HUE054832T2 - Pirido-imidazo rifamicinszármazékok baktériumellenes szerként - Google Patents

Pirido-imidazo rifamicinszármazékok baktériumellenes szerként

Info

Publication number
HUE054832T2
HUE054832T2 HUE18755539A HUE18755539A HUE054832T2 HU E054832 T2 HUE054832 T2 HU E054832T2 HU E18755539 A HUE18755539 A HU E18755539A HU E18755539 A HUE18755539 A HU E18755539A HU E054832 T2 HUE054832 T2 HU E054832T2
Authority
HU
Hungary
Prior art keywords
pyrido
antibacterial agent
rifamycin derivatives
imidazo rifamycin
imidazo
Prior art date
Application number
HUE18755539A
Other languages
English (en)
Inventor
Egidio Marchi
Sacchetti Alessandro Lapini
Claudia Ori
Lisa Preti
Original Assignee
Biofer Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IT102017000091912A external-priority patent/IT201700091912A1/it
Application filed by Biofer Spa filed Critical Biofer Spa
Publication of HUE054832T2 publication Critical patent/HUE054832T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HUE18755539A 2017-06-26 2018-06-25 Pirido-imidazo rifamicinszármazékok baktériumellenes szerként HUE054832T2 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP17177894 2017-06-26
IT102017000091912A IT201700091912A1 (it) 2017-08-08 2017-08-08 Nuove pirido-imidazo rifamicine

Publications (1)

Publication Number Publication Date
HUE054832T2 true HUE054832T2 (hu) 2021-10-28

Family

ID=64742822

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE18755539A HUE054832T2 (hu) 2017-06-26 2018-06-25 Pirido-imidazo rifamicinszármazékok baktériumellenes szerként

Country Status (10)

Country Link
US (2) US11028086B2 (hu)
EP (1) EP3645539B1 (hu)
CN (1) CN110770244A (hu)
DK (1) DK3645539T3 (hu)
ES (1) ES2868180T3 (hu)
HU (1) HUE054832T2 (hu)
MX (1) MX2019015681A (hu)
PL (1) PL3645539T3 (hu)
RU (1) RU2020102511A (hu)
WO (1) WO2019003076A1 (hu)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1698630E (pt) 2005-03-03 2014-09-15 Alfa Wassermann Spa Novas formas polimorfas de rifaximina, processos para a sua produção e a sua utilização nas preparações medicinais
DK3645539T3 (da) 2017-06-26 2021-05-10 Biofer Spa Pyrido-imidazo-rifamycin-derivater som antibakterielt middel
WO2024076693A1 (en) * 2022-10-05 2024-04-11 Regents Of The University Of Minnesota Rifamycins for nontuberculous mycobacteria

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1090759B (it) 1977-11-29 1985-06-26 Alfa Farmaceutici Spa Procedimento per la preparazione di 3 iodio e 3 bromo rifamicina s
IT1154655B (it) * 1980-05-22 1987-01-21 Alfa Farmaceutici Spa Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica
IT1199374B (it) * 1984-05-15 1988-12-30 Alfa Farmaceutici Spa Processo per la preparazione di pirido-imidazo-rifamicine
ITMI20032144A1 (it) 2003-11-07 2005-05-08 Alfa Wassermann Spa Forme polimorfe di rifaximina, processi per ottenerle e
US7250413B2 (en) * 2004-04-26 2007-07-31 Cumbre Pharmaceuticals Inc. C-25 carbamate rifamycin derivatives with activity against drug-resistant microbes
PT1698630E (pt) 2005-03-03 2014-09-15 Alfa Wassermann Spa Novas formas polimorfas de rifaximina, processos para a sua produção e a sua utilização nas preparações medicinais
WO2007096703A2 (en) * 2005-08-11 2007-08-30 Targanta Therapeutics Inc. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
IT1397617B1 (it) * 2009-04-20 2013-01-18 Alfa Wassermann Spa Nuovi derivati della rifamicina
UA120030C2 (uk) * 2012-08-13 2019-09-25 Адіфарм Еад Фармацевтичні склади, які містять 3-(4-цинаміл-1-піперазиніл)амінопохідні 3-формілрифаміцину s та їх застосування
DK3645539T3 (da) 2017-06-26 2021-05-10 Biofer Spa Pyrido-imidazo-rifamycin-derivater som antibakterielt middel

Also Published As

Publication number Publication date
US11028086B2 (en) 2021-06-08
DK3645539T3 (da) 2021-05-10
RU2020102511A (ru) 2021-07-27
EP3645539B1 (en) 2021-04-07
PL3645539T3 (pl) 2021-10-25
ES2868180T3 (es) 2021-10-21
US20210363143A1 (en) 2021-11-25
WO2019003076A1 (en) 2019-01-03
EP3645539A1 (en) 2020-05-06
US20200157104A1 (en) 2020-05-21
CN110770244A (zh) 2020-02-07
RU2020102511A3 (hu) 2021-07-27
MX2019015681A (es) 2020-02-26

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