FI63410C - Foerfarande foer framstaellning av antibakterial 7beta-haloarylmalonamido-7alfa-metoxi-3-heterocyklisk tiometyl-1-detia-1-oxa-3-cefem-4-karboxylsyra eller derivat daerav - Google Patents

Foerfarande foer framstaellning av antibakterial 7beta-haloarylmalonamido-7alfa-metoxi-3-heterocyklisk tiometyl-1-detia-1-oxa-3-cefem-4-karboxylsyra eller derivat daerav Download PDF

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Publication number
FI63410C
FI63410C FI781313A FI781313A FI63410C FI 63410 C FI63410 C FI 63410C FI 781313 A FI781313 A FI 781313A FI 781313 A FI781313 A FI 781313A FI 63410 C FI63410 C FI 63410C
Authority
FI
Finland
Prior art keywords
acid
oxa
detia
methoxy
thiomethyl
Prior art date
Application number
FI781313A
Other languages
English (en)
Finnish (fi)
Other versions
FI781313A (fi
FI63410B (fi
Inventor
Yoshio Hamashima
Masayuki Narisada
Sadao Hayashi
Wataru Nagata
Original Assignee
Shinogi Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP52049630A external-priority patent/JPS609717B2/ja
Priority claimed from JP52102260A external-priority patent/JPS6031835B2/ja
Application filed by Shinogi Co filed Critical Shinogi Co
Publication of FI781313A publication Critical patent/FI781313A/fi
Publication of FI63410B publication Critical patent/FI63410B/fi
Application granted granted Critical
Publication of FI63410C publication Critical patent/FI63410C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/42—Unsaturated compounds containing hydroxy or O-metal groups
    • C07C59/56—Unsaturated compounds containing hydroxy or O-metal groups containing halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI781313A 1977-04-28 1978-04-27 Foerfarande foer framstaellning av antibakterial 7beta-haloarylmalonamido-7alfa-metoxi-3-heterocyklisk tiometyl-1-detia-1-oxa-3-cefem-4-karboxylsyra eller derivat daerav FI63410C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP52049630A JPS609717B2 (ja) 1977-04-28 1977-04-28 ハロアリ―ルマロンアミドオキサセフアロスポリン
JP4963077 1977-04-28
JP10226077 1977-08-25
JP52102260A JPS6031835B2 (ja) 1977-08-25 1977-08-25 チアジアゾリルチオオキサセフアロスポリン

Publications (3)

Publication Number Publication Date
FI781313A FI781313A (fi) 1978-10-29
FI63410B FI63410B (fi) 1983-02-28
FI63410C true FI63410C (fi) 1983-06-10

Family

ID=26390044

Family Applications (1)

Application Number Title Priority Date Filing Date
FI781313A FI63410C (fi) 1977-04-28 1978-04-27 Foerfarande foer framstaellning av antibakterial 7beta-haloarylmalonamido-7alfa-metoxi-3-heterocyklisk tiometyl-1-detia-1-oxa-3-cefem-4-karboxylsyra eller derivat daerav

Country Status (29)

Country Link
US (1) US4183928A (es)
AR (1) AR227614A1 (es)
AT (1) AT357674B (es)
AU (1) AU522851B2 (es)
BG (1) BG34337A3 (es)
CA (1) CA1100962A (es)
CH (1) CH640535A5 (es)
CS (1) CS199726B2 (es)
DD (1) DD135908A5 (es)
DE (1) DE2818985C2 (es)
DK (1) DK182878A (es)
ES (1) ES469206A1 (es)
FI (1) FI63410C (es)
FR (1) FR2388815A1 (es)
GB (1) GB1574273A (es)
GR (1) GR69966B (es)
HU (1) HU178105B (es)
IE (1) IE46627B1 (es)
IL (1) IL54596A0 (es)
IT (1) IT1111469B (es)
MX (1) MX5952E (es)
NL (1) NL189669C (es)
NO (1) NO158506C (es)
NZ (1) NZ187086A (es)
PH (1) PH16851A (es)
PL (1) PL110680B1 (es)
PT (1) PT67957B (es)
SU (1) SU784779A3 (es)
YU (1) YU42477B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4259485A (en) * 1979-04-24 1981-03-31 Eli Lilly And Company Crystallization process
JPS60123490A (ja) * 1983-12-07 1985-07-02 Shionogi & Co Ltd マロニルオキサセフェムカルボン酸誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL178005C (nl) * 1972-11-06 1986-01-02 Merck & Co Inc Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
GB1510794A (en) * 1974-08-06 1978-05-17 Univ Kingston 1-oxacephems and intermediates therefor
US4045438A (en) * 1975-10-24 1977-08-30 Yeda Research And Development Co. Ltd. Cephalosporin antibiotics
US4048311A (en) * 1976-01-08 1977-09-13 Smithkline Corporation 7-Acyl-3-(sulfonic acid and sulfamoyl substituted tetrazolyl thiomethyl)cephalosporins
CA1085392A (en) * 1976-03-25 1980-09-09 Masayuki Narisada Arylmalonamido-1-oxadethiacephalosporins

Also Published As

Publication number Publication date
FI781313A (fi) 1978-10-29
ATA311378A (de) 1979-12-15
CS199726B2 (en) 1980-07-31
IE46627B1 (en) 1983-08-10
FR2388815A1 (fr) 1978-11-24
NO158506B (no) 1988-06-13
NZ187086A (en) 1981-05-15
AR227614A1 (es) 1982-11-30
MX5952E (es) 1984-09-06
BG34337A3 (en) 1983-08-15
FR2388815B1 (es) 1982-06-18
DK182878A (da) 1978-10-29
GB1574273A (en) 1980-09-03
NO781502L (no) 1978-10-31
PH16851A (en) 1984-03-19
AU522851B2 (en) 1982-07-01
IT1111469B (it) 1986-01-13
DE2818985A1 (de) 1978-11-02
CA1100962A (en) 1981-05-12
AT357674B (de) 1980-07-25
HU178105B (en) 1982-03-28
IE780844L (en) 1978-10-25
GR69966B (es) 1982-07-22
DD135908A5 (de) 1979-06-06
NL189669C (nl) 1993-06-16
US4183928A (en) 1980-01-15
IT7867986A0 (it) 1978-04-28
YU42477B (en) 1988-10-31
FI63410B (fi) 1983-02-28
PL110680B1 (en) 1980-07-31
NO158506C (no) 1988-09-21
NL7804628A (nl) 1978-10-31
PT67957B (en) 1980-03-05
AU3552778A (en) 1979-11-01
DE2818985C2 (de) 1995-08-17
ES469206A1 (es) 1979-09-16
IL54596A0 (en) 1978-07-31
YU103578A (en) 1983-06-30
SU784779A3 (ru) 1980-11-30
PT67957A (en) 1978-05-01
NL189669B (nl) 1993-01-18
CH640535A5 (de) 1984-01-13
PL206451A1 (pl) 1979-04-09

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Legal Events

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MM Patent lapsed
MM Patent lapsed

Owner name: SHINOGI & CO., LTD.