FI58635C - Foerfarande foer framstaellning av nya antimikrobiska pleuromutiliner - Google Patents
Foerfarande foer framstaellning av nya antimikrobiska pleuromutiliner Download PDFInfo
- Publication number
- FI58635C FI58635C FI2645/72A FI264572A FI58635C FI 58635 C FI58635 C FI 58635C FI 2645/72 A FI2645/72 A FI 2645/72A FI 264572 A FI264572 A FI 264572A FI 58635 C FI58635 C FI 58635C
- Authority
- FI
- Finland
- Prior art keywords
- carbon atoms
- deoxy
- alkyl
- solution
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/57—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
- C07C323/58—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups with amino groups bound to the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI794061A FI60204C (fi) | 1971-10-05 | 1979-12-27 | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara pleuromutiliner |
FI794060A FI60198C (fi) | 1971-10-05 | 1979-12-27 | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara pleuromutiliner |
Applications Claiming Priority (10)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH1445171A CH559719A5 (en) | 1971-10-05 | 1971-10-05 | Pleuromutilin derivs - with antibacterial activity |
CH1445071 | 1971-10-05 | ||
CH1445071A CH560180A5 (en) | 1971-10-05 | 1971-10-05 | Pleuromutilin derivs - with antibacterial activity |
CH1445171 | 1971-10-05 | ||
CH773972 | 1972-05-25 | ||
CH773872 | 1972-05-25 | ||
CH773872A CH572893A5 (en) | 1972-05-25 | 1972-05-25 | Pleuromutilin derivs - with antibacterial activity |
CH773972A CH568272A5 (en) | 1972-05-25 | 1972-05-25 | (Para-substd phenoxy- or phenylthio-acetoxy)-pleuromutilin deriv - prepd by reacting para-hydroxy or-mercapto cpds with e.g. aminoalkyl halides |
CH774072A CH575375A5 (hu) | 1972-05-25 | 1972-05-25 | |
CH774072 | 1972-05-25 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI58635B FI58635B (fi) | 1980-11-28 |
FI58635C true FI58635C (fi) | 1981-03-10 |
Family
ID=27509313
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI2645/72A FI58635C (fi) | 1971-10-05 | 1972-09-26 | Foerfarande foer framstaellning av nya antimikrobiska pleuromutiliner |
Country Status (20)
Country | Link |
---|---|
US (1) | US4278674A (hu) |
JP (1) | JPS577147B2 (hu) |
BE (1) | BE789629A (hu) |
BG (2) | BG21386A3 (hu) |
CA (1) | CA979447A (hu) |
DD (1) | DD100706A5 (hu) |
DE (2) | DE2265666C2 (hu) |
DK (1) | DK139720B (hu) |
FI (1) | FI58635C (hu) |
FR (1) | FR2157828B1 (hu) |
GB (1) | GB1410505A (hu) |
HU (1) | HU168436B (hu) |
IE (1) | IE37699B1 (hu) |
IL (1) | IL40494A (hu) |
NL (1) | NL177403C (hu) |
NO (3) | NO136459C (hu) |
OA (1) | OA04192A (hu) |
PH (1) | PH11870A (hu) |
RO (2) | RO67479A (hu) |
SE (3) | SE398348B (hu) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3987194A (en) * | 1975-05-12 | 1976-10-19 | E. R. Squibb & Sons, Inc. | Use of pleuromutilin derivatives for the treatment of swine dysentery |
DE2823712C2 (de) | 1978-05-31 | 1987-04-09 | Sandoz-Patent-GmbH, 7850 Lörrach | Verfahren zur Herstellung von Pleuromutilin-Derivaten |
FR2428030A1 (fr) * | 1978-06-06 | 1980-01-04 | Sandoz Sa | Procede de preparation de derives de la pleuromutiline |
JPS56168463A (en) * | 1980-05-30 | 1981-12-24 | Iwao Koyama | Telephone set |
LU82738A1 (fr) * | 1980-08-29 | 1982-05-10 | Continental Pharma | Derives d'aminothiols,leur preparation et utilisation ainsi que compositions contenant ces derives |
JPS60121870A (ja) * | 1983-12-06 | 1985-06-29 | Matsushita Electric Ind Co Ltd | インタ−ホン装置 |
JPS62137952A (ja) * | 1985-12-12 | 1987-06-20 | Sakuragi Kunio | 電話機 |
JPH0418190Y2 (hu) * | 1986-09-19 | 1992-04-23 | ||
JPH01105238U (hu) * | 1988-01-05 | 1989-07-14 | ||
AU715229B2 (en) * | 1996-01-03 | 2000-01-20 | Smithkline Beecham Plc | Carbamoyloxy derivatives of mutiline and their use as antibacterials |
FR2746012B1 (fr) * | 1996-03-13 | 1998-05-22 | Utilisation de la tiamuline pour la preparation d'un medicament comme agent de reversion de la multichimioresistance cancereuse | |
