ES476755A1 - Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas. - Google Patents

Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas.

Info

Publication number
ES476755A1
ES476755A1 ES476755A ES476755A ES476755A1 ES 476755 A1 ES476755 A1 ES 476755A1 ES 476755 A ES476755 A ES 476755A ES 476755 A ES476755 A ES 476755A ES 476755 A1 ES476755 A1 ES 476755A1
Authority
ES
Spain
Prior art keywords
amino
orthoanisamides
preparing
methods
application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES476755A
Other languages
English (en)
Spanish (es)
Original Assignee
Ile De France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ile De France filed Critical Ile De France
Publication of ES476755A1 publication Critical patent/ES476755A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
ES476755A 1978-01-20 1979-01-11 Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas. Expired ES476755A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7801632A FR2415099A1 (fr) 1978-01-20 1978-01-20 Nouveaux derives de 4-amino-5-alkylsulfonyl ortho-anisamides, leurs procedes de preparation et leur application comme psychotropes

Publications (1)

Publication Number Publication Date
ES476755A1 true ES476755A1 (es) 1979-06-01

Family

ID=9203689

Family Applications (2)

Application Number Title Priority Date Filing Date
ES476755A Expired ES476755A1 (es) 1978-01-20 1979-01-11 Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas.
ES477782A Expired ES477782A1 (es) 1978-01-20 1979-02-16 Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES477782A Expired ES477782A1 (es) 1978-01-20 1979-02-16 Procedimiento de preparacion de nuevos derivados de 4-amino-5-alcohilsulfonil-orto-anisamidas.

Country Status (42)

Country Link
US (2) US4294828A (OSRAM)
JP (1) JPS6049192B2 (OSRAM)
AR (2) AR221354A1 (OSRAM)
AT (1) AT377977B (OSRAM)
AU (1) AU528561B2 (OSRAM)
BE (1) BE872585A (OSRAM)
BG (2) BG31496A3 (OSRAM)
CA (1) CA1101430A (OSRAM)
CH (1) CH637927A5 (OSRAM)
CS (1) CS226181B2 (OSRAM)
CY (1) CY1201A (OSRAM)
DD (1) DD141520A5 (OSRAM)
DE (1) DE2901181C2 (OSRAM)
DK (1) DK158346C (OSRAM)
EG (1) EG14045A (OSRAM)
ES (2) ES476755A1 (OSRAM)
FI (1) FI71126C (OSRAM)
FR (1) FR2415099A1 (OSRAM)
GB (2) GB2012765B (OSRAM)
GR (1) GR64431B (OSRAM)
HK (1) HK12184A (OSRAM)
HU (1) HU179793B (OSRAM)
IE (1) IE47798B1 (OSRAM)
IL (1) IL56411A (OSRAM)
IN (1) IN150226B (OSRAM)
IT (1) IT1164655B (OSRAM)
LU (1) LU80786A1 (OSRAM)
MC (1) MC1232A1 (OSRAM)
MX (2) MX5793E (OSRAM)
NL (1) NL191707C (OSRAM)
NO (1) NO151320C (OSRAM)
NZ (1) NZ189378A (OSRAM)
OA (1) OA06156A (OSRAM)
PH (2) PH15725A (OSRAM)
PL (2) PL116532B1 (OSRAM)
PT (1) PT69068A (OSRAM)
RO (2) RO80311A (OSRAM)
SE (2) SE448874B (OSRAM)
SU (1) SU820659A3 (OSRAM)
YU (2) YU42172B (OSRAM)
ZA (1) ZA79219B (OSRAM)
ZM (1) ZM579A1 (OSRAM)

