ES2435997T3 - Aminopirimidinas útiles como inhibidores de las proteínas cinasas - Google Patents
Aminopirimidinas útiles como inhibidores de las proteínas cinasas Download PDFInfo
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- ES2435997T3 ES2435997T3 ES08731830T ES08731830T ES2435997T3 ES 2435997 T3 ES2435997 T3 ES 2435997T3 ES 08731830 T ES08731830 T ES 08731830T ES 08731830 T ES08731830 T ES 08731830T ES 2435997 T3 ES2435997 T3 ES 2435997T3
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- A61P31/12—Antivirals
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US90608607P | 2007-03-09 | 2007-03-09 | |
| US906086P | 2007-03-09 | ||
| US95302007P | 2007-07-31 | 2007-07-31 | |
| US953020P | 2007-07-31 | ||
| PCT/US2008/056423 WO2008112642A1 (en) | 2007-03-09 | 2008-03-10 | Aminopyrimidines useful as inhibitors of protein kinases |
Publications (1)
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| ES2435997T3 true ES2435997T3 (es) | 2013-12-26 |
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| ES08731830T Active ES2435997T3 (es) | 2007-03-09 | 2008-03-10 | Aminopirimidinas útiles como inhibidores de las proteínas cinasas |
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| EP (1) | EP2134707B1 (OSRAM) |
| JP (1) | JP5520057B2 (OSRAM) |
| CN (1) | CN101663295B (OSRAM) |
| AU (2) | AU2008226457B2 (OSRAM) |
| CA (1) | CA2679884A1 (OSRAM) |
| ES (1) | ES2435997T3 (OSRAM) |
| MX (1) | MX2009009590A (OSRAM) |
| NZ (1) | NZ579446A (OSRAM) |
| WO (1) | WO2008112642A1 (OSRAM) |
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| CN101801959A (zh) | 2007-05-02 | 2010-08-11 | 沃泰克斯药物股份有限公司 | 可用作激酶抑制剂的氨基嘧啶类化合物 |
| CN101687852A (zh) | 2007-05-24 | 2010-03-31 | 沃泰克斯药物股份有限公司 | 可用作激酶抑制剂的噻唑类和吡唑类化合物 |
| JP5553751B2 (ja) * | 2007-07-31 | 2014-07-16 | バーテックス ファーマシューティカルズ インコーポレイテッド | ５−フルオロ−１Ｈ−ピラゾロ［３，４−ｂ］ピリジン−３−アミンおよびその誘導体を調製するためのプロセス |
| EP2821400B1 (en) | 2009-03-20 | 2017-09-27 | Vertex Pharmaceuticals Incorporated | Process for making modulators of cystic fibrosis transmembrane conductance regulator |
-
2008
- 2008-03-10 WO PCT/US2008/056423 patent/WO2008112642A1/en not_active Ceased
- 2008-03-10 MX MX2009009590A patent/MX2009009590A/es active IP Right Grant
- 2008-03-10 AU AU2008226457A patent/AU2008226457B2/en not_active Ceased
- 2008-03-10 NZ NZ579446A patent/NZ579446A/en not_active IP Right Cessation
- 2008-03-10 ES ES08731830T patent/ES2435997T3/es active Active
- 2008-03-10 CA CA002679884A patent/CA2679884A1/en not_active Abandoned
- 2008-03-10 CN CN200880012693.9A patent/CN101663295B/zh not_active Expired - Fee Related
- 2008-03-10 JP JP2009552927A patent/JP5520057B2/ja not_active Expired - Fee Related
- 2008-03-10 EP EP08731830.9A patent/EP2134707B1/en not_active Not-in-force
-
2010
- 2010-06-02 US US12/791,976 patent/US8664219B2/en not_active Expired - Fee Related
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2014
- 2014-01-15 US US14/155,624 patent/US20140194444A1/en not_active Abandoned
- 2014-06-18 AU AU2014203289A patent/AU2014203289A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US8664219B2 (en) | 2014-03-04 |
| EP2134707A1 (en) | 2009-12-23 |
| AU2008226457A1 (en) | 2008-09-18 |
| CA2679884A1 (en) | 2008-09-18 |
| CN101663295A (zh) | 2010-03-03 |
| AU2014203289A1 (en) | 2014-07-17 |
| US20140194444A1 (en) | 2014-07-10 |
| EP2134707B1 (en) | 2013-09-11 |
| AU2008226457B2 (en) | 2014-03-20 |
| CN101663295B (zh) | 2014-11-05 |
| MX2009009590A (es) | 2009-11-10 |
| WO2008112642A1 (en) | 2008-09-18 |
| JP2010520886A (ja) | 2010-06-17 |
| NZ579446A (en) | 2012-02-24 |
| US20110020376A1 (en) | 2011-01-27 |
| JP5520057B2 (ja) | 2014-06-11 |
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