NL8002656A - Gesubstitueerde pyrido 1.2-a pyrimidinen. - Google Patents

Gesubstitueerde pyrido 1.2-a pyrimidinen. Download PDF

Info

Publication number
NL8002656A
NL8002656A NL8002656A NL8002656A NL8002656A NL 8002656 A NL8002656 A NL 8002656A NL 8002656 A NL8002656 A NL 8002656A NL 8002656 A NL8002656 A NL 8002656A NL 8002656 A NL8002656 A NL 8002656A
Authority
NL
Netherlands
Prior art keywords
pyrido
trans
oxo
pyrimidine
carboxylic acid
Prior art date
Application number
NL8002656A
Other languages
English (en)
Dutch (nl)
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NL8002656A publication Critical patent/NL8002656A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NL8002656A 1979-05-08 1980-05-08 Gesubstitueerde pyrido 1.2-a pyrimidinen. NL8002656A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7915810 1979-05-08
GB7915810 1979-05-08

Publications (1)

Publication Number Publication Date
NL8002656A true NL8002656A (nl) 1980-11-11

Family

ID=10504995

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8002656A NL8002656A (nl) 1979-05-08 1980-05-08 Gesubstitueerde pyrido 1.2-a pyrimidinen.

Country Status (28)

Country Link
US (2) US4310526A (fr)
JP (1) JPS562983A (fr)
AT (1) AT375370B (fr)
AU (1) AU527931B2 (fr)
BE (1) BE883150A (fr)
CA (1) CA1134359A (fr)
CH (1) CH647777A5 (fr)
CS (2) CS528780A2 (fr)
DE (1) DE3015738A1 (fr)
DK (1) DK200280A (fr)
ES (1) ES8104287A1 (fr)
FI (1) FI68824C (fr)
FR (1) FR2456093A1 (fr)
GB (1) GB2050353B (fr)
GR (1) GR68075B (fr)
HU (1) HU181778B (fr)
IE (1) IE49787B1 (fr)
IL (1) IL59802A (fr)
IT (1) IT1209326B (fr)
LU (1) LU82419A1 (fr)
NL (1) NL8002656A (fr)
NO (1) NO153137C (fr)
NZ (1) NZ193579A (fr)
PH (1) PH16695A (fr)
PT (1) PT71197A (fr)
SE (1) SE437158B (fr)
SU (2) SU1217259A3 (fr)
ZA (1) ZA802390B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT377586B (de) 1981-06-30 1985-04-10 Erba Farmitalia Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
CA1211111A (fr) * 1982-02-15 1986-09-09 Isao Yanagisawa Methode de preparation de composes nouveau genre de pyrimidone
ES8406476A1 (es) * 1982-04-29 1984-07-01 Erba Farmitalia Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas.
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
GB8501015D0 (en) * 1985-01-16 1985-02-20 Riker Laboratories Inc Drug
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
JP5419894B2 (ja) * 2008-01-11 2014-02-19 グレンマーク ファーマシューティカルズ， エセ．アー． Ｔｒｐｖ３モジュレーターとしての縮合ピリミジン誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones
HU178910B (en) 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180701B (en) 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
HU184058B (en) 1977-12-29 1984-06-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing new compounds with nitrogen bridge head