Families Citing this family (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2440946A2 (fr) * 1978-01-20 1980-06-06 Ile De France Nouveaux benzamides heterocycliques substitues, leurs procedes de preparation et leur application comme modificateurs du comportement
ZA818221B (en) * 1980-12-12 1982-10-27 Beecham Group Plc Pharmaceutical compounds
FR2550447B1 (fr) * 1983-08-10 1986-01-17 Ile De France Application du n-(ally-2-pyrrolidinylmethyl) 2-methoxy 4-amino 5-methylsulfamoyl benzamide comme antiagregant plaquettaire
FR2574795B1 (fr) * 1984-12-18 1987-11-20 Ile De France Nouveau procede industriel de synthese du n-((1'-allyl 2'-pyrrolidinyl) methyl) 2-methoxy 4,5-azimido benzamide
FR2584401B1 (fr) * 1985-07-04 1987-11-20 Ile De France Nouveau benzamide, son procede de preparation et son application dans le domaine therapeutique
US5227388A (en) * 1989-12-26 1993-07-13 Hoechst-Roussel Pharmaceuticals Incorporated Thienobenzoxepins and naphthothiophenes
US5260319A (en) * 1989-12-26 1993-11-09 Hoechst-Roussel Pharmaceuticals Incorporated Thienobenzoxepins and naphthothiophenes
FR2678266A1 (fr) * 1991-06-28 1992-12-31 Delagrange Laboratoires Nouveaux derives de 2-hydroxy 4-amino 5-ethylsulfonyl benzamide utiles comme anxiolytiques.
FR2699533A1 (fr) * 1992-12-21 1994-06-24 Mouhtaram Mohamed Dérivés de N-((1,4-dialkyl-6-arylpipérazine-2-yl)méthyl)benzamides. (Isomères cis et trans) Propriétés pharmacologiques et applications.
FR2753376B1 (fr) * 1996-09-18 1998-10-16 Synthelabo Compositions pharmaceutiques comprenant de l'amisulpride et leurs applications therapeutiques
FR2762213B1 (fr) * 1997-04-18 1999-05-14 Synthelabo Composition pharmaceutique a retention gastrique
US6169094B1 (en) * 1998-07-14 2001-01-02 Sanofi-Synthelabo Compositions of (S) (-)-amisulpride
ATE445838T1 (de) 2001-07-25 2009-10-15 Raptor Pharmaceutical Inc Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke
JP2006528676A (ja) * 2003-05-16 2006-12-21 ファイザー・プロダクツ・インク 非定形型抗精神病薬と、ｇａｂａ調節薬及び／又は抗痙攣薬の治療上の組合せ
FR2857263B1 (fr) * 2003-07-09 2005-09-09 Sanofi Synthelabo Nouvelle composition pharmaceutique solide comprenant de l'amisulpride
BRPI0510942A (pt) * 2004-05-11 2007-07-17 Pfizer Prod Inc combinação de antipsicóticos atìpicos e antagonistas do receptor 5-ht1b
WO2006116221A2 (en) * 2005-04-22 2006-11-02 Wyeth Therapeutic combinations for the treatment or prevention of psychotic disorders
CN101287411B (zh) 2005-04-28 2013-03-06 普罗秋斯生物医学公司 药物信息系统及其用途
KR20090071598A (ko) 2006-09-18 2009-07-01 랩터 파마슈티컬 인코포레이티드 수용체 결합 단백질(ｒａｐ)-접합체 투여에 의한 간 질환의 치료
US7825156B2 (en) * 2007-02-02 2010-11-02 Copharms Method of treating bipolar depression with a benzamide derivative
WO2009156889A1 (en) * 2008-06-25 2009-12-30 Pfizer Inc. Diaryl compounds and uses thereof
US20100105755A1 (en) * 2008-09-12 2010-04-29 Auspex Pharmaceuticals, Inc. Substituted benzamide modulators of dopamine receptor
NZ594310A (en) 2009-02-20 2014-02-28 To Bbb Holding B V Glutathione-based drug delivery system
TWI556839B (zh) 2009-05-06 2016-11-11 研究室護膚股份有限公司 包含活性劑－磷酸鈣粒子複合物之皮膚遞送組成物及其使用方法
CN101898991B (zh) * 2009-05-31 2013-09-25 江苏天士力帝益药业有限公司 一种(s)(-)-氨磺必利d-(-)-酒石酸盐的合成方法
CN101628886B (zh) * 2009-08-25 2012-12-12 北京紫萌同达科技有限公司 一种2-甲氧基-4-氨基-5-乙砜基苯甲酸的合成方法
AU2016216578B2 (en) * 2010-03-11 2017-11-23 Acacia Pharma Limited The use of amisulpride as an anti-emetic
GB201004020D0 (en) 2010-03-11 2010-04-21 Acacia Pharma Ltd New therapeutic use
AU2014202535B2 (en) * 2010-03-11 2016-05-26 Acacia Pharma Limited The use of amisulpride as an anti-emetic
BR112012031959A2 (pt) 2010-06-17 2015-09-22 Lupin Ltd um processo aperfeiçoado para preparação de amisulpride
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
CN103319384A (zh) * 2013-06-18 2013-09-25 苏州诚和医药化学有限公司 制备2-甲氧基-4-氨基-5-乙砜基苯甲酸的方法
CN103304453A (zh) * 2013-06-18 2013-09-18 苏州诚和医药化学有限公司 两步法合成2-甲氧基-4-氨基-5-乙砜基苯甲酸
CN103450058B (zh) * 2013-09-18 2015-10-14 广安凯特医药化工有限公司 一种氨磺必利酸的制备方法
CN104725292B (zh) * 2015-03-23 2017-07-25 湖北荆江源制药股份有限公司 一种(s)(‑)‑氨磺必利的制备方法
GB201618425D0 (en) * 2016-11-01 2016-12-14 Acacia Pharma Ltd method
ES2908949T3 (es) * 2016-11-28 2022-05-04 Lb Pharmaceuticals Inc Agentes psicotrópicos y sus usos
US11377421B2 (en) 2016-11-28 2022-07-05 Lb Pharmaceuticals Inc. Psychotropic agents and uses thereof
CN106995397B (zh) * 2016-12-12 2020-01-14 河北医科大学 R-氨磺必利药用盐、制备方法、晶型及其用途
GB201702250D0 (en) 2017-02-10 2017-03-29 Acacia Pharma Ltd Method
CA3088356A1 (en) 2017-12-05 2019-06-13 Sunovion Pharmaceuticals Inc. Crystal forms and production methods thereof
KR20200110648A (ko) 2017-12-05 2020-09-24 선오비온 파마슈티컬스 인코포레이티드 비라세믹 혼합물 및 이의 용도
CN110790693A (zh) * 2018-08-02 2020-02-14 北京万全德众医药生物技术有限公司 一种(s)(-)-氨磺必利的制备方法
MX2021014774A (es) 2019-06-04 2022-02-03 Sunovion Pharmaceuticals Inc Formulaciones de liberacion modificada y usos de las mismas.
USD1047552S1 (en) * 2021-04-23 2024-10-22 Krueger International, Inc. Furniture leg with frame
CN116003304A (zh) * 2023-02-08 2023-04-25 浙江皓华制药有限公司 一种氨磺必利的合成方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
FR2313935A1 (fr) * 1975-06-10 1977-01-07 Ile De France Nouveaux benzamides substitues, leurs derives et leur procede de preparation
US3862139A (en) * 1972-06-23 1975-01-21 Delmar Chem Heterocyclic benzamide compounds
FR2244760B1 (OSRAM) * 1973-09-25 1980-06-27 Ile De France
FR2299862B1 (en) * 1975-02-07 1978-07-21 Soc Et Scient Et Ind Substd. N-(1-benzylpyrrolidinyl-2-alkyl)benzamides - used as antiemetics, anti-ulcer agents and CNS active
FR2294698A1 (fr) * 1974-12-18 1976-07-16 Synthelabo Nouveaux derives des methoxy-2 benzamides substitues, leurs sels, leur preparation et les medicaments qui en renferment
SE412908B (sv) * 1974-12-18 1980-03-24 Synthelabo Forfarande for framstellning av terapeutiskt aktiva 2-metoxibensamider innehallande en pyrrolidin- eller en piperidinrest

