NO136459C - Analogifremgangsm}te for fremstilling av antimikrobielt virksomme pleuromutiliner. - Google Patents

Analogifremgangsm}te for fremstilling av antimikrobielt virksomme pleuromutiliner.

Info

Publication number
NO136459C
NO136459C NO3453/72A NO345372A NO136459C NO 136459 C NO136459 C NO 136459C NO 3453/72 A NO3453/72 A NO 3453/72A NO 345372 A NO345372 A NO 345372A NO 136459 C NO136459 C NO 136459C
Authority
NO
Norway
Prior art keywords
pleuromutilines
preparation
antimicrobially active
analogical procedure
analogical
Prior art date
Application number
NO3453/72A
Other languages
English (en)
Other versions
NO136459B (no
Inventor
Helmut Egger
Hellmuth Reinshagen
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27509313&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO136459(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from CH1445171A external-priority patent/CH559719A5/de
Priority claimed from CH1445071A external-priority patent/CH560180A5/de
Priority claimed from CH773872A external-priority patent/CH572893A5/xx
Priority claimed from CH774072A external-priority patent/CH575375A5/de
Priority claimed from CH773972A external-priority patent/CH568272A5/de
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of NO136459B publication Critical patent/NO136459B/no
Publication of NO136459C publication Critical patent/NO136459C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/57—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C323/58—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups with amino groups bound to the carbon skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO3453/72A 1971-10-05 1972-09-27 Analogifremgangsm}te for fremstilling av antimikrobielt virksomme pleuromutiliner. NO136459C (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CH1445171A CH559719A5 (en) 1971-10-05 1971-10-05 Pleuromutilin derivs - with antibacterial activity
CH1445071A CH560180A5 (en) 1971-10-05 1971-10-05 Pleuromutilin derivs - with antibacterial activity
CH773872A CH572893A5 (en) 1972-05-25 1972-05-25 Pleuromutilin derivs - with antibacterial activity
CH774072A CH575375A5 (no) 1972-05-25 1972-05-25
CH773972A CH568272A5 (en) 1972-05-25 1972-05-25 (Para-substd phenoxy- or phenylthio-acetoxy)-pleuromutilin deriv - prepd by reacting para-hydroxy or-mercapto cpds with e.g. aminoalkyl halides

Publications (2)

Publication Number Publication Date
NO136459B NO136459B (no) 1977-05-31
NO136459C true NO136459C (no) 1977-09-07

Family

ID=27509313

Family Applications (3)

Application Number Title Priority Date Filing Date
NO3453/72A NO136459C (no) 1971-10-05 1972-09-27 Analogifremgangsm}te for fremstilling av antimikrobielt virksomme pleuromutiliner.
NO4617/73A NO136837C (no) 1971-10-05 1973-12-04 Analogifremgangsm}te for fremstilling av terapeutisk aktive pleuromutiliner
NO4618/73A NO137440C (no) 1971-10-05 1973-12-04 Analogifremgangsmaate for fremstilling av terapeutisk aktive pleuromutiliner

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO4617/73A NO136837C (no) 1971-10-05 1973-12-04 Analogifremgangsm}te for fremstilling av terapeutisk aktive pleuromutiliner
NO4618/73A NO137440C (no) 1971-10-05 1973-12-04 Analogifremgangsmaate for fremstilling av terapeutisk aktive pleuromutiliner

Country Status (20)