Also Published As

Publication number Publication date
GR68075B (fr) 1981-10-30
IT1209326B (it) 1989-07-16
IE49787B1 (en) 1985-12-11
SE8003433L (sv) 1980-11-09
ES491238A0 (es) 1981-04-01
DK200280A (da) 1980-11-09
NO153137B (no) 1985-10-14
IE800945L (en) 1980-11-08
SE437158B (sv) 1985-02-11
GB2050353B (en) 1983-04-27
LU82419A1 (fr) 1980-07-31
FR2456093B1 (fr) 1984-02-03
DE3015738A1 (de) 1980-11-13
US4310526A (en) 1982-01-12
FR2456093A1 (fr) 1980-12-05
FI68824C (fi) 1985-11-11
FI68824B (fi) 1985-07-31
ES8104287A1 (es) 1981-04-01
SU1217259A3 (ru) 1986-03-07
NO801342L (no) 1980-11-10
BE883150A (fr) 1980-11-07
AT375370B (de) 1984-07-25
CS321380A2 (en) 1984-12-14
JPS562983A (en) 1981-01-13
NO153137C (no) 1986-01-22
CS244107B2 (en) 1986-07-17
US4341780A (en) 1982-07-27
IT8021821A0 (it) 1980-05-06
AU527931B2 (en) 1983-03-31
PT71197A (en) 1980-06-01
HU181778B (en) 1983-11-28
ZA802390B (en) 1981-04-29
IL59802A0 (en) 1980-06-30
SU1158045A3 (ru) 1985-05-23
PH16695A (en) 1984-01-06
CH647777A5 (de) 1985-02-15
CA1134359A (fr) 1982-10-26
ATA245680A (de) 1983-12-15
CS528780A2 (en) 1985-09-17
IL59802A (en) 1983-07-31
FI801464A (fi) 1980-11-09
GB2050353A (en) 1981-01-07
NZ193579A (en) 1982-09-07
AU5731980A (en) 1980-11-13

Similar Documents

Publication Publication Date Title
EP0091241B1 (fr) Dérivés condensés de pyrrolinone, et leur préparation
EP0086422B1 (fr) Pyrazolo (4,3-c)pyridines à activité pharmacologique
DK157868B (da) Analogifremgangsmaade til fremstilling af tetracykliske forbindelser
US3784551A (en) 2-oxo-1,4-dioxa-8-azaspiro (4.5) decanes and related compounds
JPH01190680A (ja) インドール誘導体およびその製造方法
JPH0383985A (ja) 新規４―メチレン―２―オキソ―８―アザスピロ〔４，５〕デカン誘導体，それらを含む医薬組成物およびそれらの調整方法
JPS6172751A (ja) カルボニル化合物、その製造方法及び該化合物を含む医薬製剤
NL8002656A (nl) Gesubstitueerde pyrido 1.2-a pyrimidinen.
SK283288B6 (sk) Tetrahydropyridínové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie
JPH0377885A (ja) ２―オキソ―１―オキサ―８―アザスピロ〔４，５〕デカン誘導体、それを含む医薬組成物及びその製造方法
AU609559B2 (en) Heterocyclic oxophthalazinyl acetic acids
JPH09510992A (ja) ブラジキニンアンタゴニストとしてのジヒドロピリジン誘導体
RO108347B1 (ro) DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
CA1175428A (fr) Methode de preparation de derives d'imidazo ¬1,2-a| quinoline
US3949081A (en) 4-Carbamoyl-1-benzazepines as antiinflammatory agents
FI72516C (fi) Foerfarande foer framstaellning av farmaceutiskt aktiva 3,6-disubstituerade 2-cyklopropyl-kromoner.
US3594378A (en) Thiazolopyrimidine derivatives and preparation thereof
US5380748A (en) Trialkylamine derivative and ameliorant for digestive tract movement containing the same
US5008282A (en) Cyclic guanidine derivatives, anti-ulceratives and methods of manufacturing the same
US3989689A (en) 4-Carbamoyl-1-benzazepines
JPS59130891A (ja) 置換カルボキシ−チアゾロ〔３，２−ａ〕ピリミジン誘導体およびそれらの製法
JPH04244081A (ja) １，４−ジヒドロピリジン誘導体およびそれを有効成分とするアレルギー性または炎症性疾患治療剤
CH660485A5 (de) Mit einem substituierten cycloaliphatischen ring kondensierte pyrido-(1,2-a)-pyrimidinone.
JPH11503432A (ja) オルト位で縮合環化したβ−カルボリン
JPH02212486A (ja) イミダゾピリジン誘導体

Legal Events

Date Code Title Description
A1B A search report has been drawn up
BT A notification was added to the application dossier and made available to the public
BT A notification was added to the application dossier and made available to the public
A85 Still pending on 85-01-01
BC A request for examination has been filed
BV The patent application has lapsed