ES2316758T3 - Uso de aglutinantes del receptor edg en el cancer. - Google Patents
Uso de aglutinantes del receptor edg en el cancer. Download PDFInfo
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- ES2316758T3 ES2316758T3 ES03730049T ES03730049T ES2316758T3 ES 2316758 T3 ES2316758 T3 ES 2316758T3 ES 03730049 T ES03730049 T ES 03730049T ES 03730049 T ES03730049 T ES 03730049T ES 2316758 T3 ES2316758 T3 ES 2316758T3
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- alkyl
- inhibitor
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- halogen
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- A61P35/04—Antineoplastic agents specific for metastasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0211261 | 2002-05-16 | ||
| GB0211261A GB0211261D0 (en) | 2002-05-16 | 2002-05-16 | Organic compounds |
| US39041102P | 2002-06-20 | 2002-06-20 | |
| US390411P | 2002-06-20 | ||
| GB0217150A GB0217150D0 (en) | 2002-07-24 | 2002-07-24 | Organic compounds |
| GB0217150 | 2002-07-24 | ||
| US44973903P | 2003-02-24 | 2003-02-24 | |
| US449739P | 2003-02-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2316758T3 true ES2316758T3 (es) | 2009-04-16 |
Family
ID=29554311
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES03730049T Expired - Lifetime ES2316758T3 (es) | 2002-05-16 | 2003-05-15 | Uso de aglutinantes del receptor edg en el cancer. |
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| JP (3) | JP5227492B2 (enExample) |
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| CN (1) | CN1652757B (enExample) |
| AT (1) | ATE412408T1 (enExample) |
| AU (1) | AU2003240655B2 (enExample) |
| BR (1) | BR0311173A (enExample) |
| CA (1) | CA2483594C (enExample) |
| CY (1) | CY1108719T1 (enExample) |
| DE (1) | DE60324416D1 (enExample) |
| DK (1) | DK1505959T3 (enExample) |
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| IL (3) | IL164838A (enExample) |
| MX (1) | MXPA04011384A (enExample) |
| NO (2) | NO334074B1 (enExample) |
| NZ (2) | NZ536513A (enExample) |
| PL (1) | PL372103A1 (enExample) |
| PT (1) | PT1505959E (enExample) |
| SI (1) | SI1505959T1 (enExample) |
| WO (1) | WO2003097028A1 (enExample) |
| ZA (1) | ZA200408575B (enExample) |
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| ITRM20010688A1 (it) | 2001-11-21 | 2003-05-21 | Univ Roma | Composti immunoregolatori. |
| KR100836547B1 (ko) | 2002-01-11 | 2008-06-10 | 상꾜 가부시키가이샤 | 아미노 알코올 유도체 또는 포스폰산 유도체 및 이들을함유하는 의약 조성물 |
| WO2003104442A1 (en) * | 2002-06-07 | 2003-12-18 | Es Cell International Pte Ltd | Methods of regulating differentiation in stem cells |
| EP1602660B1 (en) * | 2003-02-18 | 2011-04-06 | Kyorin Pharmaceutical Co., Ltd. | Aminophosphonic acid derivatives, addition salts thereof and s1p receptor modulators |
| GB0500020D0 (en) * | 2005-01-04 | 2005-02-09 | Novartis Ag | Organic compounds |
| NZ549162A (en) | 2004-02-24 | 2009-12-24 | Sankyo Co | Amino-pyrrol alcohol compounds |
| US7794713B2 (en) | 2004-04-07 | 2010-09-14 | Lpath, Inc. | Compositions and methods for the treatment and prevention of hyperproliferative diseases |
| WO2006013948A1 (ja) * | 2004-08-04 | 2006-02-09 | Taisho Pharmaceutical Co., Ltd. | トリアゾール誘導体 |
| EP1781595A1 (en) | 2004-08-13 | 2007-05-09 | Praecis Pharmaceuticals Inc. | Methods and compositions for modulating sphingosine-1-phosphate (s1p) receptor activity |
