ES543115A0 - Un nuevo procedimiento para la preparacion de pirido-imidazorifamicinas - Google Patents
Un nuevo procedimiento para la preparacion de pirido-imidazorifamicinasInfo
- Publication number
- ES543115A0 ES543115A0 ES543115A ES543115A ES543115A0 ES 543115 A0 ES543115 A0 ES 543115A0 ES 543115 A ES543115 A ES 543115A ES 543115 A ES543115 A ES 543115A ES 543115 A0 ES543115 A0 ES 543115A0
- Authority
- ES
- Spain
- Prior art keywords
- imidazorifamicinas
- pirido
- preparation
- new procedure
- procedure
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT03463/84A IT1199374B (it) | 1984-05-15 | 1984-05-15 | Processo per la preparazione di pirido-imidazo-rifamicine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8603489A1 ES8603489A1 (es) | 1986-01-01 |
| ES543115A0 true ES543115A0 (es) | 1986-01-01 |
Family
ID=11107845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES543115A Granted ES543115A0 (es) | 1984-05-15 | 1985-05-14 | Un nuevo procedimiento para la preparacion de pirido-imidazorifamicinas |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4557866A (OSRAM) |
| EP (1) | EP0161534B1 (OSRAM) |
| JP (1) | JPS60252483A (OSRAM) |
| AR (1) | AR241913A1 (OSRAM) |
| AT (1) | ATE46512T1 (OSRAM) |
| AU (1) | AU568934B2 (OSRAM) |
| CA (1) | CA1215708A (OSRAM) |
| DE (1) | DE3573120D1 (OSRAM) |
| DK (1) | DK162647C (OSRAM) |
| ES (1) | ES543115A0 (OSRAM) |
| FI (1) | FI81101C (OSRAM) |
| GR (1) | GR851144B (OSRAM) |
| IE (1) | IE58392B1 (OSRAM) |
| IT (1) | IT1199374B (OSRAM) |
| NO (1) | NO164242C (OSRAM) |
| PH (1) | PH22007A (OSRAM) |
| PT (1) | PT80446B (OSRAM) |
| ZA (1) | ZA852971B (OSRAM) |
Families Citing this family (62)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7048906B2 (en) | 1995-05-17 | 2006-05-23 | Cedars-Sinai Medical Center | Methods of diagnosing and treating small intestinal bacterial overgrowth (SIBO) and SIBO-related conditions |
| US6861053B1 (en) | 1999-08-11 | 2005-03-01 | Cedars-Sinai Medical Center | Methods of diagnosing or treating irritable bowel syndrome and other disorders caused by small intestinal bacterial overgrowth |
| WO2003051299A2 (en) * | 2001-12-13 | 2003-06-26 | Activbiotics, Inc. | Sulfhydryl rifamycins and uses thereof |
| US7906542B2 (en) | 2004-11-04 | 2011-03-15 | Alfa Wassermann, S.P.A. | Pharmaceutical compositions comprising polymorphic forms α, β, and γ of rifaximin |
| ITMI20032144A1 (it) * | 2003-11-07 | 2005-05-08 | Alfa Wassermann Spa | Forme polimorfe di rifaximina, processi per ottenerle e |
| US7923553B2 (en) | 2003-11-07 | 2011-04-12 | Alfa Wassermann, S.P.A. | Processes for the production of polymorphic forms of rifaximin |
| US7902206B2 (en) | 2003-11-07 | 2011-03-08 | Alfa Wassermann, S.P.A. | Polymorphic forms α, β and γ of rifaximin |
| US20080262024A1 (en) * | 2003-11-07 | 2008-10-23 | Giuseppe Claudio Viscomi | Rifaximin compositions and method of use |
| US8003118B2 (en) * | 2005-03-02 | 2011-08-23 | Kodsi Robert E | Use of rifaximin for the prevention of aspiration pneumonia and/or sepsis |