Country Link
US (1) US4278674A (no)
JP (1) JPS577147B2 (no)
BE (1) BE789629A (no)
BG (2) BG20773A3 (no)
CA (1) CA979447A (no)
DD (1) DD100706A5 (no)
DE (2) DE2265666C2 (no)
DK (1) DK139720B (no)
FI (1) FI58635C (no)
FR (1) FR2157828B1 (no)
GB (1) GB1410505A (no)
HU (1) HU168436B (no)
IE (1) IE37699B1 (no)
IL (1) IL40494A (no)
NL (1) NL177403C (no)
NO (3) NO136459C (no)
OA (1) OA04192A (no)
PH (1) PH11870A (no)
RO (2) RO67479A (no)
SE (3) SE398348B (no)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987194A (en) * 1975-05-12 1976-10-19 E. R. Squibb & Sons, Inc. Use of pleuromutilin derivatives for the treatment of swine dysentery
DE2823712C2 (de) 1978-05-31 1987-04-09 Sandoz-Patent-GmbH, 7850 Lörrach Verfahren zur Herstellung von Pleuromutilin-Derivaten
FR2428030A1 (fr) * 1978-06-06 1980-01-04 Sandoz Sa Procede de preparation de derives de la pleuromutiline
JPS56168463A (en) * 1980-05-30 1981-12-24 Iwao Koyama Telephone set
LU82738A1 (fr) * 1980-08-29 1982-05-10 Continental Pharma Derives d'aminothiols,leur preparation et utilisation ainsi que compositions contenant ces derives
JPS60121870A (ja) * 1983-12-06 1985-06-29 Matsushita Electric Ind Co Ltd インタ−ホン装置
JPS62137952A (ja) * 1985-12-12 1987-06-20 Sakuragi Kunio 電話機
JPH0418190Y2 (no) * 1986-09-19 1992-04-23
JPH01105238U (no) * 1988-01-05 1989-07-14
TR199801282T2 (xx) * 1996-01-03 1998-12-21 Smithkline Beecham P.L.C. Mutilin'in karbamoiloksi t�revleri ve antibakteriyel olarak kullan�m�.
FR2746012B1 (fr) * 1996-03-13 1998-05-22 Utilisation de la tiamuline pour la preparation d'un medicament comme agent de reversion de la multichimioresistance cancereuse
UY25225A1 (es) * 1997-10-29 2000-12-29 Smithkline Beecham Plc Derivados de pleuromutilina utiles como agentes antimicrobianos
WO2000027790A1 (en) * 1998-11-11 2000-05-18 Smithkline Beecham P.L.C. Mutilin compounds
AU3036200A (en) * 1998-12-18 2000-07-12 Smithkline Beecham Plc Mutilin 14-ester derivatives having antibacterial activity
GB9912657D0 (en) * 1999-06-01 1999-07-28 Smithkline Beecham Plc Novel compounds
GB9918037D0 (en) 1999-07-30 1999-09-29 Biochemie Gmbh Organic compounds
GB0017031D0 (en) * 2000-07-11 2000-08-30 Biochemie Gmbh Antimicrobials
PE20020676A1 (es) * 2000-09-13 2002-08-27 Biochemie Gmbh Compuestos de mutilina como antibacterianos
GB0207495D0 (en) * 2002-03-28 2002-05-08 Biochemie Gmbh Organic compounds
GB0308114D0 (en) * 2003-04-08 2003-05-14 Glaxo Group Ltd Novel compounds
US7875630B2 (en) * 2003-09-03 2011-01-25 Glaxo Group Limited Process salts compositions and use
GB0504314D0 (en) * 2005-03-02 2005-04-06 Glaxo Group Ltd Novel polymorph
US20080171766A1 (en) * 2005-03-10 2008-07-17 Smithkline Beecham Corporation Novel Method
GB0513058D0 (en) * 2005-06-27 2005-08-03 Sandoz Ag Organic compounds
EP1808431A1 (en) * 2006-01-16 2007-07-18 Nabriva Therapeutics Forschungs GmbH Mutilin derivatives and their use as pharmaceutical
WO2008117796A1 (ja) * 2007-03-28 2008-10-02 Dainippon Sumitomo Pharma Co., Ltd. 新規ムチリン誘導体
CN101434567B (zh) * 2008-12-19 2012-10-24 李扬 一种二乙氨基乙硫醇的制备方法
CN103709115A (zh) * 2012-10-09 2014-04-09 山东亨利医药科技有限责任公司 截短侧耳素类抗生素衍生物
DK2925725T3 (en) 2012-12-03 2017-01-16 Pfizer androgen receptor modulators
CN104447449B (zh) * 2014-12-30 2016-06-15 陕西师范大学 一锅法合成泰妙菌素的方法
CN110981769B (zh) * 2019-12-19 2022-02-18 江苏威凌生化科技有限公司 一种制备泰秒菌素的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT301753B (de) * 1969-07-25 1972-09-25 Biochemie Gmbh Verfahren zur Herstellung neuer Pleuromutilin-Derivate
US4107164A (en) * 1971-10-05 1978-08-15 Sandoz Ltd. Certain pleuromulilin ester derivatives
US4032530A (en) * 1971-10-05 1977-06-28 Sandoz Ltd. Certain pleuromutilins
US3919290A (en) * 1972-10-03 1975-11-11 Sandoz Ltd Substituted 14-desoxy-mutilins