| SI1812797T1 (sl) * | 2004-10-28 | 2013-06-28 | Lpath, Inc. | Pripravki in metode zdravljenja ter preprečevanja hiperprolifetarivnih bolezni |
| GB0513431D0 (en) | 2005-06-30 | 2005-08-10 | Kherion Technology Ltd | Prophylactic compositions and uses |
| GT200600350A (es) * | 2005-08-09 | 2007-03-28 | Formulaciones líquidas | |
| CN101415691B (zh) | 2006-02-03 | 2011-12-14 | 大正制药株式会社 | 三唑衍生物 |
| JP5218737B2 (ja) | 2006-02-06 | 2013-06-26 | 大正製薬株式会社 | スフィンゴシン−１−リン酸結合阻害物質 |
| CN101460197A (zh) * | 2006-04-06 | 2009-06-17 | 诺瓦提斯公司 | 有机化合物的组合 |
| US7862812B2 (en) | 2006-05-31 | 2011-01-04 | Lpath, Inc. | Methods for decreasing immune response and treating immune conditions |
| GB0612721D0 (en) | 2006-06-27 | 2006-08-09 | Novartis Ag | Organic compounds |
| EP1923058A1 (en) * | 2006-09-26 | 2008-05-21 | Novartis AG | Coated pharmaceutical composition comprising an S1P agonist or modulator |
| WO2008055072A2 (en) * | 2006-10-27 | 2008-05-08 | Lpath, Inc. | Compositions and methods for treating ocular diseases and conditions |
| RU2468009C2 (ru) | 2007-08-01 | 2012-11-27 | Тайсо Фармасьютикал Ко., Лтд. | Ингибитор связывания s1p1 |
| EP2177521A1 (en) | 2008-10-14 | 2010-04-21 | Almirall, S.A. | New 2-Amidothiadiazole Derivatives |
| KR20130109254A (ko) * | 2008-11-11 | 2013-10-07 | 노파르티스 아게 | 핑골리모드 ｈｃｌ의 결정질 형태 |
| EP2358660A2 (en) | 2008-11-11 | 2011-08-24 | Novartis AG | Salts of fingolimod |
| CN105213372A (zh) | 2008-12-22 | 2016-01-06 | 诺华股份有限公司 | S1p受体激动剂的给药方案 |
| PT4098256T (pt) | 2008-12-22 | 2025-04-10 | Novartis Ag | Regime de dosagem para um agonista do recetor de s1p |
| EP2202232A1 (en) | 2008-12-26 | 2010-06-30 | Laboratorios Almirall, S.A. | 1,2,4-oxadiazole derivatives and their therapeutic use |
| EP2210890A1 (en) | 2009-01-19 | 2010-07-28 | Almirall, S.A. | Oxadiazole derivatives as S1P1 receptor agonists |
| KR20120032538A (ko) | 2009-07-24 | 2012-04-05 | 라티오팜 게엠베하 | 핀골리모드 염의 제조 방법 |
| EP2305660A1 (en) | 2009-09-25 | 2011-04-06 | Almirall, S.A. | New thiadiazole derivatives |
| JP2013505983A (ja) | 2009-09-29 | 2013-02-21 | ノバルティス アーゲー | Ｓ１ｐ受容体モジュレーターの投与計画 |
| EP2343287A1 (en) | 2009-12-10 | 2011-07-13 | Almirall, S.A. | New 2-aminothiadiazole derivatives |
| EP2366702A1 (en) | 2010-03-18 | 2011-09-21 | Almirall, S.A. | New oxadiazole derivatives |
| EP2390252A1 (en) | 2010-05-19 | 2011-11-30 | Almirall, S.A. | New pyrazole derivatives |
| WO2012071524A1 (en) | 2010-11-24 | 2012-05-31 | Ratiopharm Gmbh | Arylsulfonate salts of fingolimod and processes for preparation thereof |
| FR2968556B1 (fr) | 2010-12-13 | 2013-12-27 | Centre Nat Rech Scient | Inhibiteurs des infections a vih et leurs utilisations |
| UA114283C2 (uk) | 2011-01-07 | 2017-05-25 | Новартіс Аг | Композиції імуносупресантів |
| ES2772258T3 (es) | 2011-02-07 | 2020-07-07 | Biogen Ma Inc | Agentes moduladores de S1P |
| MX2014004813A (es) | 2011-10-21 | 2014-05-20 | Novartis Ag | Regimen de dosificacion para un modulador o agonista del receptor s1p. |
| KR101889131B1 (ko) * | 2011-12-23 | 2018-09-20 | 메이지 세이카 파루마 가부시키가이샤 | 신규 s1p 수용체 조정제 |
| HK1211237A1 (en) | 2012-08-06 | 2016-05-20 | Biogen Ma Inc. | Compounds that are s1p modulating agents and/or atx modulating agents |
| EP2879673B1 (en) | 2012-08-06 | 2018-07-25 | Biogen MA Inc. | 1,5,6-substituted naphthalene derivatives as sphingosine 1 phosphate (S1P) receptor and/or autotaxin (ATX) modulators for treating inflammatory and autoimmune disorders |
