-11-13

Similar Documents

Publication Publication Date Title
EP0091241B1 (fr) Dérivés condensés de pyrrolinone, et leur préparation
US6160119A (en) Fused dihydropyrans
FI68824C (fi) Foerfarande foer framstaellning av terapeutiskt effektiva substituerade 2-etenyl-4-oxo-4h-pyrido(1,2-a)pyrimidiner
PL132141B1 (en) Process for preparing novel derivatives of dibenzoimidazoazepins
AU740578B2 (en) Tetrahydropyrido compounds
FI57949B (fi) Foerfarande foer framstaellning av terapeutiskt anvaendbara 4-oxo-6,7,8,9-tetrahydropyrido (1,2-a) pyrimidinderivat
US4912104A (en) Tricyclic fused pryimidine derivatives, and their use as pharmaceuticals
US4085111A (en) 1H-tetrazole derivatives
GB2061944A (en) New pyridothienotriazines
US3404157A (en) Substituted pyrroloindazole compounds
US3519628A (en) Aralkyl diazabicyclo(4,4,0)decanes
EP0229823B1 (fr) Derives polycycliques de quinoline, naphthyridine et pyrazinopyridine
CA1154766A (fr) Composes antiallergiques et procede de preparation
US3949081A (en) 4-Carbamoyl-1-benzazepines as antiinflammatory agents
FI77869C (fi) Foerfarande foer framstaellning av substituerade karboxitiazolo/3,2-a/pyrimidinderivat med en antiallergisk verkan.
US3594378A (en) Thiazolopyrimidine derivatives and preparation thereof
PT100767A (pt) Tetra-hidrobenzotienopiridinas e processo para a sua preparacao
FI74467C (fi) Foerfarande foer framstaellning av 1,2,3,10-tetrahydro-10-oxo-cyklopenta/d/pyrido/1,2-a/pyrimidin- och 1,2,3,4-tetrahydro-11-oxo-11h-pyrido/2,1-b/kinazolinderivat.
KR840000104B1 (ko) 치환 피리도[1, 2-a] 피리미딘의 제조방법
IE59728B1 (en) Substituted 1,3,4,9-tetrahydropyrano[3,4-b] indole-1-acetic acids
US3989689A (en) 4-Carbamoyl-1-benzazepines
US3931151A (en) Dibenzo (b,f) azepines
US4978671A (en) Thieno (3',4'-4,5)imidazo(2,1-b)thiazole derivatives, a process for their preparation and their use in medicaments
US3498980A (en) Oxazinoisoquinoline derivatives
NO166586B (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive cykloalka-(b)-pyrazolo(3,4-d)-pyrridin-3-on-derivater.

Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A