| US20060210492A1 (en) * | 2005-03-02 | 2006-09-21 | Kodsi Robert E | Use of rifaximin for treatment and prevention of periodontal conditions |
| US20060210483A1 (en) * | 2005-03-02 | 2006-09-21 | Kodsi Robert E | Non-systemic antibiotic formulations and related method of use and treatment of upper respiratory infections |
| PT1698630E (pt) | 2005-03-03 | 2014-09-15 | Alfa Wassermann Spa | Novas formas polimorfas de rifaximina, processos para a sua produção e a sua utilização nas preparações medicinais |
| ITBO20050123A1 (it) | 2005-03-07 | 2005-06-06 | Alfa Wassermann Spa | Formulazioni farmaceutiche gastroresistenti contenenti rifaximina |
| MX2008011305A (es) | 2006-03-09 | 2009-02-10 | Salix Pharmaceuticals Inc | Preparacion anti-disfunsion rectal con rifaximina. |
| EP2054066B1 (en) | 2006-08-02 | 2015-04-15 | Salix Pharmaceuticals, Inc. | Methods for treatment of radiation enteritis |
| ITMI20061692A1 (it) | 2006-09-05 | 2008-03-06 | Alfa Wassermann Spa | Uso di polioli per ottenere forme polimorfe stabili di rifaximina |
| AU2007298733B2 (en) * | 2006-09-22 | 2012-11-08 | Cipla Limited | Rifaximin |
| US20080159987A1 (en) * | 2007-01-03 | 2008-07-03 | Leonard Weinstock | Use of Rifaximin for the Treatment of Restless Legs Syndrome |
| US20080161337A1 (en) * | 2007-01-03 | 2008-07-03 | Leonard Weinstock | Use of Rifaximin for the Treatment of Chronic Prostatitis |
| ITMI20071241A1 (it) * | 2007-06-20 | 2008-12-21 | Solmag S P A | Processo per la preparazione di rifaximina amorfa e rifaximina amorfa cosi' ottenuta |
| US7709634B2 (en) | 2007-09-20 | 2010-05-04 | Apotex Pharmachem Inc. | Amorphous form of rifaximin and processes for its preparation |
| SG188931A1 (en) | 2008-02-25 | 2013-04-30 | Salix Pharmaceuticals Ltd | Forms of rifaximin and uses thereof |
| US8486956B2 (en) | 2008-02-25 | 2013-07-16 | Salix Pharmaceuticals, Ltd | Forms of rifaximin and uses thereof |
| US11779571B2 (en) | 2008-02-26 | 2023-10-10 | Salix Pharmaceuticals, Inc. | Methods for treating irritable bowel syndrome (IBS) |
| DK2252148T3 (da) | 2008-02-26 | 2019-05-06 | Salix Pharmaceuticals Ltd | Fremgangsmåder til behandling af irritabel tarmsyndrom |
| HRP20140939T1 (hr) | 2008-05-07 | 2014-11-21 | Salix Pharmaceuticals, Ltd. | Davanje preparata za äśišä†enje crijeva i antibiotika za lijeäśenje bolesti crijeva |
| CN101585843B (zh) * | 2008-05-21 | 2011-07-06 | 重庆赛诺生物药业股份有限公司 | 一种利福昔明的制备工艺 |
| EP3628319B1 (en) | 2008-10-02 | 2024-02-14 | Salix Pharmaceuticals, Ltd. | Treatment of hepatic encephalopathy using rifaximin |
| US12285414B2 (en) | 2008-10-02 | 2025-04-29 | Salix Pharmaceuticals, Inc. | Methods of treating hepatic encephalopathy |
| US7928115B2 (en) | 2008-10-02 | 2011-04-19 | Salix Pharmaceuticals, Ltd. | Methods of treating travelers diarrhea and hepatic encephalopathy |
| US20110035232A1 (en) * | 2008-10-02 | 2011-02-10 | Salix Pharmaceuticals, Ltd. | Methods of treating hepatic encephalopathy |