| ES2749467T3 (es) | 2012-11-20 | 2020-03-20 | Biogen Ma Inc | Agentes moduladores de S1p y/o ATX |
| US9850206B2 (en) | 2012-11-20 | 2017-12-26 | Biogen Ma Inc. | S1P and/or ATX modulating agents |
| AU2014212465B2 (en) | 2013-01-29 | 2018-07-12 | Biogen Ma Inc. | S1P modulating agents |
| EP2970302A1 (en) | 2013-03-15 | 2016-01-20 | Biogen MA Inc. | S1p and/or atx modulating agents |
| CN103417970A (zh) * | 2013-08-15 | 2013-12-04 | 泰山医学院 | 雌激素上调内皮系统保护分子鞘氨醇1-磷酸的应用 |
| WO2016135644A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
| US11434200B2 (en) | 2017-03-09 | 2022-09-06 | Novartis Ag | Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof |
| EP3443986A1 (en) | 2017-08-17 | 2019-02-20 | AC BioScience | Enhancement of chemotherapy efficiency by sphingosine-1-phosphate |
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2003
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- 2003-05-15 CN CN038111942A patent/CN1652757B/zh not_active Expired - Fee Related
- 2003-05-15 EP EP08152489.4A patent/EP1944026B1/en not_active Expired - Lifetime
- 2003-05-15 NZ NZ560662A patent/NZ560662A/en not_active IP Right Cessation
- 2003-05-15 JP JP2004505027A patent/JP5227492B2/ja not_active Expired - Fee Related
- 2003-05-15 EP EP03730049A patent/EP1505959B1/en not_active Expired - Lifetime
- 2003-05-15 ES ES03730049T patent/ES2316758T3/es not_active Expired - Lifetime
- 2003-05-15 AU AU2003240655A patent/AU2003240655B2/en not_active Ceased
- 2003-05-15 AT AT03730049T patent/ATE412408T1/de active
- 2003-05-15 MX MXPA04011384A patent/MXPA04011384A/es active IP Right Grant
- 2003-05-15 PT PT03730049T patent/PT1505959E/pt unknown
- 2003-05-15 SI SI200331499T patent/SI1505959T1/sl unknown
- 2003-05-15 PL PL03372103A patent/PL372103A1/xx not_active IP Right Cessation
- 2003-05-15 WO PCT/EP2003/005125 patent/WO2003097028A1/en not_active Ceased
- 2003-05-15 BR BR0311173-3A patent/BR0311173A/pt not_active IP Right Cessation
- 2003-05-15 EP EP08152484.5A patent/EP1955696B1/en not_active Expired - Lifetime
- 2003-05-15 DE DE60324416T patent/DE60324416D1/de not_active Expired - Lifetime
- 2003-05-15 CA CA2483594A patent/CA2483594C/en not_active Expired - Fee Related
- 2003-05-15 KR KR1020127025694A patent/KR20120125398A/ko not_active Ceased
- 2003-05-15 DK DK03730049T patent/DK1505959T3/da active
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2004
- 2004-10-22 ZA ZA2004/08575A patent/ZA200408575B/en unknown
- 2004-10-25 IL IL164838A patent/IL164838A/en not_active IP Right Cessation
- 2004-12-03 NO NO20045312A patent/NO334074B1/no not_active IP Right Cessation
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2009
- 2009-01-27 CY CY20091100091T patent/CY1108719T1/el unknown
- 2009-04-09 US US12/420,913 patent/US20090209495A1/en not_active Abandoned
- 2009-12-21 JP JP2009289475A patent/JP2010100637A/ja not_active Withdrawn
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2013
- 2013-01-17 NO NO20130106A patent/NO20130106L/no not_active Application Discontinuation
- 2013-01-22 JP JP2013009158A patent/JP2013136584A/ja active Pending
- 2013-11-21 IL IL229559A patent/IL229559A0/en unknown
- 2013-11-21 IL IL229550A patent/IL229550A0/en unknown
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2014
- 2014-06-23 US US14/311,838 patent/US20140303257A1/en not_active Abandoned
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