Also Published As

Publication number Publication date
YU42172B (en) 1988-06-30
NL191707C (nl) 1996-04-02
SE460968B (sv) 1989-12-11
FR2415099A1 (fr) 1979-08-17
US4401822A (en) 1983-08-30
FI790182A7 (fi) 1979-07-21
NO151320B (no) 1984-12-10
DE2901181C2 (de) 1984-07-19
CA1101430A (en) 1981-05-19
YU25483A (en) 1983-10-31
CH637927A5 (fr) 1983-08-31
SE448874B (sv) 1987-03-23
GB2083458B (en) 1983-03-09
SE8603773L (sv) 1986-09-09
IL56411A (en) 1982-09-30
JPS54145658A (en) 1979-11-14
ATA39879A (de) 1983-12-15
BE872585A (fr) 1979-06-07
NL7900457A (nl) 1979-07-24
PL118151B1 (en) 1981-09-30
EG14045A (en) 1983-09-30
DK20979A (da) 1979-07-21
GB2083458A (en) 1982-03-24
JPS6049192B2 (ja) 1985-10-31
IN150226B (OSRAM) 1982-08-21
DK158346C (da) 1990-10-08
YU5079A (en) 1983-06-30
RO80311A (ro) 1982-12-06
NO151320C (no) 1985-04-17
IE790092L (en) 1979-07-20
DD141520A5 (de) 1980-05-07
BG31496A3 (bg) 1982-01-15
GB2012765A (en) 1979-08-01
HK12184A (en) 1984-02-24
NL191707B (nl) 1995-12-01
PH15725A (en) 1983-03-18
AU528561B2 (en) 1983-05-05
GR64431B (en) 1980-03-21
MX5793E (es) 1984-07-19
SE8603773D0 (sv) 1986-09-09
LU80786A1 (fr) 1979-09-07
HU179793B (en) 1982-12-28
DE2901181A1 (de) 1979-07-26
NO790180L (no) 1979-07-23
MC1232A1 (fr) 1979-10-26
AR220574A1 (es) 1980-11-14
ZM579A1 (en) 1979-12-21
US4294828A (en) 1981-10-13
CY1201A (en) 1983-12-31
PT69068A (fr) 1979-02-01
DK158346B (da) 1990-05-07
NZ189378A (en) 1983-03-15
PL116532B1 (en) 1981-06-30
IT1164655B (it) 1987-04-15
SU820659A3 (ru) 1981-04-07
ES477782A1 (es) 1979-09-16
AU4337379A (en) 1979-07-26
BG31497A3 (bg) 1982-01-15
ZA79219B (en) 1980-01-30
OA06156A (fr) 1981-06-30
FR2415099B1 (OSRAM) 1981-02-20
PL212899A1 (OSRAM) 1980-01-14
PH22287A (en) 1988-07-22
IE47798B1 (en) 1984-06-27
AR221354A1 (es) 1981-01-30
SE7900380L (sv) 1979-07-21
AT377977B (de) 1985-05-28
IT7947706A0 (it) 1979-01-18
YU41278B (en) 1986-12-31
FI71126C (fi) 1986-11-24
CS226181B2 (en) 1984-03-19
RO76393A (ro) 1981-03-30
MX7623E (es) 1990-03-27
IL56411A0 (en) 1979-03-12
FI71126B (fi) 1986-08-14
GB2012765B (en) 1982-09-08

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