ES439690A1 - Procedimiento para preparar derivados de quinazolina. - Google Patents

Procedimiento para preparar derivados de quinazolina.

Info

Publication number
ES439690A1
ES439690A1 ES439690A ES439690A ES439690A1 ES 439690 A1 ES439690 A1 ES 439690A1 ES 439690 A ES439690 A ES 439690A ES 439690 A ES439690 A ES 439690A ES 439690 A1 ES439690 A1 ES 439690A1
Authority
ES
Spain
Prior art keywords
group
formula
see formula
aryl
hydrogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES439690A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp
Original Assignee
Pfizer Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp filed Critical Pfizer Corp
Publication of ES439690A1 publication Critical patent/ES439690A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES439690A 1974-07-25 1975-07-24 Procedimiento para preparar derivados de quinazolina. Expired ES439690A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3280574 1974-07-25

Publications (1)

Publication Number Publication Date
ES439690A1 true ES439690A1 (es) 1977-07-01

Family

ID=10344259

Family Applications (4)

Application Number Title Priority Date Filing Date
ES439690A Expired ES439690A1 (es) 1974-07-25 1975-07-24 Procedimiento para preparar derivados de quinazolina.
ES455985A Expired ES455985A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.
ES455984A Expired ES455984A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.
ES455986A Expired ES455986A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.

Family Applications After (3)

Application Number Title Priority Date Filing Date
ES455985A Expired ES455985A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.
ES455984A Expired ES455984A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.
ES455986A Expired ES455986A1 (es) 1974-07-25 1977-02-16 Procedimiento para preparar derivados de quinazolina.

Country Status (7)

Country Link
AT (1) AT344178B (de)
BE (1) BE831654A (de)
CS (1) CS192549B2 (de)
ES (4) ES439690A1 (de)
HU (1) HU174961B (de)
PL (6) PL103798B1 (de)
SU (5) SU578874A3 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070004763A1 (en) * 2005-06-10 2007-01-04 Nand Baindur Aminoquinoline and aminoquinazoline kinase modulators

Also Published As

Publication number Publication date
SU625606A3 (ru) 1978-09-25
PL193420A1 (pl) 1978-04-24
PL193423A1 (pl) 1978-04-24
AT344178B (de) 1978-07-10
ATA525275A (de) 1977-11-15
PL103791B1 (pl) 1979-07-31
PL103798B1 (pl) 1979-07-31
ES455985A1 (es) 1978-06-16
HU174961B (hu) 1980-04-28
PL193422A1 (pl) 1978-06-05
PL193419A1 (pl) 1978-04-24
PL103789B1 (pl) 1979-07-31
PL193421A1 (pl) 1978-04-24
ES455986A1 (es) 1978-06-01
SU578874A3 (ru) 1977-10-30
SU634671A3 (ru) 1978-11-25
PL99427B1 (pl) 1978-07-31
PL104615B1 (pl) 1979-08-31
CS192549B2 (en) 1979-08-31
BE831654A (fr) 1976-01-23
SU858563A3 (ru) 1981-08-23
ES455984A1 (es) 1978-06-01
SU613723A3 (ru) 1978-06-30
PL103797B1 (pl) 1979-07-31

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