| KR101906177B1 (ko) | 2008-12-10 | 2018-10-10 | 시플라 리미티드 | 리팍시민 복합체 |
| IT1397617B1 (it) * | 2009-04-20 | 2013-01-18 | Alfa Wassermann Spa | Nuovi derivati della rifamicina |
| KR20170036116A (ko) | 2009-06-02 | 2017-03-31 | 샐릭스 파마슈티컬스 리미티드 | 간성 뇌병증의 치료방법 |
| NZ598671A (en) | 2009-09-13 | 2014-02-28 | Salix Pharmaceuticals Ltd | Methods for treating irritable bowel syndrome (ibs) |
| AU2010320656B2 (en) | 2009-11-23 | 2015-07-30 | Cipla Limited | Topical foam composition |
| US8952159B2 (en) | 2009-12-28 | 2015-02-10 | Silvio Massimo Lavagna | Method for the production of amorphous rifaximin |
| CA2789929C (en) | 2010-02-18 | 2019-11-26 | Salix Pharmaceuticals, Ltd. | Methods for treating infection |
| IT1398550B1 (it) | 2010-03-05 | 2013-03-01 | Alfa Wassermann Spa | Formulazioni comprendenti rifaximina utili per ottenere un effetto prolungato nel tempo |
| WO2011156897A2 (en) * | 2010-06-16 | 2011-12-22 | Apotex Pharmachem Inc. | Polymorphic forms of rifaximin |
| SI2593463T1 (sl) | 2010-07-12 | 2020-10-30 | Salix Pharmaceuticals, Inc. | Formulacije rifaksimina in njihove uporabe |
| WO2012035544A2 (en) | 2010-09-13 | 2012-03-22 | Sequent Scientific Ltd. | A novel polymorphic form of rifaximin and process for its preparation |
| PT2672970T (pt) | 2011-02-11 | 2018-10-11 | Salix Pharmaceuticals Ltd | Formas de rifaximina e suas utilizações |
| CA2834829A1 (en) | 2011-05-02 | 2012-11-08 | Ranbaxy Laboratories Limited | Rifaximin dimethylformamide solvate |
| WO2012155981A1 (en) | 2011-05-19 | 2012-11-22 | Friulchem Spa | New process for the synthesis of rifaximin and a new pseudo-crystalline form of rifaximin obtained thereby |
| ITBO20110461A1 (it) | 2011-07-29 | 2013-01-30 | Alfa Wassermann Spa | Composizioni farmaceutiche comprendenti rifaximina, processi per la loro preparazione e loro uso nel trattamento di infezioni vaginali. |
| ES2986825T3 (es) | 2011-11-02 | 2024-11-12 | Salix Pharmaceuticals Inc | Rifaximina para la repetición de tratamiento del síndrome del intestino irritable con predominio de diarrea |
| CA2876737A1 (en) | 2012-06-13 | 2013-12-19 | Apotex Pharmachem Inc. | Polymorphic forms of rifaximin |
| ITBO20120368A1 (it) | 2012-07-06 | 2014-01-07 | Alfa Wassermann Spa | Composizioni comprendenti rifaximina e amminoacidi, cristalli di rifaximina derivanti da tali composizioni e loro uso. |
| JP2016516988A (ja) | 2013-03-15 | 2016-06-09 | アルファ ワッセルマン ソシエタ ペル アチオニAlfa Wassermann S.P.A. | 膣感染症を診断するための方法 |
| EA201591267A1 (ru) | 2013-03-15 | 2016-03-31 | Альфа Вассерманн С.П.А. | Рифаксимин для применения в лечении вагинальных инфекций |
| JP6433980B2 (ja) | 2013-04-12 | 2018-12-05 | アルファシグマ ソシエタ ペル アチオニ | Nsaid投与並びに関連する組成物、方法及びシステム |
| US9018225B1 (en) | 2013-07-26 | 2015-04-28 | Novel Laboratories | Rifaximin crystalline forms and methods of preparation thereof |
| ITMI20131307A1 (it) | 2013-08-02 | 2015-02-02 | A M S A Anonima Materie Sint & Affini S P A | Processo per la preparazione di refaximina k |
