ES2951809T3 - Derivados de quinazolina-pirazol para el tratamiento de trastornos relacionados con el cáncer - Google Patents
Derivados de quinazolina-pirazol para el tratamiento de trastornos relacionados con el cáncer Download PDFInfo
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- ES2951809T3 ES2951809T3 ES18803171T ES18803171T ES2951809T3 ES 2951809 T3 ES2951809 T3 ES 2951809T3 ES 18803171 T ES18803171 T ES 18803171T ES 18803171 T ES18803171 T ES 18803171T ES 2951809 T3 ES2951809 T3 ES 2951809T3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US201762507540P | 2017-05-17 | 2017-05-17 | |
| PCT/US2018/032868 WO2018213377A1 (en) | 2017-05-17 | 2018-05-16 | Quinazoline-pyrazole derivatives for the treatment of cancer-related disorders |
Publications (1)
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| ES2951809T3 true ES2951809T3 (es) | 2023-10-25 |
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| ES (1) | ES2951809T3 (enExample) |
| PL (1) | PL3634417T3 (enExample) |
| WO (1) | WO2018213377A1 (enExample) |
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| EP3947463A4 (en) | 2019-03-29 | 2022-12-21 | Arcus Biosciences, Inc. | TREATMENT OF CANCER USING AN IDENTIFIED ADENOSINE FINGERPRINT |
| IL295569B1 (en) | 2020-03-19 | 2026-04-01 | Arcus Biosciences Inc | Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2ALPHA |
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| CN112326961B (zh) * | 2020-10-30 | 2021-08-06 | 福州迈新生物技术开发有限公司 | 一种非小细胞肺癌中pd-l1阳性肿瘤细胞比例的分析方法和存储设备 |
| CN112691107B (zh) * | 2021-02-03 | 2022-09-02 | 北京斯利安药业有限公司 | 一种药物组合物及其应用 |
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| CN113642386B (zh) * | 2021-07-02 | 2024-06-21 | 广州金域医学检验中心有限公司 | 基于深度学习评价鼻咽癌治疗效果的方法、装置、设备和介质 |
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| US20240425497A1 (en) | 2023-05-05 | 2024-12-26 | Arcus Biosciences, Inc. | Cbl-b Inhibitors and Methods of Use Thereof |
| WO2024243502A1 (en) | 2023-05-25 | 2024-11-28 | Arcus Biosciences, Inc. | Cbl-b inhibitors and methods of use thereof |
| CN119139469A (zh) * | 2023-06-16 | 2024-12-17 | 武汉大学 | 腺苷受体抑制剂在制备用于治疗高脂血症与心脑血管疾病的药物中的应用 |
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| TW202523302A (zh) | 2023-11-02 | 2025-06-16 | 美商阿克思生物科學有限公司 | 噻唑化合物及其使用方法 |
| WO2026006759A1 (en) | 2024-06-28 | 2026-01-02 | Arcus Biosciences, Inc. | Pharmaceutical compositions, dosage forms, and methods of making and using same |
| WO2026035034A1 (ko) * | 2024-08-06 | 2026-02-12 | 주식회사 대웅제약 | 신규한 퀴나졸린 유도체 및 이를 포함하는 약학 조성물 |
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| EP3634417B1 (en) | 2023-07-12 |
| EP3634417C0 (en) | 2023-07-12 |
| PL3634417T3 (pl) | 2023-09-25 |
| EP3634417A1 (en) | 2020-04-15 |
| US20210214346A1 (en) | 2021-07-15 |
| EP3634417A4 (en) | 2021-01-13 |
| JP7189155B2 (ja) | 2022-12-13 |
| US11220492B2 (en) | 2022-01-11 |
| CN110636846A (zh) | 2019-12-31 |
| JP2020519664A (ja) | 2020-07-02 |
| CN110636846B (zh) | 2023-05-16 |
| WO2018213377A1 (en) | 2018-11-22 |
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