FI63574C - Foerfarande foer framstaellning av nya terapeutiskt anvaendbara pyrido(1,2-a)pyrimidinderivat - Google Patents
Foerfarande foer framstaellning av nya terapeutiskt anvaendbara pyrido(1,2-a)pyrimidinderivat Download PDFInfo
- Publication number
- FI63574C FI63574C FI770453A FI770453A FI63574C FI 63574 C FI63574 C FI 63574C FI 770453 A FI770453 A FI 770453A FI 770453 A FI770453 A FI 770453A FI 63574 C FI63574 C FI 63574C
- Authority
- FI
- Finland
- Prior art keywords
- pyrido
- methyl
- compound
- pyrimidine
- alkoxycarbonyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU76CI1642A HU174693B (hu) | 1976-02-12 | 1976-02-12 | Sposob poluchenija kondensirovannykh proizvodnykh pirimidina |
| HUCI001642 | 1976-02-12 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI770453A7 FI770453A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-08-13 |
| FI63574B FI63574B (fi) | 1983-03-31 |
| FI63574C true FI63574C (fi) | 1983-07-11 |
Family
ID=10994601
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI770453A FI63574C (fi) | 1976-02-12 | 1977-02-11 | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara pyrido(1,2-a)pyrimidinderivat |
Country Status (28)
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU173438B (hu) * | 1975-11-27 | 1979-05-28 | Chinoin Gyogyszer Es Vegyeszet | Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom |
| HU180439B (en) * | 1977-12-29 | 1983-03-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing 9-amino-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives |
| HU184058B (en) * | 1977-12-29 | 1984-06-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing new compounds with nitrogen bridge head |
| HU185925B (en) * | 1977-12-29 | 1985-04-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing compounds with nitrogen bridge head |
| HU178496B (en) * | 1977-12-29 | 1982-05-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity |
| HU180701B (en) * | 1977-12-29 | 1983-04-29 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering |
| US4642384A (en) * | 1979-03-19 | 1987-02-10 | Riker Laboratories, Inc. | Process for the preparation of derivatives of pyrrolidine and piperidine |
| AT370731B (de) * | 1979-05-02 | 1983-04-25 | Chinoin Gyogyszer Es Vegyeszet | Verfahren zur herstellung von neuen kondensierten pyrimidin-derivaten sowie von deren optischen antipoden und salzen |
| HU183408B (en) * | 1981-04-28 | 1984-05-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing oral ratard pharmaceutical compositions |
| AT377586B (de) * | 1981-06-30 | 1985-04-10 | Erba Farmitalia | Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen |
| ES521739A0 (es) * | 1982-04-29 | 1984-07-01 | Erba Farmitalia | Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas. |
| ES524262A0 (es) * | 1982-08-05 | 1984-11-16 | Erba Farmitalia | "procedimiento para preparar derivados de quinazolina" |
| US5252572A (en) * | 1988-02-03 | 1993-10-12 | Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt. | Pyridopyrimidine derivatives, pharmaceutical compositions containing them and process for preparing same |
| EP1539762A2 (en) * | 2002-06-26 | 2005-06-15 | Bristol-Myers Squibb Company | Bicyclic pyrimidinones as coagulation cascade inhibitors |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3376304A (en) * | 1962-03-14 | 1968-04-02 | Mcneilab Inc | 2-(r-r1-r2-methyl)-6-r3-6-r4-fulvenes |
| US3907798A (en) * | 1966-06-15 | 1975-09-23 | Sterling Drug Inc | Preparation of 4H-pyrido{8 1,2-a{9 pyrimidin-4-ones from cyclic alkylidene 2-pyridylaminomethylenemalonates |