| CN103509038B (zh) * | 2013-09-30 | 2016-01-20 | 浙江思贤制药有限公司 | 一种新晶型利福昔明ζ及其制备方法 |
| EP2927235B1 (en) | 2014-03-31 | 2017-02-08 | Euticals S.P.A. | Polymorphic mixture of rifaximin and its use for the preparation of solid formulations |
| MX375805B (es) | 2014-05-04 | 2025-03-07 | Salix Pharmaceuticals Inc | Microbiota ibs y sus usos. |
| ES2742106T3 (es) | 2014-05-12 | 2020-02-13 | Alfasigma Spa | Nueva forma de cristal solvatado de rifaximina, producción, composiciones y usos de la misma |
| EP2982764A1 (en) | 2014-08-05 | 2016-02-10 | ALFA WASSERMANN S.p.A. | Identification of vaginal bacteria |
| US9988398B2 (en) | 2016-06-07 | 2018-06-05 | Cadila Healthcare Limited | Crystalline form of rifaximin and process for its preparation |
| CN110072525B (zh) | 2016-09-30 | 2022-12-02 | 萨利克斯药品公司 | 利福昔明的固态分散形式 |
| EP3645539B1 (en) * | 2017-06-26 | 2021-04-07 | Biofer S.p.A. | Pyrido-imidazo rifamycin derivatives as antibacterial agent |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1154655B (it) * | 1980-05-22 | 1987-01-21 | Alfa Farmaceutici Spa | Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica |
-
1984
- 1984-05-15 IT IT03463/84A patent/IT1199374B/it active
-
1985
- 1985-04-19 DE DE8585104790T patent/DE3573120D1/de not_active Expired
- 1985-04-19 ZA ZA852971A patent/ZA852971B/xx unknown
- 1985-04-19 AT AT85104790T patent/ATE46512T1/de not_active IP Right Cessation
- 1985-04-19 EP EP85104790A patent/EP0161534B1/en not_active Expired
- 1985-04-25 PH PH32186A patent/PH22007A/en unknown
- 1985-04-26 US US06/727,521 patent/US4557866A/en not_active Expired - Lifetime
- 1985-04-29 CA CA000480321A patent/CA1215708A/en not_active Expired
- 1985-05-13 PT PT80446A patent/PT80446B/pt unknown
- 1985-05-13 GR GR851144A patent/GR851144B/el unknown
- 1985-05-14 DK DK214685A patent/DK162647C/da not_active IP Right Cessation
- 1985-05-14 NO NO851921A patent/NO164242C/no not_active IP Right Cessation
- 1985-05-14 IE IE119185A patent/IE58392B1/en not_active IP Right Cessation
- 1985-05-14 ES ES543115A patent/ES543115A0/es active Granted
- 1985-05-14 JP JP60102528A patent/JPS60252483A/ja active Granted
- 1985-05-14 FI FI851907A patent/FI81101C/fi not_active IP Right Cessation
- 1985-05-15 AU AU42515/85A patent/AU568934B2/en not_active Expired
- 1985-05-15 AR AR85300385A patent/AR241913A1/es active
Also Published As
| Publication number | Publication date |
|---|---|
| AR241913A1 (es) | 1993-01-29 |
| ES8603489A1 (es) | 1986-01-01 |
| EP0161534B1 (en) | 1989-09-20 |
| DK214685D0 (da) | 1985-05-14 |
| US4557866A (en) | 1985-12-10 |
| PT80446A (en) | 1985-06-01 |
| EP0161534A3 (en) | 1987-03-04 |
| CA1215708A (en) | 1986-12-23 |
| AU568934B2 (en) | 1988-01-14 |
| NO164242B (no) | 1990-06-05 |
| GR851144B (OSRAM) | 1985-11-25 |
| DK162647B (da) | 1991-11-25 |
| PH22007A (en) | 1988-05-02 |
| NO851921L (no) | 1985-11-18 |
| FI81101B (fi) | 1990-05-31 |
| DE3573120D1 (en) | 1989-10-26 |
| DK162647C (da) | 1992-04-13 |
| NO164242C (no) | 1990-09-12 |
| FI81101C (fi) | 1990-09-10 |
| ZA852971B (en) | 1985-12-24 |