UY25225A1 (es) | 1997-10-29 | 2000-12-29 | Smithkline Beecham Plc | Derivados de pleuromutilina utiles como agentes antimicrobianos |
WO2000027790A1 (en) * | 1998-11-11 | 2000-05-18 | Smithkline Beecham P.L.C. | Mutilin compounds |
AU3036200A (en) * | 1998-12-18 | 2000-07-12 | Smithkline Beecham Plc | Mutilin 14-ester derivatives having antibacterial activity |
GB9912657D0 (en) * | 1999-06-01 | 1999-07-28 | Smithkline Beecham Plc | Novel compounds |
GB9918037D0 (en) * | 1999-07-30 | 1999-09-29 | Biochemie Gmbh | Organic compounds |
GB0017031D0 (en) * | 2000-07-11 | 2000-08-30 | Biochemie Gmbh | Antimicrobials |
PE20020676A1 (es) * | 2000-09-13 | 2002-08-27 | Biochemie Gmbh | Compuestos de mutilina como antibacterianos |
GB0207495D0 (en) * | 2002-03-28 | 2002-05-08 | Biochemie Gmbh | Organic compounds |
GB0308114D0 (en) * | 2003-04-08 | 2003-05-14 | Glaxo Group Ltd | Novel compounds |
EP1663220B1 (en) * | 2003-09-03 | 2009-12-02 | Glaxo Group Limited | Novel process for the preparation of pleuromutilin derivatives |
GB0504314D0 (en) * | 2005-03-02 | 2005-04-06 | Glaxo Group Ltd | Novel polymorph |
JP2008534444A (ja) * | 2005-03-10 | 2008-08-28 | スミスクライン・ビーチャム・コーポレイション | 新規な方法 |
GB0513058D0 (en) * | 2005-06-27 | 2005-08-03 | Sandoz Ag | Organic compounds |
EP1808431A1 (en) * | 2006-01-16 | 2007-07-18 | Nabriva Therapeutics Forschungs GmbH | Mutilin derivatives and their use as pharmaceutical |
WO2008117796A1 (ja) * | 2007-03-28 | 2008-10-02 | Dainippon Sumitomo Pharma Co., Ltd. | 新規ムチリン誘導体 |
CN101434567B (zh) * | 2008-12-19 | 2012-10-24 | 李扬 | 一种二乙氨基乙硫醇的制备方法 |
CN103709115A (zh) * | 2012-10-09 | 2014-04-09 | 山东亨利医药科技有限责任公司 | 截短侧耳素类抗生素衍生物 |
CN104854093B (zh) | 2012-12-03 | 2016-10-12 | 辉瑞大药厂 | 新的选择性雄激素受体调节剂 |
CN104447449B (zh) * | 2014-12-30 | 2016-06-15 | 陕西师范大学 | 一锅法合成泰妙菌素的方法 |
CN110981769B (zh) * | 2019-12-19 | 2022-02-18 | 江苏威凌生化科技有限公司 | 一种制备泰秒菌素的方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AT301753B (de) * | 1969-07-25 | 1972-09-25 | Biochemie Gmbh | Verfahren zur Herstellung neuer Pleuromutilin-Derivate |
US4107164A (en) * | 1971-10-05 | 1978-08-15 | Sandoz Ltd. | Certain pleuromulilin ester derivatives |
US3919290A (en) * | 1972-10-03 | 1975-11-11 | Sandoz Ltd | Substituted 14-desoxy-mutilins |
US4032530A (en) * | 1971-10-05 | 1977-06-28 | Sandoz Ltd. | Certain pleuromutilins |
-
0
- BE BE789629D patent/BE789629A/xx not_active IP Right Cessation
-
1972
- 1972-09-26 SE SE7212374A patent/SE398348B/xx unknown
- 1972-09-26 DK DK475372AA patent/DK139720B/da not_active IP Right Cessation
- 1972-09-26 FI FI2645/72A patent/FI58635C/fi active
- 1972-09-27 NO NO3453/72A patent/NO136459C/no unknown
- 1972-09-29 PH PH13949A patent/PH11870A/en unknown
- 1972-09-29 NL NLAANVRAGE7213254,A patent/NL177403C/xx not_active IP Right Cessation
- 1972-10-02 DE DE2265666A patent/DE2265666C2/de not_active Expired
- 1972-10-02 GB GB4525972A patent/GB1410505A/en not_active Expired
- 1972-10-02 DE DE2248237A patent/DE2248237C2/de not_active Expired
- 1972-10-03 HU HUSA2407A patent/HU168436B/hu unknown
- 1972-10-03 IE IE1339/72A patent/IE37699B1/xx unknown
- 1972-10-03 RO RO7281506A patent/RO67479A/ro unknown
- 1972-10-03 CA CA153,116A patent/CA979447A/en not_active Expired
- 1972-10-03 RO RO7281505A patent/RO67478A/ro unknown
- 1972-10-04 OA OA54711A patent/OA04192A/xx unknown
- 1972-10-04 IL IL40494A patent/IL40494A/en unknown
- 1972-10-04 BG BG23481A patent/BG21386A3/xx unknown
- 1972-10-04 JP JP9913872A patent/JPS577147B2/ja not_active Expired
- 1972-10-04 BG BG23482A patent/BG20773A3/xx unknown
- 1972-10-05 DD DD166051A patent/DD100706A5/xx unknown
- 1972-10-05 FR FR7235340A patent/FR2157828B1/fr not_active Expired
-
1973
- 1973-12-04 NO NO4617/73A patent/NO136837C/no unknown
- 1973-12-04 NO NO4618/73A patent/NO137440C/no unknown
-
1975
- 1975-08-26 SE SE7509457A patent/SE419984B/xx unknown
- 1975-08-26 SE SE7509456A patent/SE424074B/xx unknown
-
1979
- 1979-11-29 US US06/098,333 patent/US4278674A/en not_active Expired - Lifetime
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