| AT299212B (de) * | 1966-11-02 | 1972-06-12 | Chinoin Gyogyszer Es Vegyeszet | Verfahren zur Herstellung von neuen Homopyrimidazol-Derivaten sowie von deren Salzen |
| US3567719A (en) * | 1967-05-17 | 1971-03-02 | Eastman Kodak Co | Methods for preparing dyes and novel dye intermediates |
| US3635956A (en) * | 1968-03-01 | 1972-01-18 | Squibb & Sons Inc | Benzothiazines related compounds derivatives and salts thereof |
| FR2187311B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1972-06-02 | 1975-06-20 | Bouchara Emile | |
| HU168014B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1973-03-30 | 1976-02-28 | ||
| US3897420A (en) * | 1973-06-28 | 1975-07-29 | Squibb & Sons Inc | 2-Aminoalkyl-7-substituted-3,3a,4,5,6,7-hexahydro-3-substituted-2H-pyrazolo(4,3-c)pyridines |
| US3929787A (en) * | 1974-04-22 | 1975-12-30 | Squibb & Sons Inc | 6,7,8,9-Tetrahydro-pyrido(1,2-a)pyrimidin-4-ones |
| DE2427614A1 (de) * | 1974-06-07 | 1976-01-02 | Gruenenthal Chemie | Neue pyrrolderivate und verfahren zu ihrer herstellung |
| US3898224A (en) * | 1974-09-09 | 1975-08-05 | Squibb & Sons Inc | 1,6,7,8-Tetrahydro-4-oxo-4H-pyrido {8 1,2-A{9 pyrimidine-9-carboalkoxy compounds |
| US3965100A (en) * | 1975-02-26 | 1976-06-22 | E. R. Squibb & Sons, Inc. | 2,3-Dihydrocyclopenta[d]pyrido[1,2-a]pyrimidin-10(1H)-one and its derivatives |
| US3935197A (en) * | 1975-05-16 | 1976-01-27 | E. R. Squibb & Sons, Inc. | 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones |
-
1976
- 1976-02-12 HU HU76CI1642A patent/HU174693B/hu not_active IP Right Cessation
-
1977
- 1977-02-04 IL IL51388A patent/IL51388A/xx unknown
- 1977-02-04 BG BG035340A patent/BG29723A3/xx unknown
- 1977-02-04 US US05/765,595 patent/US4123533A/en not_active Expired - Lifetime
- 1977-02-08 SE SE7701375A patent/SE431334B/xx not_active IP Right Cessation
- 1977-02-09 AT AT84277A patent/AT357539B/de not_active IP Right Cessation
- 1977-02-09 YU YU00337/77A patent/YU33777A/xx unknown
- 1977-02-10 ES ES455800A patent/ES455800A1/es not_active Expired
- 1977-02-10 AU AU22172/77A patent/AU512470B2/en not_active Expired
- 1977-02-10 FR FR7703774A patent/FR2340945A1/fr active Granted
- 1977-02-10 IN IN190/CAL/77A patent/IN146173B/en unknown
- 1977-02-10 JP JP1309577A patent/JPS5297996A/ja active Granted
- 1977-02-10 GR GR52763A patent/GR62466B/el unknown
- 1977-02-11 SU SU772452003A patent/SU969165A3/ru active
- 1977-02-11 AR AR266516A patent/AR220675A1/es active
- 1977-02-11 PT PT66184A patent/PT66184B/pt unknown
- 1977-02-11 PL PL1977195949A patent/PL109346B1/pl unknown
- 1977-02-11 NO NO770457A patent/NO146775C/no unknown
- 1977-02-11 CA CA271,582A patent/CA1082699A/en not_active Expired
- 1977-02-11 GB GB5737/77A patent/GB1554370A/en not_active Expired
- 1977-02-11 FI FI770453A patent/FI63574C/fi not_active IP Right Cessation
- 1977-02-11 CH CH170177A patent/CH637651A5/de not_active IP Right Cessation
- 1977-02-11 DK DK059177A patent/DK152431C/da not_active IP Right Cessation
- 1977-02-11 DE DE19772705778 patent/DE2705778A1/de active Granted
- 1977-02-11 NL NL7701461A patent/NL7701461A/xx not_active Application Discontinuation
- 1977-02-11 BE BE174870A patent/BE851346A/xx not_active IP Right Cessation
- 1977-02-11 DD DD7700197345A patent/DD131557A5/xx unknown
- 1977-02-14 CS CS77971A patent/CS199288B2/cs unknown
-
1978
- 1978-08-08 US US05/931,908 patent/US4252807A/en not_active Expired - Lifetime
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM | Patent lapsed | ||
| MM | Patent lapsed |
Owner name: CHINOIN GYOGUSZER ES VEGYESZETI TERMEKEK |