| ATE46512T1 (de) | 1989-10-15 |
| IT8403463A0 (it) | 1984-05-15 |
| IE58392B1 (en) | 1993-09-08 |
| JPH0469634B2 (OSRAM) | 1992-11-06 |
| AU4251585A (en) | 1985-11-21 |
| PT80446B (pt) | 1987-11-11 |
| DK214685A (da) | 1985-11-16 |
| FI851907A0 (fi) | 1985-05-14 |
| EP0161534A2 (en) | 1985-11-21 |
| FI851907L (fi) | 1985-11-16 |
| JPS60252483A (ja) | 1985-12-13 |
| IT1199374B (it) | 1988-12-30 |
| IE851191L (en) | 1985-11-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES543115A0 (es) | Un nuevo procedimiento para la preparacion de pirido-imidazorifamicinas | |
| ES547840A0 (es) | Un procedimiento para la preparacion de alquilsulfonamidofe-nilalquilaminas | |
| ES539852A0 (es) | Un nuevo procedimiento para la preparacion de nuevos derivados. de carbazolona. | |
| ES557126A0 (es) | Un procedimiento para la preparacion de triazolobenzodiazepinas | |
| ES557364A0 (es) | Un procedimiento para la preparacion de nuevas benzamidas sustituidas | |
| ES541781A0 (es) | Un procedimiento para la preparacion de nuevos benzotiopenos. | |
| ES551552A0 (es) | Un procedimiento para la preparacion de nuevos compuestos de sulfonilurea | |
| ES548033A0 (es) | Un procedimiento para la preparacion de nuevos derivados pe-nem | |
| ES540200A0 (es) | Un procedimiento para la preparacion de acidos 7-amino-3-me-til sustituido-3-defem-4-carboxilicos | |
| ES543116A0 (es) | Un nuevo procedimiento para la preparacion de imidazorrifa- micinas | |
| ES553602A0 (es) | Un procedimiento para la preparacion de nuevas quinazolindionas | |
| ES545298A0 (es) | Un procedimiento para la preparacion de 4-amino-2-fenilqui- nolinas | |
| ES551755A0 (es) | Un procedimiento para la preparacion de derivados de d4-y-d5-androsteno nuevos | |
| ES547265A0 (es) | Un nuevo procedimiento para la preparacion de pirido-imida- zo-rifamicinas | |
| ES551508A0 (es) | Un procedimiento para la preparacion de nuevas sulfonilureas | |
| ES541277A0 (es) | Procedimiento para la preparacion de un nuevo derivado de lafructosa | |
| ES541450A0 (es) | Un procedimiento para la preparacion de nuevas espiro-3-heteroazolidindionas. | |
| ES542517A0 (es) | Un procedimiento para la preparacion de monoalquil-polial- quilenpoliaminas | |
| ES550207A0 (es) | Procedimiento para la fabricacion de un nuevo derivado de labenzoilfenilurea | |
| ES548147A0 (es) | Un procedimiento para la preparacion de nuevos derivados pe-nem | |
| ES551129A0 (es) | Un procedimiento para la preparacion de nuevas 3-alcoxi-2-(n-pirrolidino)-n-pirimidinil- o n-pirazinil-propilaminas | |
| ES552986A0 (es) | Un procedimiento para la preparacion de piridazinilimidazolidinonas | |
| ES542674A0 (es) | Un procedimiento para la preparacion de compuestos de cefa- losporina | |
| ES551506A0 (es) | Un procedimiento para la preparacion de etanodiimidamidas | |
| ES530871A0 (es) | Un nuevo procedimiento para la preparacion de 1-aril-2-(4-diarilmetilpiperazin-1-il)etanonas |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 20051003 |