Also Published As

Publication number Publication date
SE419984B (sv) 1981-09-07
RO67479A (ro) 1981-06-21
DK139720C (no) 1979-10-01
FI58635C (fi) 1981-03-10
NO136837C (no) 1977-11-16
IL40494A (en) 1976-01-30
NO136837B (no) 1977-08-08
FR2157828A1 (no) 1973-06-08
JPS4844244A (no) 1973-06-26
NO137440C (no) 1978-03-01
PH11870A (en) 1978-08-04
FI58635B (fi) 1980-11-28
SE398348B (sv) 1977-12-19
OA04192A (fr) 1979-12-31
NO137440B (no) 1977-11-21
DE2248237A1 (de) 1973-04-12
CA979447A (en) 1975-12-09
RO67478A (ro) 1980-03-15
IE37699L (en) 1973-04-05
SE424074B (sv) 1982-06-28
BG20773A3 (bg) 1975-12-20
JPS577147B2 (no) 1982-02-09
NL177403C (nl) 1985-09-16
US4278674A (en) 1981-07-14
DE2265666C2 (de) 1983-02-03
NL7213254A (no) 1973-04-09
BE789629A (fr) 1973-04-03
DK139720B (da) 1979-04-02
SE7509457L (sv) 1975-08-26
DE2248237C2 (de) 1983-02-10
NO136459B (no) 1977-05-31
DD100706A5 (no) 1973-10-05
SE7509456L (sv) 1975-08-26
BG21386A3 (bg) 1976-05-20
NL177403B (nl) 1985-04-16
IL40494A0 (en) 1972-12-29
FR2157828B1 (no) 1975-11-28
GB1410505A (en) 1975-10-15
IE37699B1 (en) 1977-09-28
HU168436B (no) 1976-04-28

Similar Documents

Publication Publication Date Title
NO136459C (no) Analogifremgangsm}te for fremstilling av antimikrobielt virksomme pleuromutiliner.
SE382485B (sv) Anordning for framstellning av tunnveggiga bikakskonstruktioner.
NO136298C (no) Analogifremgangsm}te til fremstilling av antibakterielt virksomme imidazolderivater
NO136793C (no) Analogifremgangsm}te til fremstilling av terapeutisk virksomme substituerte 1,2,4-triazolderivater.
SE389331B (sv) Forfarande for framstellning av vissa angivna 2,2-metylendifenoler.
NO136045C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive pyridazinoner.
NO136492C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive 3-(trisubstituert benzoyl)-propionsyre.
NO147916C (no) Fremgangsmaate for fremstilling av 3-metylen-cefalosporin-forbindelser.
NO136251C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive pyridazin-derivater.
NO136712C (no) Analogifremgangsm}te ved fremstilling av terapeutisk aktive benzoxazolforbindelser.
NO136926C (no) Analogifremgangsm}te til fremstilling av terapeutisk aktive papaverinanaloger
SE7505279L (sv) Forfarande for framstellning av hydroxipyrimidiner.
NO138025C (no) Analogifremgangsmaate til fremstilling av antimykotisk virksomme 1-etyl-imidazoler
SE386175B (sv) Forfarande for framstellning av 1,4-bis-acylpiperaziner
SE406587B (sv) Forfarande for framstellning av 4-hydroximetyl-1-keto-1,2-dihydroftalazin
NO137093C (no) Fremgangsm}te til fremstilling av 2,4-diamino-5-benzylpyrimidiner
NO141851C (no) Fremgangsmaate for fremstilling av metyl-3-(2-kinoksalinylmetylen)-karbazat-n1.n4-dioksyd.
SE394677B (sv) Forfarande for framstellning av 4-hydroxi-2h-1-bensotiopyran-3-karboxanilid-1,1-dioxider
SE403612B (sv) Analogiforfarande for framstellning av antibakteriellt aktiva hexametylen-bis-biguanider
DK132700C (da) Herbicidt virksomme forbindelser
SE387936B (sv) Forfarande for framstellning av substituerade metoxiaminer
NO136410C (no) Analogifremgangsm}te til fremstilling av antidiabetisk virksomme 3-metyl-pyrazol-5-karboksamider.
NO139173C (no) Analogifremgangsmaate for fremstilling av antimikrobielt aktive 2-kinoksalin-karboksamid-1,4-dioksyder
NO136198C (no) Analogifremgangsm}te ved fremstilling av terapeutisk aktivt 16-carboxy-17-methoxy-eburnan.
SE390025B (sv) Forfarande for framstellning av 3 alfa-hydroxi-19-5 alfa-pregnan-11,20-dion